Synthesis and insecticidal activity of spinosyn analogs functionally altered at the 2'-, 3'- and 4'-positions of the rhamnose moiety

Journal of Antibiotics

Volumn 53, Issue 2, 2000, Pages 171-178

  Creemer, Lawrence C ^a   Kirst, Herbert A ^a   Paschal, Jonathan W ^b   Worden, Thomas V ^c  

^a ELANCO ANIMAL HEALTH   (United States)

^b ELI LILLY AND COMPANY   (United States)

^c DOW AGROSCIENCES LLC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DRUG ANALOG; INSECTICIDE; RHAMNOSE; SPINOSYN A;

ACYLATION; ARTICLE; CONTROLLED STUDY; DRUG OXIDATION; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

EID: 0034054070     PISSN: 00218820     EISSN: None     Source Type: Journal    
DOI: 10.7164/antibiotics.53.171     Document Type: Article

References (8)

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5. TURNER, J. R.; M. L. B. HUBER, M. C. BROUGHTON, J. S. MYNDERSE & J. W. MARTIN: A83543A compounds; factors Q, R, S, and T. U.S. Pat. 5, 767, 253, 1998
6. MYNDERSE, J. S.; M. C. BROUGHTON, W. M. NAKATSUKASA, J. A. MABE, J. R. TURNER, L. C. CREEMER, M. L. B. HUBER, H. A. KIRST & J. W. MARTIN: A83543 compounds and processes for production thereof. U.S. Pat. 5, 840, 861, 1998
7. BOECK, L. D.; E. H. CHIO, T. E. EATON, O. W. Jr. GODFREY, K. H. MICHEL, W. M. NAKATSUKASA & R. C. YAO: Insecticide and miticide A83543 compounds and their method of production by fermentation. U.S. Pat. 5, 496, 931, 1996
8. CREEMER, L. C.; H. A. KIRST & J. W. PASCHAL: Conversion of spinosyn A and spinosyn D to their respective 9-and 17-pseudoaglycones and their aglycones. J. Antibiotics 51: 795, 1998