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Volumn 20, Issue 9, 1999, Pages 429-439

Pharmacokinetics of ezlopitant, a novel non-peptidic neurokinin-1 receptor antagonist in preclinical species and metabolite kinetics of the pharmacologically active metabolites

(5) Reed Hagen, Anne E a Tsuchiya, Megumi a Shimada, Kaoru a Wentland, Jo Ann a Scott Obach, R a

a PFIZER INC (United States)

Author keywords

Active metabolites; Cerebrospinal fluid; Ezlopitant; NK 1 antagonist; Pharmacokinetics

Indexed keywords

2 DIPHENYLMETHYL 3 (5 ISOPROPYL 2 METHOXY BENZYLAMINO)1 AZABICYCLO[2.2.2]OCTANE; CJ 12458; CJ 12764; EZLOPITANT; NEUROKININ 1 RECEPTOR ANTAGONIST; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG CLEARANCE; DRUG METABOLISM; DRUG RECEPTOR BINDING; DRUG STRUCTURE; FEMALE; FERRET; GERBIL; GUINEA PIG; LIVER BLOOD FLOW; MALE; NONHUMAN; RAT; STEADY STATE;

EID: 0033864633 PISSN: 01422782 EISSN: None Source Type: Journal
DOI: 10.1002/1099-081X(199912)20:9<429::AID-BDD209>3.0.CO;2-D Document Type: Article

Times cited : (20)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.