Streptavidin-binding and -dimerizing ligands discovered by phage display, topochemistry, and structure-based design

Biomolecular Engineering

Volumn 16, Issue 1-4, 1999, Pages 57-65

  Katz, Bradley A ^a  

^a Axys Pharmaceuticals Inc   (United States)

Author keywords

Crystallographically determined pK(a) shifts; Phage display; Streptavidin binding and dimerizing ligands; Structure based drug design

Indexed keywords

AZOBENZENE DERIVATIVE; BIOTIN; CYCLOPEPTIDE; LIGAND; STREPTAVIDIN;

BINDING SITE; CONFORMATIONAL TRANSITION; CRYSTAL STRUCTURE; DIMERIZATION; DRUG DESIGN; LIGAND BINDING; PHAGE DISPLAY; PRIORITY JOURNAL; PROTEIN STRUCTURE; REVIEW; STRUCTURE ACTIVITY RELATION;

EID: 0033621522     PISSN: 13890344     EISSN: None     Source Type: Journal    
DOI: 10.1016/S1050-3862(99)00036-4     Document Type: Article

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