Reductive methylation of secondary amines containing reducible, hydrolyzable and sterically hindered groups

Synthetic Communications

Volumn 30, Issue 18, 2000, Pages 3353-3362

  Davis, Bruce A ^a   Durden, David A ^a  

^a UNIVERSITY OF SASKATCHEWAN   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

ARTICLE; CHEMICAL STRUCTURE; METHYLATION; REACTION ANALYSIS; REACTION TIME; REDUCTION;

EID: 0033862286     PISSN: 00397911     EISSN: None     Source Type: Journal    
DOI: 10.1080/00397910008086975     Document Type: Article

References (9)

1. Ainsworth, C.; Easton, N.R. J. Org. Chem. 1961, 26, 3776.
2. Djuric, S.W. J. Org. Chem. 1984, 49, 1311.
3. Barbry, D.; Torchy, S. Synth. Commun. 1996, 26, 3919.
4. Gribble, G.W.; Nutaitis, C.F. Synthesis 1987, 709.
5. Ramanjulu, J.M.; Joullie, M.M. Synth. Commun. 1996, 26, 1379.
6. Loibner, H.; Pruckner, A.; Stutz, A. Tetrahedron Lett. 1984, 25, 2535.
7. Yu, P.H.; Davis, B.A.; Boulton, A.A. J. Med. Chem. 1992, 35, 3705.; U.S. Patent No. 5,169,868; December 8, 1992.
8. Dyck, L.E.; Davis, B.A.; Paterson, I.A.; Liu, Y.D.; Durden, D.A.; Boulton, A.A. International Patent Application No. PCT/CA/00250. International filing date: March 25, 1999.
9. The authors thank Saskatchewan Health for continuing financial support.