Mechanism of biochemical action of substituted 4-methylbenzopyran-2-ones. Part 7: Assay and characterization of 7,8-diacetoxy-4-methylcoumarin:protein transacetylase from rat liver microsomes based on the irreversible inhibition of cytosolic glutathione S-transferase

Bioorganic and Medicinal Chemistry

Volumn 8, Issue 7, 2000, Pages 1707-1712

  Raj, Hanumantharao G ^a   Parmar, Virinder S ^b   Jain, Subhash C ^b   Kohli, Ekta ^a   Ahmad, Nizamuddin ^c   Goel, Sanjay ^a   Tyagi, Yogesh K ^a   Sharma, Sunil K ^b   Wengel, Jesper ^d   Olsen, Carl E ^e  

^a UNIVERSITY OF DELHI   (India)

^b UNIVERSITY OF DELHI   (India)

^c INDIAN VETERINARY RESEARCH INSTITUTE   (India)

^d UNIVERSITY OF COPENHAGEN   (Denmark)

^e UNIVERSITY OF COPENHAGEN   (Denmark)

Author keywords

[No Author keywords available]

Indexed keywords

7,8 DIACETOXY 4 METHYLCOUMARIN; COUMARIN DERIVATIVE; GLUTATHIONE TRANSFERASE; UNCLASSIFIED DRUG;

ACETYLATION; ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; DRUG MECHANISM; ENZYME INHIBITION; ION EXCHANGE CHROMATOGRAPHY; LIVER MICROSOME; METHODOLOGY; NONHUMAN; RAT;

ACETYLATION; ACETYLTRANSFERASES; ANIMALS; BENZOPYRANS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; COUMARINS; CYTOSOL; DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME INHIBITORS; GLUTATHIONE TRANSFERASE; KINETICS; MALE; MICROSOMES, LIVER; RATS; RATS, WISTAR; SUBSTRATE SPECIFICITY; TIME FACTORS;

EID: 0033944241     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(00)00104-8     Document Type: Article

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