Differential down-regulation of the human d-opioid receptor by SNC80 and [D-Pen2, D-Pen5]enkephalin

European Journal of Pharmacology

Volumn 387, Issue 2, 2000, Pages R11-R13

  Okura, Takashi ^a   Cowell, Scott M ^a   Varga, Eva ^a   Burkey, Thomas H ^a   Roeske, William R ^a   Hruby, Victor J ^a   Yamamura, Henry I ^a  

^a UNIVERSITY OF ARIZONA   (United States)

Author keywords

Carboxyl terminal tail; d Opioid receptor; Down regulation

Indexed keywords

4 [ALPHA (4 ALLYL 2,5 DIMETHYL 1 PIPERAZINYL) 3 METHOXYBENZYL] N,N DIETHYLBENZAMIDE; DELTA OPIATE RECEPTOR; ENKEPHALIN[2 DEXTRO ALANINE 5 DEXTRO LEUCINE]; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE]; NALTRINDOLE;

ANIMAL CELL; ARTICLE; CARBOXY TERMINAL SEQUENCE; CHO CELL; CONTROLLED STUDY; DRUG RECEPTOR BINDING; NEUROMODULATION; NONHUMAN; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION;

BENZAMIDES; DOWN-REGULATION; ENKEPHALIN, D-PENICILLAMINE (2,5)-; HUMANS; NALTREXONE; PIPERAZINES; RECEPTORS, OPIOID, DELTA;

EID: 0033984575     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(99)00761-X     Document Type: Article

References (5)

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3. 284 of the human δ opioid receptor is required for SNC121 binding but not binding of pCl-DPDPE, deltorphin II or naltrindole. Analgesia. 1:1995;539-542.
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