Mucoadhesive liposomes: Physicochemical properties and release behavior of water-soluble drugs from chitosan-coated liposomes

S.T.P. Pharma Sciences

Volumn 10, Issue 1, 2000, Pages 63-68

  Yamamoto, H ^a   Takeuchi, H ^a   Hino, T ^b   Kawashima, Y ^a  

^a GIFU PHARMACEUTICAL UNIVERSITY   (Japan)

^b UNIVERSITY OF TOKUSHIMA   (Japan)

Author keywords

Bioadhesive dosage form; Chitosan; Insulin; Liposome

Indexed keywords

CARBOXYFLUORESCEIN; CHITOSAN; FLUORESCEIN ISOTHIOCYANATE DEXTRAN; INSULIN; LIPOSOME;

ANIMAL EXPERIMENT; ARTICLE; DRUG COATING; DRUG DELIVERY SYSTEM; DRUG DIFFUSION; DRUG RELEASE; MALE; NONHUMAN; PARTICLE SIZE; PH; PHYSICAL CHEMISTRY; RAT; SUSTAINED DRUG RELEASE;

EID: 0034000597     PISSN: 11571489     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (23)

1. SESSA G., WEISSMANN J. - Effect of polymer antibiotics on phospholipid spherules containing varying amounts of charged components. - Biochim. Biophys. Acta., 135, 416-426, 1967.
2. SASAKIH., KAKUTANI T., HASHIDA M., SEZAKIH.-Absorption characteristics of the lipophilic prodrug of mitomycin C from injected liposomes or an emulsion. - J. Pharm. Pharmacol., 37, 461-465, 1985.
3. ARAMAKI Y., TOMIZAWA H., HARA T., YACHI K., KIKUCHI H., TSUCHIYA S. - Stability of liposomes in vitro and their uptake by rat Peyer's patches following oral administration. - Pharm. Res., 10, 1228-1231, 1993.
4. MAITANIY. - Physicochemical characterization and application for drug carrier of soybean-derived sterols and their glucoside-containing liposomes. - Yakugaku Zasshi, 116, 901-910, 1996.
5. VERSLUIS A. J., RUMP E. T., RENSEN P. C., VAN BERKEL T. J., BIJSTERBOSCH M. K. - Synthesis of a lipophilic daunorubicin derivative and its incorporation into lipidic carriers developed for LDL receptor-mediated tumor therapy. - Pharm. Res., 15, 531-537, 1998.
6. TRUBETSKOY V. S., WHITEMAN K. R., TORCHILIN V. P., WOLF G. L. - Massage-induced release of subcutaneously injected liposome-encapsulated drugs to the blood. - J. Control. Release, 50, 13-19, 1998.
7. YOTSUYANAGI T., MIZUTANI J., IWATA M., IKEDA K. -Kinetic aspects and mechanism of liposome disintegration in polyoxyethylene lauryl ether and sodium cholate solutions. -Biochem. Biophys. Acta, 731, 304-311, 1983.
8. YOTSUYANAGI T., HASHIMOTO H., IWATA M., IKEDA K. -Effect of cholesterol on liposome stability to ultrasonic disintegration and sodium cholate solubilization. - Chem. Pharm. Bull., 35, 1228-1233, 1987.
9. NAGATA M., YOTSUYANAGI T., IKEDA K. - A two-step model of disintegration kinetics of liposomes in bile salts. - Chem. Pharm. Bull., 36, 1508-1513, 1988.
10. JAIN U. K., HIGUCHI W. I., LIU C. L., LEE P. H., MAZER N. A. -Cholesterol (thermodynamic) activity determinations in bile salt-lecithin-cholesterol systems and cholesterol-rich liquid crystalline mesophase formation. - Pharm. Res., 9, 792-799, 1992.
11. ALAMELU S., RAO K. P. - Effect of surfactants on the stability of modified egg-yolk phosphatidyl choline liposomes. - J. Microencapsul., 7, 541-551, 1990.
12. ALAMELU S., RAO K. P. - Studies on the carboxymethyl chitosan-containing liposomes for their stability and controlled release of dapsone. - J. Microencapsul., 8, 505-519, 1991.
13. ASSADULLAHI T. P., HAMID K., HIDER R. C. - In vitro stability of liposomes in the presence of polymers, trehalose and sodium taurocholate. - J. Microencapsulation, 9, 317-327, 1992.
14. KATO A., ARAKAWA M., KONDOT. - Preparation and stability of liposome-type artificial red blood cell stabilized with carboxymethyl chitin. - J. Microencapsul., 1, 105-112, 1984.
15. DONG C., ROGERS J. A. - Poly(4-vinylpyridine)-coated liposomes: stability studies and release of acetylsalicylic acid. - J. Microencapsul., 9, 437-448, 1992.
16. DONG C., ROGERS J.A. - Quantitative determination of carboxymethyl chitin in polymer-coated liposomes. - J. Microencapsul., 8, 153-160, 1991.
17. DONG C., ROGERS J. A. - Polymer-coated liposomes: stability and release of ASA from carboxymethyl chitin-coated liposomes. - J. Control. Release, 17, 217-224, 1991.
18. PAJEAN M., HUC A., HERBAGE D. - Stabilization of liposomes with collagen. - Int. J. Pharm., 77, 31-40, 1991.
19. DAVIES N. M., FARR S. J., HADGRAFT J., KELLAWAY I. W. - Evaluation of mucoadhesive polymers in ocular drug delivery. II. Polymer-coated vesicles. - Pharm. Res., 9, 1137-1144, 1992.
20. MARGALIT R., OKON M., YERUSHALMI N., AVIDOR E. -Bioadhesive liposomes as topical delivery systems: molecular and cellular studies. - J. Control. Release, 19, 275-288, 1992.
21. TAKEUCHI H., YAMAMOTO H., NIWA T., HINO T., KAWASHIMA Y. - Mucoadhesion of polymer-coated liposomes to rat intestine in vitro. - Chem. Pharm. Bull., 42, 1954-1956, 1994.
22. TAKEUCHI H., YAMAMOTO H., NIWA T., HINO T., KAWASHIMA Y. - Enteral absorption of insulin in rats from mucoadhesive chitosan-coated liposomes. - Pharm. Res., 13, 896-901, 1996.
23. Encyclopeadia chimica, Kyouritsu Shuppan Co. Ltd., 719-720, 1963.