Differential modes of agonist binding to 5-hydroxytryptamine2(A) serotonin receptors revealed by mutation and molecular modeling of conserved residues in transmembrane region 5

Molecular Pharmacology

Volumn 58, Issue 5, 2000, Pages 877-886

  Shapiro, David A ^a   Kristiansen, Kurt ^b   Kroeze, Wesley K ^a   Roth, Bryan L ^a  

^a CASE WESTERN RESERVE UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b UNIVERSITY OF TROMSØ   (Norway)

Author keywords

[No Author keywords available]

Indexed keywords

4 IODO 2,5 DIMETHOXYAMPHETAMINE; 5 METHYL N,N DIMETHYLTRYPTAMINE; ALPHA METHYLSEROTONIN; KETANSERIN; N METHYLSEROTONIN; PHOSPHATIDYLINOSITIDE; RITANSERIN; SEROTONIN; SEROTONIN 2A AGONIST; SEROTONIN 2A RECEPTOR; SPIPERONE; TRYPTAMINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CELL STRAIN COS7; CONTROLLED STUDY; DRUG RECEPTOR BINDING; FIBROBLAST CULTURE; GENETIC TRANSFECTION; HYDROLYSIS; MOLECULAR DYNAMICS; MOLECULAR INTERACTION; MOLECULAR MODEL; NONHUMAN; PRIORITY JOURNAL; PROTEIN STRUCTURE; SECOND MESSENGER; SITE DIRECTED MUTAGENESIS;

EID: 0033786003     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.58.5.877     Document Type: Article

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