Molecular modeling of the complex of endothelin-1(ET-1) with the endothelin type a (ET(A)) receptor and the rational design of a peptide antagonist

Journal of Biomolecular Structure and Dynamics

Volumn 17, Issue 6, 2000, Pages 957-964

  Bhatnagar, Sonika ^a   Rao, Gita Subba ^a  

^a ALL INDIA INSTITUTE OF MEDICAL SCIENCES   (India)

Author keywords

[No Author keywords available]

Indexed keywords

CYCLO(DEXTRO TRYPTOPHYL DEXTRO ASPARTYLPROLYL DEXTRO VALYLLEUCYL); ENDOTHELIN 1; ENDOTHELIN A RECEPTOR; ENDOTHELIN RECEPTOR ANTAGONIST;

ARTICLE; COMPETITIVE INHIBITION; COMPLEX FORMATION; DRUG BINDING SITE; DRUG CONFORMATION; DRUG DESIGN; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; MOLECULAR MODEL; PRIORITY JOURNAL; REACTION ANALYSIS; RECEPTOR BLOCKING; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

ANTIHYPERTENSIVE AGENTS; DRUG DESIGN; ENDOTHELIN-1; HUMANS; MODELS, MOLECULAR; MUTAGENESIS, SITE-DIRECTED; PEPTIDES; PEPTIDES, CYCLIC; PROTEIN BINDING; PROTEIN CONFORMATION; PROTEIN FOLDING; RECEPTOR, ENDOTHELIN A; RECEPTORS, ENDOTHELIN; SIGNAL TRANSDUCTION; VASOCONSTRICTOR AGENTS;

EID: 0033926599     PISSN: 07391102     EISSN: None     Source Type: Journal    
DOI: 10.1080/07391102.2000.10506584     Document Type: Article

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