Preparation of remacemide hydrochloride labelled with carbon-14, carbon-13, deuterium and tritium

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 43, Issue 6, 2000, Pages 533-543

  Coombs, M E ^a   Dawson, G E ^a   Fedorchuk, M ^a   Kingston, L P ^a   Lockley, W J S ^a   Mather, A N ^a   McLachlan, T R B ^a   Morlin, A J G ^a   Spink, E ^a   Wilkinson, D J ^a  

^a ASTRAZENECA   (United Kingdom)

Author keywords

3H exchange; Crabtree's catalyst; Friedel Crafts acylation; NMDA receptor; Remacemide; RhCl3; Ritter reaction; 13C(6 )acetophenone

Indexed keywords

AMINO ACIDS; CARBON; CHLORINE COMPOUNDS; KETONES; RHODIUM COMPOUNDS;

3H-EXCHANGE; ACETOPHENONES; CARBON 14; CRABTREE CATALYST; FRIEDEL-CRAFTS ACYLATION; NMDA RECEPTOR; REMACEMIDE; RITTER REACTIONS; [13C(6])ACETOPHENONE; ]+ CATALYST;

TRITIUM;

ACETOPHENONE DERIVATIVE; ACETYL CHLORIDE; ANTICONVULSIVE AGENT; BENZENE; CARBON 13; CARBON 14; DEUTERIUM; GLYCINE; HYDROGEN; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; REMACEMIDE; TRITIUM; UNCLASSIFIED DRUG;

ACYLATION; ARTICLE; CHEMICAL REACTION; CHEMICAL STRUCTURE; CRYSTALLIZATION; DRUG SYNTHESIS; METHODOLOGY; RADIOCHEMISTRY;

TRITIUM;

EID: 0034018981     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(200005)43:6<533::AID-JLCR338>3.0.CO;2-K     Document Type: Article

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