A Gα(s) carboxyl-terminal peptide prevents G(s) activation by the A(2A) adenosine receptor

Molecular Pharmacology

Volumn 58, Issue 1, 2000, Pages 226-236

  Mazzoni, Maria R ^a,g   Taddei, Simone ^a   Giusti, Laura ^a   Rovero, Paolo ^b   Galoppini, Claudia ^d   D'Ursi, Annamaria ^b   Albrizio, Stefania ^b   Triolo, Antonio ^e   Novellino, Ettore ^c   Greco, Giovanni ^c   Lucacchini, Antonio ^a   Hamm, Heidi E ^f  

^a UNIVERSITY OF PISA   (Italy)

^b UNIVERSITY OF SALERNO   (Italy)

^c UNIVERSITY OF NAPLES FEDERICO II   (Italy)

^d CNR   (Italy)

^e Menarini Ricerche SpA   (Italy)

^f NORTHWESTERN UNIVERSITY   (United States)

^g Dipto Psichiatria Neurbio F   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); 5 AMINO 2 (2 FURYL) 7 (2 PHENYLETHYL)PYRAZOLO[4,3 E][1,2,4]TRIAZOLO[1,5 C]PYRIMIDINE; ADENOSINE A2A RECEPTOR; ADENOSINE; ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE RECEPTOR; DRUG DERIVATIVE; PEPTIDE; PHENETHYLAMINE DERIVATIVE; PYRIMIDINE DERIVATIVE; STIMULATORY GUANINE NUCLEOTIDE BINDING PROTEIN; TRIAZOLE DERIVATIVE; TRITIUM;

ALPHA HELIX; ANIMAL TISSUE; ARTICLE; CARBOXY TERMINAL SEQUENCE; DRUG EFFECT; DRUG SYNTHESIS; ENZYME ACTIVITY; MOLECULAR INTERACTION; NONHUMAN; PEPTIDE SYNTHESIS; PRIORITY JOURNAL; PROTEIN PROTEIN INTERACTION; RAT; RECEPTOR BINDING; STRIATE CORTEX; ANIMAL; BINDING COMPETITION; CELL MEMBRANE; CHEMISTRY; IN VITRO STUDY; MALE; METABOLISM; MOLECULAR GENETICS; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PROTEIN CONFORMATION; RADIOASSAY; SIGNAL TRANSDUCTION; SPRAGUE DAWLEY RAT; SYNTHESIS;

ADENOSINE; ADENOSINE-5'-(N-ETHYLCARBOXAMIDE); ANIMALS; BINDING, COMPETITIVE; CELL MEMBRANE; GTP-BINDING PROTEIN ALPHA SUBUNITS, GS; MAGNETIC RESONANCE SPECTROSCOPY; MALE; MOLECULAR SEQUENCE DATA; PEPTIDES; PHENETHYLAMINES; PROTEIN CONFORMATION; PYRIMIDINES; RADIOLIGAND ASSAY; RATS; RATS, SPRAGUE-DAWLEY; RECEPTOR, ADENOSINE A2A; RECEPTORS, PURINERGIC P1; SIGNAL TRANSDUCTION; TRIAZOLES; TRITIUM;

EID: 0033623804     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.58.1.226     Document Type: Article

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