Noncompetitive antagonist-binding sites of rat and housefly γ-aminobutyric acid receptors display different enantiospecificities for tert-butyl(isopropyl)bicyclophosphorothionate

Bioorganic and Medicinal Chemistry

Volumn 8, Issue 9, 2000, Pages 2337-2341

  Ju, Xiu Lian ^a   Ozoe, Yoshihisa ^a  

^a SHIMANE UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID RECEPTOR; 4 AMINOBUTYRIC ACID RECEPTOR BLOCKING AGENT; 4 TERT BUTYL 3 ISOPROPYL 2,6,7 TRIOXA 1 PHOSPHA BICYCLO[2.2.2]OCTANE 1 SULFIDE; IONOTROPIC RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BRAIN; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ENANTIOMER; HOUSE FLY; IN VITRO STUDY; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; RAT; SPECIES DIFFERENCE; STRUCTURE ACTIVITY RELATION;

ANIMALS; BICYCLO COMPOUNDS, HETEROCYCLIC; BINDING SITES; BINDING, COMPETITIVE; BRAIN; CELL MEMBRANE; DOSE-RESPONSE RELATIONSHIP, DRUG; GABA AGONISTS; HOUSEFLIES; INHIBITORY CONCENTRATION 50; MAGNETIC RESONANCE SPECTROSCOPY; ORGANOPHOSPHORUS COMPOUNDS; PROTEIN STRUCTURE, TERTIARY; RATS; RECEPTORS, GABA; STEREOISOMERISM; THIOPHOSPHORIC ACID ESTERS;

EID: 0033879529     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(00)00162-0     Document Type: Article

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