메뉴 건너뛰기




Volumn 10, Issue 1, 2000, Pages 9-15

Comparison of in vitro cytotoxicity of N-acetyl and N-propionyl derivatives of phenolic thioether amines in melanoma and neuroblastoma cells and the relationship to tyrosinase and tyrosine hydroxylase enzyme activity

Author keywords

Chemotherapy; Melanoma; Tyrosinase; Tyrosine hydroxylase

Indexed keywords

MONOPHENOL MONOOXYGENASE; N PROPIONYL 4 S CYSTEAMINYLPHENOL; N [2 [(4 PROPIONYLOXYPHENYL)THIO]ETHYL]PROPIONAMIDE; PHENOL DERIVATIVE; SULFIDE; TYROSINE 3 MONOOXYGENASE; UNCLASSIFIED DRUG;

EID: 0034050429     PISSN: 09608931     EISSN: None     Source Type: Journal    
DOI: 10.1097/00008390-200010010-00002     Document Type: Article
Times cited : (21)

References (21)
  • 2
    • 0026550080 scopus 로고
    • Effects of tyrosinase activity on the cytotoxicity of 4-S-cysteaminylphenol and N-acetyl-4-S-cysteaminylphenol in melanoma cells
    • 2. Prezioso JA, Epperly MW, Wang N, et al. Effects of tyrosinase activity on the cytotoxicity of 4-S-cysteaminylphenol and N-acetyl-4-S-cysteaminylphenol in melanoma cells. Cancer Lett 1992; 63: 73-79.
    • (1992) Cancer Lett , vol.63 , pp. 73-79
    • Prezioso, J.A.1    Epperly, M.W.2    Wang, N.3
  • 3
    • 0028227817 scopus 로고
    • Selective in vivo accumulation of N-acetyl-4-S-cysteaminylphenol in B16F10 murine melanoma and enhancement of its in vitro and in vivo antimelanoma effect by combination of buthionine sulfoximine
    • 3. Alena F, Iwashina T, Gili A, et al. Selective in vivo accumulation of N-acetyl-4-S-cysteaminylphenol in B16F10 murine melanoma and enhancement of its in vitro and in vivo antimelanoma effect by combination of buthionine sulfoximine. Cancer Res 1994; 54: 2661-2666.
    • (1994) Cancer Res , vol.54 , pp. 2661-2666
    • Alena, F.1    Iwashina, T.2    Gili, A.3
  • 4
    • 0023187868 scopus 로고
    • Selective cytotoxicity of 4-S-cysteaminylphenol on follicular melanocytes of the black mouse: Rational basis for its application to melanoma chemotherapy
    • 4. Ito Y, Jimbow K. Selective cytotoxicity of 4-S-cysteaminylphenol on follicular melanocytes of the black mouse: rational basis for its application to melanoma chemotherapy. Cancer Res 1987; 47: 3278-3284.
    • (1987) Cancer Res , vol.47 , pp. 3278-3284
    • Ito, Y.1    Jimbow, K.2
  • 5
    • 0030722720 scopus 로고    scopus 로고
    • Evidence of the indirect formation of the catecholic intermediate substrate responsible for the autoactivation kinetics of tyrosinase
    • 5. Cooksey CJ, Garratt PJ, Land EJ, Pavel S, Ramsden CA, Riley PA, Smit NP. Evidence of the indirect formation of the catecholic intermediate substrate responsible for the autoactivation kinetics of tyrosinase. J Biol Chem 1997; 272: 26226-26235.
    • (1997) J Biol Chem , vol.272 , pp. 26226-26235
    • Cooksey, C.J.1    Garratt, P.J.2    Land, E.J.3    Pavel, S.4    Ramsden, C.A.5    Riley, P.A.6    Smit, N.P.7
  • 6
    • 0028086396 scopus 로고
    • Recombinant human tyrosinase hydroxylase types 1-4 show regulating kinetic properties for the natural (6R)-tetraydrobiopterin cofactor
    • 6. Nasrin S, Ichinose H, Hidaka H, et al. Recombinant human tyrosinase hydroxylase types 1-4 show regulating kinetic properties for the natural (6R)-tetraydrobiopterin cofactor. J Biochem 1994; 116: 393-398.
    • (1994) J Biochem , vol.116 , pp. 393-398
    • Nasrin, S.1    Ichinose, H.2    Hidaka, H.3
  • 7
    • 0023234953 scopus 로고
    • Synthesis of cysteinylphenol, cysteaminylphenol and related compounds and in vivo evaluation of anti-melanoma effect
    • 7. Miura S, Ueda T, Jimbow K, et al. Synthesis of cysteinylphenol, cysteaminylphenol and related compounds and in vivo evaluation of anti-melanoma effect. Arch Dermatol Res 1987; 279: 219-225.
    • (1987) Arch Dermatol Res , vol.279 , pp. 219-225
    • Miura, S.1    Ueda, T.2    Jimbow, K.3
  • 8
    • 0025339155 scopus 로고
    • Melanocytotoxicity and antimelanoma effects of phenolic amine compounds in mice in vivo
    • 8. Alena F, Jimbow K, Ito S. Melanocytotoxicity and antimelanoma effects of phenolic amine compounds in mice in vivo. Cancer Res 1990; 50: 3743-3747.
    • (1990) Cancer Res , vol.50 , pp. 3743-3747
    • Alena, F.1    Jimbow, K.2    Ito, S.3
  • 9
    • 0028452893 scopus 로고
    • 14C] phenol as a basis for development of antimelanoma and melanoma-radio-imaging agent
    • 14C] phenol as a basis for development of antimelanoma and melanoma-radio-imaging agent. Appl Radiat Isot 1994; 45: 703-705.
    • (1994) Appl Radiat Isot , vol.45 , pp. 703-705
    • Iwashina, T.1    Jimbow, K.2    Wiebe, L.3
  • 10
    • 0028849032 scopus 로고
    • The in vivo melanocytotoxicity and depigmenting potency of N-2,4-acetoxyphenyl thioethyl acetamide in the skin and hair
    • 10. Jimbow M, Marusyk H, Jimbow K. The in vivo melanocytotoxicity and depigmenting potency of N-2,4-acetoxyphenyl thioethyl acetamide in the skin and hair. Br J Dermatol 1995; 133: 526-536.
    • (1995) Br J Dermatol , vol.133 , pp. 526-536
    • Jimbow, M.1    Marusyk, H.2    Jimbow, K.3
  • 11
    • 0032525735 scopus 로고    scopus 로고
    • Synthesis of the melanogenesis-based antimelanoma agent, N-propionyl-4-S-cysteaminylphenol, and screening of depigmenting and anti-tumour effects
    • 11. Tandon M, Thomas PD, Shokravi M, Singh S, Samra S, Chang D, Jimbow K. Synthesis of the melanogenesis-based antimelanoma agent, N-propionyl-4-S-cysteaminylphenol, and screening of depigmenting and anti-tumour effects. Biochem Pharm 1998; 55: 2023-2029.
    • (1998) Biochem Pharm , vol.55 , pp. 2023-2029
    • Tandon, M.1    Thomas, P.D.2    Shokravi, M.3    Singh, S.4    Samra, S.5    Chang, D.6    Jimbow, K.7
  • 12
    • 84965822602 scopus 로고
    • Feasibility of drug screening with panels of human tumor cell lines using a microculture tetrazolium assay
    • 12. Alley MC, Scudlero DA, Monks A, et al. Feasibility of drug screening with panels of human tumor cell lines using a microculture tetrazolium assay. Cancer Res 1988; 48: 589-601.
    • (1988) Cancer Res , vol.48 , pp. 589-601
    • Alley, M.C.1    Scudlero, D.A.2    Monks, A.3
  • 13
    • 0013770081 scopus 로고
    • Tyrosine hydroxylation catalyzed by mammalian tyrosinase: An improved method of assay
    • 13. Pomerantz SH. Tyrosine hydroxylation catalyzed by mammalian tyrosinase: an improved method of assay. Biochem Biophys Res Commun 1964; 16: 188-194.
    • (1964) Biochem Biophys Res Commun , vol.16 , pp. 188-194
    • Pomerantz, S.H.1
  • 15
    • 0017184389 scopus 로고
    • A rapid and sensitive method for the quantitation of microgram quantities of protein using the principle of protein-dye binding
    • 15. Bradford M. A rapid and sensitive method for the quantitation of microgram quantities of protein using the principle of protein-dye binding. Anal Biochem 1976; 72: 248-254.
    • (1976) Anal Biochem , vol.72 , pp. 248-254
    • Bradford, M.1
  • 16
    • 0031692129 scopus 로고    scopus 로고
    • N-propionyl-4-S-cysteaminylphenol exerts selective melanocytotoxicity through apoptotic process
    • 16. Minamitsuji Y, Sugtyama S, Singh S, et al. N-propionyl-4-S-cysteaminylphenol exerts selective melanocytotoxicity through apoptotic process. Sapporo Med J 1998; 67: 23-37.
    • (1998) Sapporo Med J , vol.67 , pp. 23-37
    • Minamitsuji, Y.1    Sugtyama, S.2    Singh, S.3
  • 19
    • 0027414380 scopus 로고
    • Exploitation of pigment biosynthesis pathway as a selective chemotherapeutic approach for malignant melanoma
    • 19. Jimbow K, Iwashina T, Alena F, et al. Exploitation of pigment biosynthesis pathway as a selective chemotherapeutic approach for malignant melanoma. J Invest Dermatol 1993; 100: 231S-238S.
    • (1993) J Invest Dermatol , vol.100
    • Jimbow, K.1    Iwashina, T.2    Alena, F.3
  • 20
    • 0027439861 scopus 로고
    • Mechanism regulating inhibition of thymidylate synthase and growth by gamma-L-glutaminyI-4-hydroxy-3-iodobenzene, a novel melanin precursor, in melanogenic melanoma cells
    • 20. Prezioso JA, Damodaran KM, Wang N, Bloomer WD. Mechanism regulating inhibition of thymidylate synthase and growth by gamma-L-glutaminyI-4-hydroxy-3-iodobenzene, a novel melanin precursor, in melanogenic melanoma cells. Biochem Pharmacol 1993; 45: 473-481.
    • (1993) Biochem Pharmacol , vol.45 , pp. 473-481
    • Prezioso, J.A.1    Damodaran, K.M.2    Wang, N.3    Bloomer, W.D.4
  • 21
    • 0029077703 scopus 로고
    • Glutathione plays a key role in the depigmenting and melanocytotoxic action of N-acetyl-4-S-cysteaminylphenol in black and yellow hair follicles
    • 21. Alena F, Dixon W, Thomas P, et al. Glutathione plays a key role in the depigmenting and melanocytotoxic action of N-acetyl-4-S-cysteaminylphenol in black and yellow hair follicles. J Invest Dermatol 1995; 104: 792-797.
    • (1995) J Invest Dermatol , vol.104 , pp. 792-797
    • Alena, F.1    Dixon, W.2    Thomas, P.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.