Tetrapeptide derivatives of [D-Pen2,D-Pen5]-enkephalin (DPDPE) lacking an N-terminal tyrosine residue are agonists at the μ-opioid receptor

Journal of Pharmacology and Experimental Therapeutics

Volumn 295, Issue 3, 2000, Pages 960-966

  McFadyen, Iain J ^a   Sobczyk Kojiro, Katarzyna ^b   Schaefer, Michael J ^a   Ho, Jeffrey C ^b   Omnaas, John R ^b   Mosberg, Henry I ^b   Traynor, John R ^a  

^a UNIVERSITY OF MICHIGAN MEDICAL SCHOOL   (United States)

^b UNIVERSITY OF MICHIGAN   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DISULFIDE; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE]; ISOQUINOLINE DERIVATIVE; JH 54; MU OPIATE RECEPTOR; MU OPIATE RECEPTOR AGONIST; NAPHTHYL GROUP; PHENYL GROUP; PROLINE DERIVATIVE; TETRALIN DERIVATIVE; TETRAPEPTIDE; TYROSINE;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; DRUG CONFORMATION; DRUG EFFICACY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SYNTHESIS; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION;

ANIMALS; CELLS, CULTURED; ENKEPHALIN, D-PENICILLAMINE (2,5)-; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); GUINEA PIGS; PEPTIDES, CYCLIC; RADIOLIGAND ASSAY; RECEPTORS, OPIOID, MU; STRUCTURE-ACTIVITY RELATIONSHIP; TYROSINE;

EID: 0033680378     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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