Characterization of a binding site of UCN-01, a novel anticancer drug on α1-acid glycoprotein

Biological and Pharmaceutical Bulletin

Volumn 23, Issue 7, 2000, Pages 893-895

  Kurata, Noriaki ^a   Matsushita, Sadaharu ^b   Nishi, Koji ^b   Watanabe, Hiroshi ^b   Kobayashi, Satoshi ^a   Suenaga, Ayaka ^b   Otagiri, Masaki ^b  

^a KYOWA HAKKO KOGYO CO LTD   (Japan)

^b KUMAMOTO UNIVERSITY   (Japan)

Author keywords

Binding site; Competitive displacement; UCN 01; 1 acid glycoprotein

Indexed keywords

7 HYDROXYSTAUROSPORINE; OROSOMUCOID; PROGESTERONE; PROPRANOLOL; WARFARIN;

ARTICLE; BINDING AFFINITY; BINDING SITE; DRUG BINDING SITE; DRUG PROTEIN BINDING;

EID: 0033943747     PISSN: 09186158     EISSN: None     Source Type: Journal    
DOI: 10.1248/bpb.23.893     Document Type: Article

References (15)

1. Akinaga S., Gomi K., Morimoto M., Tamaoki T., Okabe M., Cancer Res., 51, 4888-4892 (1991).
2. Akinaga S., Nomura K., Gomi K., Okabe M., Cancer Chemother. Pharmacol., 33, 273-280 (1994).
3. Fuse E., Tanii H., Kurata N., Kobayashi H., Shimada Y., Tamura T., Sasaki Y., Tanigawara Y., Lush R. D., Headlee D., Figg W. D., Arbuck S. G., Senderowicz A. M., Sausville E. A., Akinaga S., Kuwabara T., Kobayashi S., Cancer Res., 58, 3248-3253 (1998).
4. Fuse E., Tanii H., Takai K., Asanome K., Kurata N., Kobayashi H., Kuwabara T., Kobayashi S., Sugiyama Y., Cancer Res., 59, 1054-1060 (1999).
5. Takahashi I., Kobayashi E., Asano K., Yoshida M., Nakano H., J. Antibiot., 40, 1782-1784 (1987).
6. Bombardt P. A., Brewer J. E., Johnson M. G., J. Pharmacol. Exp. Ther., 269, 145-150 (1994).
7. Yamaoka K., Tanigawara Y., Nakagawa T., Uno T., J. PharmacobioDyn, 4, 879-885 (1981).
8. Eap C. B., Baumann P., Electrophoresis, 9, 650-654 (1988).
9. Yuasa I., Weidinger S., Umetsu K., Suenaga K., Ishimoto G., Eap B. C., Duche J. C., Baumann P., Vox Sang., 64, 47-55 (1993).
10. Herve F., Caron G., Duche J. C., Gaillard P., Abd Rahman N., Tsantili-Kakoulidou A., Carrupt P. A., d'Athis P., Tillement J. P., Testa B., Mol. Pharmacol., 54, 129-138 (1998).
11. Herve F., Foache F., Marche C., Tillement J. P., J. Chromatogr. B, 688, 35-46 (1997).
12. Imamura H., Maruyama T., Okabe H., Shimada H., Otagiri M., Pharm. Res., 11, 566-570 (1994).
13. Urien S., Giroud Y., Tsai R. S., Carrupt P. A., Bree F., Testa B., Tilliment J. P., Biochem. J., 306, 545-549 (1995).
14. Otagiri M., Miyoshi T., Yamamichi R., Maruyama T., Perrin J. H., Biochem. Pharmacol., 42, 729-733 (1991).
15. Miyoshi T., Yamamichi R., Maruyama T., Takadate A., Otagiri M., Biochem. Pharmacol., 43, 2161-2167 (1992).