메뉴 건너뛰기




Volumn 147, Issue 1, 1999, Pages 73-80

Effects of E-2078, a stable dynorphin A(1-8) analog, on sedation and serum prolactin levels in rhesus monkeys

Author keywords

opioid receptor; Dynorphin; E 2078; Macaca mulatta; Naltrexone; Prolactin; Sedation

Indexed keywords

3 [1 (3,4 DICHLORO N METHYLPHENYLACETAMIDO) 2 (1 PYRROLIDINYL)ETHYL]PHENOXYACETIC ACID; DYNORPHIN A [1-8][1 (N METHYLTYROSINE) 7 (N METHYLARGININE) 8 DEXTRO LEUCINE N ETHYLAMIDE]; NALTREXONE; PROLACTIN; QUADAZOCINE; SPIRADOLINE;

EID: 0033988331     PISSN: 00333158     EISSN: None     Source Type: Journal    
DOI: 10.1007/s002130051144     Document Type: Article
Times cited : (27)

References (39)
  • 1
    • 0023521010 scopus 로고
    • Early ontogeny of kappa-opioid receptor regulation of prolactin secretion in the rat
    • Bero LA, Lurie SN, Kuhn CM (1987) Early ontogeny of kappa-opioid receptor regulation of prolactin secretion in the rat. Brain Res 465:189-196
    • (1987) Brain Res , vol.465 , pp. 189-196
    • Bero, L.A.1    Lurie, S.N.2    Kuhn, C.M.3
  • 2
    • 0026482766 scopus 로고
    • Mu- and kappa- opiate receptor control of prolactin secretion in rats: Ontogeny and interaction with serotonin
    • Blackford SP, Little P, Kuhn CM (1992) Mu- and kappa- opiate receptor control of prolactin secretion in rats: ontogeny and interaction with serotonin. Endocrinology 131:2891-2897
    • (1992) Endocrinology , vol.131 , pp. 2891-2897
    • Blackford, S.P.1    Little, P.2    Kuhn, C.M.3
  • 4
    • 0032766057 scopus 로고    scopus 로고
    • Effects of systemically administered dynorphin A(1-17) in rhesus monkeys
    • Butelman ER, Harris TJ, Perez A and Kreek MJ (1999a) Effects of systemically administered dynorphin A(1-17) in rhesus monkeys. J Pharmacol Exp Ther 290:678-686
    • (1999) J Pharmacol Exp Ther , vol.290 , pp. 678-686
    • Butelman, E.R.1    Harris, T.J.2    Perez, A.3    Kreek, M.J.4
  • 5
    • 0032894930 scopus 로고    scopus 로고
    • Systemic effects of E-2078, a stabilized dynorphin A(1-8) analog, in rhesus monkeys
    • Butelman ER, Vivian JA, Yu J, Kreek MJ, Woods JH (1999b) Systemic effects of E-2078, a stabilized dynorphin A(1-8) analog, in rhesus monkeys. Psychopharmacology 143:190-196
    • (1999) Psychopharmacology , vol.143 , pp. 190-196
    • Butelman, E.R.1    Vivian, J.A.2    Yu, J.3    Kreek, M.J.4    Woods, J.H.5
  • 6
    • 0022479347 scopus 로고
    • A tail withdrawal procedure for assessment of analgesic activity in rhesus monkeys
    • Dykstra LA, Woods JH (1986) A tail withdrawal procedure for assessment of analgesic activity in rhesus monkeys. J Pharmacol Methods 15:263-269
    • (1986) J Pharmacol Methods , vol.15 , pp. 263-269
    • Dykstra, L.A.1    Woods, J.H.2
  • 7
    • 0023637786 scopus 로고
    • Kappa opioids in rhesus monkeys. I. Diuresis, sedation, analgesia, and discriminative stimulus effects
    • Dykstra LA, Gmerek DE, Winger G, Woods JH (1987a) Kappa opioids in rhesus monkeys. I. Diuresis, sedation, analgesia, and discriminative stimulus effects. J Pharmacol Exp Ther 242:413-420
    • (1987) J Pharmacol Exp Ther , vol.242 , pp. 413-420
    • Dykstra, L.A.1    Gmerek, D.E.2    Winger, G.3    Woods, J.H.4
  • 8
    • 0023626436 scopus 로고
    • Kappa opioids in rhesus monkeys. II. Analysis of the antagonistic actions of quadazocine and beta-funaltrexamine
    • Dykstra LA, Gmerek DE, Winger GD, Woods JH (1987b) Kappa opioids in rhesus monkeys. II. Analysis of the antagonistic actions of quadazocine and beta-funaltrexamine. J Pharmacol Exp Ther 242:421-427
    • (1987) J Pharmacol Exp Ther , vol.242 , pp. 421-427
    • Dykstra, L.A.1    Gmerek, D.E.2    Winger, G.D.3    Woods, J.H.4
  • 9
    • 0024414685 scopus 로고
    • Pharmacological characterization of supersensitivity to naltrexone in squirrel monkeys
    • France CP, Morse WH (1989) Pharmacological characterization of supersensitivity to naltrexone in squirrel monkeys. J Pharmacol Exp Ther 250:928-936
    • (1989) J Pharmacol Exp Ther , vol.250 , pp. 928-936
    • France, C.P.1    Morse, W.H.2
  • 10
    • 0028013439 scopus 로고
    • Comparison of kappa opioids in rhesus monkeys: Behavioral effects and binding affinities
    • France CP, Medzihradsky F, Woods JH (1994) Comparison of kappa opioids in rhesus monkeys: behavioral effects and binding affinities. J Pharmacol Exp Ther 268:47-58
    • (1994) J Pharmacol Exp Ther , vol.268 , pp. 47-58
    • France, C.P.1    Medzihradsky, F.2    Woods, J.H.3
  • 11
  • 12
    • 0029077098 scopus 로고
    • Central and peripheral analgesic agents: Chemical strategies for limiting brain penetration in kappa-opioid agonists belonging to different chemical classes
    • Giardina G, Clarke GD, Grugni M, Sbacchi M, Vecchietti V (1995) Central and peripheral analgesic agents: chemical strategies for limiting brain penetration in kappa-opioid agonists belonging to different chemical classes. Farmaco 50:405-418
    • (1995) Farmaco , vol.50 , pp. 405-418
    • Giardina, G.1    Clarke, G.D.2    Grugni, M.3    Sbacchi, M.4    Vecchietti, V.5
  • 13
    • 0022534411 scopus 로고
    • Dynorphin effects on plasma concentrations of anterior pituitary hormones in the nonhuman primate
    • Gilbeau PM, Hosobuchi Y, Lee NM (1986) Dynorphin effects on plasma concentrations of anterior pituitary hormones in the nonhuman primate. J Pharmacol Exp Ther 238:974-977
    • (1986) J Pharmacol Exp Ther , vol.238 , pp. 974-977
    • Gilbeau, P.M.1    Hosobuchi, Y.2    Lee, N.M.3
  • 14
    • 0020457110 scopus 로고
    • Kappa opiate receptors localized by autoradiography to deep layers of cerebral cortex: Relation to sedative effects
    • Goodman RR, Snyder SH (1982) Kappa opiate receptors localized by autoradiography to deep layers of cerebral cortex: relation to sedative effects. Proc Natl Acad Sci USA 79:5703-5707
    • (1982) Proc Natl Acad Sci USA , vol.79 , pp. 5703-5707
    • Goodman, R.R.1    Snyder, S.H.2
  • 15
    • 0029560396 scopus 로고
    • Opioid mechanisms controlling renal function
    • Kapusta DR (1995) Opioid mechanisms controlling renal function. Clin Exp Pharmacol Physiol 22:891-202
    • (1995) Clin Exp Pharmacol Physiol , vol.22 , pp. 891-202
    • Kapusta, D.R.1
  • 17
    • 0023234304 scopus 로고
    • Kappa-agonist induced diuresis:evidence for stereoselectivity, strain differences, independence of hydration variables and a result of decreased plasma vasopressin levels
    • Leander JD, Hart JC, Zerbe RL (1987) Kappa-agonist induced diuresis:evidence for stereoselectivity, strain differences, independence of hydration variables and a result of decreased plasma vasopressin levels. J Pharmacol Exp Ther 242:33-39
    • (1987) J Pharmacol Exp Ther , vol.242 , pp. 33-39
    • Leander, J.D.1    Hart, J.C.2    Zerbe, R.L.3
  • 18
    • 0021737545 scopus 로고
    • Anatomical relationship between opioid peptides and receptors in rhesus monkey brain
    • Lewis ME, Khachaturian H, Akil H, Watson SJ (1984) Anatomical relationship between opioid peptides and receptors in rhesus monkey brain. Brain Res Bull 13:801-812
    • (1984) Brain Res Bull , vol.13 , pp. 801-812
    • Lewis, M.E.1    Khachaturian, H.2    Akil, H.3    Watson, S.J.4
  • 19
    • 0020428008 scopus 로고
    • Effects of opiate antagonists and putative mu- and kappa- agonists on milk intake in rat and squirrel monkey
    • Locke KW, Brown DR, Holtzman SG (1982) Effects of opiate antagonists and putative mu- and kappa- agonists on milk intake in rat and squirrel monkey. Pharmacol Biochem Behav 17:1275-1279
    • (1982) Pharmacol Biochem Behav , vol.17 , pp. 1275-1279
    • Locke, K.W.1    Brown, D.R.2    Holtzman, S.G.3
  • 20
    • 0025742665 scopus 로고
    • Neurons with access to the general circulation in the central nervous system of the rat: A retrograde tracing study with fluoro-gold
    • Merchenthaler I (1991) Neurons with access to the general circulation in the central nervous system of the rat: a retrograde tracing study with fluoro-gold. Neuroscience 44:655-662
    • (1991) Neuroscience , vol.44 , pp. 655-662
    • Merchenthaler, I.1
  • 21
    • 0002131424 scopus 로고
    • Dopaminergic neuronal systems in the hypothalamus
    • Bloom FE, Kupfer DE (eds) Raven Press, New York
    • Moore KE, Lookingland KJ (1995) Dopaminergic neuronal systems in the hypothalamus. In: Bloom FE, Kupfer DE (eds) Psychopharmacology: the fourth generation of progress. Raven Press, New York, pp 245-256
    • (1995) Psychopharmacology: The Fourth Generation of Progress , pp. 245-256
    • Moore, K.E.1    Lookingland, K.J.2
  • 24
    • 0026019747 scopus 로고
    • Spinal kappa-receptor mediated analgesia of E-2078, a systemically active dynorphin analog, in mice
    • Nakazawa T, Furuya Y, Kaneko T, Yamatsu K (1991) Spinal kappa-receptor mediated analgesia of E-2078, a systemically active dynorphin analog, in mice. J Pharmacol Exp Ther 256:76-81
    • (1991) J Pharmacol Exp Ther , vol.256 , pp. 76-81
    • Nakazawa, T.1    Furuya, Y.2    Kaneko, T.3    Yamatsu, K.4
  • 25
    • 0027495926 scopus 로고
    • Effects of opioid agonists selective for mu, kappa and delta opioid receptors on schedule controlled responding in rhesus monkeys: Antagonism by quadazocine
    • Negus SS, Burke TF, Medzhiradsky F, Woods JH (1993) Effects of opioid agonists selective for mu, kappa and delta opioid receptors on schedule controlled responding in rhesus monkeys: antagonism by quadazocine. J Pharmacol Exp Ther 267:896-903
    • (1993) J Pharmacol Exp Ther , vol.267 , pp. 896-903
    • Negus, S.S.1    Burke, T.F.2    Medzhiradsky, F.3    Woods, J.H.4
  • 26
    • 0031817881 scopus 로고    scopus 로고
    • Behavioral effects of the delta-selective opioid agonist SNC80 and related compounds in rhesus monkeys
    • Negus SS, Gatch MB, Mello NK, Zhang X, Rice K (1998) Behavioral effects of the delta-selective opioid agonist SNC80 and related compounds in rhesus monkeys. J Pharmacol Exp Ther 286:362-375
    • (1998) J Pharmacol Exp Ther , vol.286 , pp. 362-375
    • Negus, S.S.1    Gatch, M.B.2    Mello, N.K.3    Zhang, X.4    Rice, K.5
  • 28
    • 0026805532 scopus 로고
    • Analgesic and discriminative stimulus properties of U-62,066E, the selective kappa-opioid receptor agonist, in the rat
    • Ohno M, Yamamoto T, Ueki S (1992) Analgesic and discriminative stimulus properties of U-62,066E, the selective kappa-opioid receptor agonist, in the rat. Psychopharmacology 106:31-38
    • (1992) Psychopharmacology , vol.106 , pp. 31-38
    • Ohno, M.1    Yamamoto, T.2    Ueki, S.3
  • 29
    • 0023139711 scopus 로고
    • The effects of the systemic administration of n-methylmorphine chloride, a quaternary analogue of morphine that does not cross the blood-brain barrier, on the release of anterior pituitary hormones in the rat
    • Pechnick RN, George R, Poland RE (1987) The effects of the systemic administration of n-methylmorphine chloride, a quaternary analogue of morphine that does not cross the blood-brain barrier, on the release of anterior pituitary hormones in the rat. Psychoneuroendocrinology 12:67-71
    • (1987) Psychoneuroendocrinology , vol.12 , pp. 67-71
    • Pechnick, R.N.1    George, R.2    Poland, R.E.3
  • 30
    • 0028006303 scopus 로고
    • Pharmacological characterization of cloned κ, δ, and μ-opioid receptors
    • Raynor K, Hong H, Yasuda K, Yu L, Bell GI, Reisine T (1994) Pharmacological characterization of cloned κ, δ, and μ-opioid receptors. Mol Pharmacol 45:330-334
    • (1994) Mol Pharmacol , vol.45 , pp. 330-334
    • Raynor, K.1    Hong, H.2    Yasuda, K.3    Yu, L.4    Bell, G.I.5    Reisine, T.6
  • 33
    • 0026611409 scopus 로고    scopus 로고
    • Huidobro-Toro (1992) [N-methyl-Tyrl, N-methyl-Arg7-D-Leu]- Dynorphin A(1-8) ethylamide, a stable dynorphin analog, produces diuresis by kappa-opiate receptor activation in the rat
    • Salas SP, Roblero JS, Lopez LF, Tachibana T, Huidobro-Toro (1992) [N-methyl-Tyrl, N-methyl-Arg7-D-Leu]- Dynorphin A(1-8) ethylamide, a stable dynorphin analog, produces diuresis by kappa-opiate receptor activation in the rat. J Pharmacol Exp Ther 262:979-986
    • J Pharmacol Exp Ther , vol.262 , pp. 979-986
    • Salas, S.P.1    Roblero, J.S.2    Lopez, L.F.3    Tachibana, T.4
  • 34
    • 0024506654 scopus 로고
    • ICI204448: A κ-opioid agonist with limited access to the CNS
    • Shaw JS, Carroll JA, Alcock P, Main BG (1989) ICI204448: a κ-opioid agonist with limited access to the CNS. Br J Pharmacol 96:986-992
    • (1989) Br J Pharmacol , vol.96 , pp. 986-992
    • Shaw, J.S.1    Carroll, J.A.2    Alcock, P.3    Main, B.G.4
  • 35
    • 0025737104 scopus 로고
    • Evaluation of the sites of opioid influence on anterior pituitary hormone secretion using a quaternary opiate antagonist
    • Simpkins JW, Swager D, Millard WJ (1991) Evaluation of the sites of opioid influence on anterior pituitary hormone secretion using a quaternary opiate antagonist. Neuroendocrinology 54:384-390
    • (1991) Neuroendocrinology , vol.54 , pp. 384-390
    • Simpkins, J.W.1    Swager, D.2    Millard, W.J.3
  • 38
  • 39
    • 0030743498 scopus 로고    scopus 로고
    • Dynorphin A(1-8) analog, E-2078, crosses the blood-brain barrier in rhesus monkeys
    • Yu J, Butelman ER, Woods JH, Chait BT, Kreek MJ (1997b) Dynorphin A(1-8) analog, E-2078, crosses the blood-brain barrier in rhesus monkeys. J Pharmacol Exp Ther 282:633-638
    • (1997) J Pharmacol Exp Ther , vol.282 , pp. 633-638
    • Yu, J.1    Butelman, E.R.2    Woods, J.H.3    Chait, B.T.4    Kreek, M.J.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.