2,3-Dihydro-dithiin and -dithiepine-1,1,4,4-tetroxides: Small molecule non-peptide antagonists of the human galanin hGAL-1 receptor

Bioorganic and Medicinal Chemistry

Volumn 8, Issue 6, 2000, Pages 1383-1391

  Scott, Malcolm K ^a   Ross, Tina M ^a   Lee, Daniel H S ^a   Wang, Hoau Yan ^a   Shank, Richard P ^a   Wild, Kenneth D ^a   Davis, Coralie B ^a   Crooke, Jeffrey J ^a   Potocki, Alexander C ^a   Reitz, Allen B ^a  

^a R W JOHNSON PHARMACEUTICAL RES I   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

GALANIN RECEPTOR; RECEPTOR BLOCKING AGENT;

ACETYLCHOLINE RELEASE; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BRAIN SLICE; CELL VIABILITY; CONTROLLED STUDY; DRUG PROTEIN BINDING; GUINEA PIG; HIPPOCAMPUS; IC 50; ILEUM; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ACETYLCHOLINE; AMINO ACID SEQUENCE; ANIMALS; GALANIN; GUINEA PIGS; HIPPOCAMPUS; HUMANS; ILEUM; MALE; MELANOMA; MOLECULAR SEQUENCE DATA; RATS; RECEPTORS, GALANIN; RECEPTORS, NEUROPEPTIDE; STRUCTURE-ACTIVITY RELATIONSHIP; THIEPINS; TUMOR CELLS, CULTURED;

CAVIA PORCELLUS; SUS SCROFA;

EID: 0034048001     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(00)00062-6     Document Type: Article

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