Synthesis and binding affinity of cis-(-)- and cis-(+)-N-ethyleneamino-N-nordeoxymetazocine and cis-(-)-N-normetazocine analogues at σ1, σ2 and κ opioid receptors

European Journal of Pharmaceutical Sciences

Volumn 12, Issue 3, 2001, Pages 277-284

  Ronsisvalle, Giuseppe ^a   Prezzavento, Orazio ^a   Marrazzo, Agostino ^a   Vittorio, Franco ^a   Bousquet, Ennio ^a   Di Toro, Rosanna ^b   Spampinato, Santi ^b  

^a UNIVERSITY OF CATANIA   (Italy)

^b UNIVERSITY OF BOLOGNA   (Italy)

Author keywords

Kappa opioid receptor; Normetazocine derivative; Sigma receptors

Indexed keywords

6,11 DIMETHYL 3 [2 (METHYLPHENYLAMINO)ETHYL 1,2,3,4,5,6 HEXAHYDRO 6 METHANOBENZOZOCIN 8 OL; KAPPA OPIATE RECEPTOR; KAPPA OPIATE RECEPTOR AGONIST; MU OPIATE RECEPTOR; N ETHYLENEAMINO N NORDEOXYMETAZOCINE; NORMETAZOCINE DERIVATIVE; SIGMA OPIATE RECEPTOR; SIGMA OPIATE RECEPTOR STIMULATING AGENT; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CIS ISOMER; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GUINEA PIG; LIGAND BINDING; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; STRUCTURE ACTIVITY RELATION;

EID: 0033668152     PISSN: 09280987     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0928-0987(00)00157-3     Document Type: Article

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