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Volumn 43, Issue 12, 2000, Pages 2350-2355

CCK peptides with combined features of hexa- and tetrapeptide CCK-A agonists

Author keywords

[No Author keywords available]

Indexed keywords

BENZODIAZEPINE DERIVATIVE; CHOLECYSTOKININ A RECEPTOR; CHOLECYSTOKININ RECEPTOR STIMULATING AGENT; HEXAPEPTIDE; TETRAPEPTIDE;

EID: 0033919839     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm990252e     Document Type: Article
Times cited : (8)

References (25)
  • 1
    • 0003111499 scopus 로고
    • Cholecystokinin: Isolation, structure and functions
    • Glass. G. B. J., Ed.; Raven Press: New York
    • Mutt, V. Cholecystokinin: Isolation, Structure and Functions. In Gastrointestinal Hormones; Glass. G. B. J., Ed.; Raven Press: New York, 1980; pp 169-221.
    • (1980) Gastrointestinal Hormones , pp. 169-221
    • Mutt, V.1
  • 3
    • 0028300692 scopus 로고
    • Biological actions of cholecystokinin
    • Crawley, J. N.; Corwin, R. L. Biological Actions of Cholecystokinin. Peptides 1994, 15, 731-755.
    • (1994) Peptides , vol.15 , pp. 731-755
    • Crawley, J.N.1    Corwin, R.L.2
  • 4
    • 0001669859 scopus 로고
    • Classification and function of CCK receptors
    • Dourish, C., T.; Hill, D. R. Classification and Function of CCK Receptors. Trends Pharmacol. Sci. 1987, 8, 207-208.
    • (1987) Trends Pharmacol. Sci. , vol.8 , pp. 207-208
    • Dourish, C.T.1    Hill, D.R.2
  • 5
    • 0028340876 scopus 로고
    • Satiating effect of cholecystokinin
    • Smith, G. P.; Gibbs, J. Satiating Effect of Cholecystokinin. Ann. N.Y. Acad. Sci. 1994, 773, 236-241.
    • (1994) Ann. N.Y. Acad. Sci. , vol.773 , pp. 236-241
    • Smith, G.P.1    Gibbs, J.2
  • 8
    • 0026699197 scopus 로고
    • Synthesis and biological activities of CCK heptapeptide analogues. Effects on conformational constraints and standard modifications on receptor subtype selectivity and functional activity in vitro and appetite suppression in vivo
    • Holladay, M. W.; Bennett, M.; Tufano, M.; Lin, C.; Asin, K.; Witte, D.; Miller, T.; Bianchi, B.; Bednarz, L.; Nadzan, A. Synthesis and Biological Activities of CCK Heptapeptide Analogues. Effects on Conformational Constraints and Standard Modifications on Receptor Subtype Selectivity and Functional Activity in Vitro and Appetite Suppression In Vivo. J. Med. Chem. 1992, 35, 2919-2928.
    • (1992) J. Med. Chem. , vol.35 , pp. 2919-2928
    • Holladay, M.W.1    Bennett, M.2    Tufano, M.3    Lin, C.4    Asin, K.5    Witte, D.6    Miller, T.7    Bianchi, B.8    Bednarz, L.9    Nadzan, A.10
  • 9
    • 77956808092 scopus 로고
    • Cholecystokinin agonists and antagonists
    • Bristol, J. A., Ed., Academic: San Diego, CA
    • Nadzan, A. M.; Kerwin, Jr., J. F. Cholecystokinin Agonists and Antagonists. In Annual Reports in Medicinal Chemistry, Bristol, J. A., Ed., Academic: San Diego, CA, 1991; pp 191-200.
    • (1991) Annual Reports in Medicinal Chemistry , pp. 191-200
    • Nadzan, A.M.1    Kerwin J.F., Jr.2
  • 14
    • 0026623087 scopus 로고
    • Development of potent and selective CCK-A receptor agonist from Boc-CCK-4: Tetrapeptides containing lys(N′)-Amide residues
    • Shiosaki, K.; Lin, C. W.; Kopecka, H.; Craig, R.; Bianchi, B.; Miller, T.; Witte, D.; Stashko, M.; Nadzan, A. Development of Potent and Selective CCK-A Receptor Agonist from Boc-CCK-4: Tetrapeptides Containing Lys(N′)-Amide Residues. J. Med. Chem. 1992, 35, 2007-2014.
    • (1992) J. Med. Chem. , vol.35 , pp. 2007-2014
    • Shiosaki, K.1    Lin, C.W.2    Kopecka, H.3    Craig, R.4    Bianchi, B.5    Miller, T.6    Witte, D.7    Stashko, M.8    Nadzan, A.9
  • 17
    • 0025103048 scopus 로고
    • A cleavage method which minimizes side reactions following fmoc solid-phase peptide synthesis
    • King, D. S.; Fields, C. G.; Fields, G. B. A Cleavage Method Which Minimizes Side Reactions Following Fmoc Solid-Phase Peptide Synthesis. Int. J. Pept. Protein Res. 1990, 36, 255-266.
    • (1990) Int. J. Pept. Protein Res. , vol.36 , pp. 255-266
    • King, D.S.1    Fields, C.G.2    Fields, G.B.3
  • 18
    • 0022557566 scopus 로고
    • 3H-(±)-L-364,718: A new potent, nonpeptide cholecystokinin antagonist radioligand selective for peripheral receptors
    • 3H-(±)-L-364,718: A New Potent, Nonpeptide Cholecystokinin Antagonist Radioligand Selective for Peripheral Receptors. Mol. Pharmacol. 1986, 30, 212-217.
    • (1986) Mol. Pharmacol. , vol.30 , pp. 212-217
    • Chang, R.S.L.1    Lotti, V.J.2    Chen, T.B.3    Kunkel, K.A.4
  • 19
    • 0001603410 scopus 로고
    • Biochemical and pharmacological characterization of an extremely potent and selective nonpeptide cholecystokinin antagonist
    • Chang, R. S. L.; Lotti, V. J. Biochemical and Pharmacological Characterization of an Extremely Potent and Selective Nonpeptide Cholecystokinin Antagonist. Proc. Natl. Acad. Sci. U.S.A. 1986, 83, 4923-4926.
    • (1986) Proc. Natl. Acad. Sci. U.S.A. , vol.83 , pp. 4923-4926
    • Chang, R.S.L.1    Lotti, V.J.2
  • 20
    • 0015318507 scopus 로고
    • Comparison of anorexigenic and behavioral potency of phenylethylamines
    • Cox, R. H.; Maickel, R. P. Comparison of Anorexigenic and Behavioral Potency of Phenylethylamines. J. Pharmacol. Exp. Ther. 1972, 181, 1-9.
    • (1972) J. Pharmacol. Exp. Ther. , vol.181 , pp. 1-9
    • Cox, R.H.1    Maickel, R.P.2
  • 21
    • 0026686132 scopus 로고
    • A-71623, a selective CCK-A receptor agonist, suppresses food intake in the mouse, dog and monkey
    • Asin, K.; Bendnarz, L.; Nikkel, A.; Gore, P.; Nadzan, A. A-71623, A Selective CCK-A Receptor Agonist, Suppresses Food Intake in the Mouse, Dog and Monkey. Pharmacol. Biochem. Behav. 1992, 42, 699-704.
    • (1992) Pharmacol. Biochem. Behav. , vol.42 , pp. 699-704
    • Asin, K.1    Bendnarz, L.2    Nikkel, A.3    Gore, P.4    Nadzan, A.5
  • 22
    • 84908742429 scopus 로고
    • Peptide nomenclature follows the guidelines of the IUPAC-IUB joint commission on biochemical nomenclature
    • Peptide nomenclature follows the guidelines of the IUPAC-IUB Joint Commission on Biochemical Nomenclature. Eur. J. Biochem. 1984, 138, 9-37.
    • (1984) Eur. J. Biochem. , vol.138 , pp. 9-37
  • 24
    • 0020446693 scopus 로고
    • Calculating the dissociation constant of an unlabeled compound from the concentration required to displace radiolabel binding by 50%
    • Linden, J. Calculating the Dissociation Constant of an Unlabeled Compound from the Concentration Required to Displace Radiolabel Binding by 50%. J. Cyc. Nucleotide Res. 1982, 8, 162-172.
    • (1982) J. Cyc. Nucleotide Res. , vol.8 , pp. 162-172
    • Linden, J.1
  • 25
    • 0015386271 scopus 로고
    • Mathematical theory of complex ligand-binding systems at equilibrium: Some methods of parameter fitting
    • Feldman, H. A. Mathematical Theory of Complex Ligand-Binding Systems at Equilibrium: Some Methods of Parameter Fitting. Anal. Biochem. 1972, 48, 317-338.
    • (1972) Anal. Biochem. , vol.48 , pp. 317-338
    • Feldman, H.A.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.