Leukotriene C4 is a tight-binding inhibitor of microsomal glutathione transferase-1. Effects of leukotriene pathway modifiers

Journal of Biological Chemistry

Volumn 274, Issue 4, 1999, Pages 1994-1999

  Bannenberg, Gerard ^a   Dahlén, Sven Erik ^a   Luijerink, Marjanka ^a   Lundqvist, Gerd ^a   Morgenstern, Ralf ^a  

^a KAROLINSKA INSTITUTE   (Sweden)

Author keywords

[No Author keywords available]

Indexed keywords

1 [2 METHOXY 4 [(PHENYLSULFONYLAMINO)CARBONYL]BENZYL] 1H INDAZOLE 6 CARBAMIC ACID CYCLOPENTYL ESTER; 2 CYCLOPENTYL 2 [4 (2 QUINOLINYLMETHOXY)PHENYL]ACETIC ACID; 3 [3 TERT BUTYLTHIO 1 (4 CHLOROBENZYL) 5 (2 QUINOLINYLMETHOXY) 2 INDOLYL] 2,2 DIMETHYLPROPIONIC ACID; 3 [3 TERT BUTYLTHIO 1 (4 CHLOROBENZYL) 5 ISOPROPYL 2 INDOLYL] 2,2 DIMETHYLPROPIONIC ACID; 6 (4 CARBOXYPHENYLTHIO) 5 HYDROXY 7,9,11,14 ICOSATETRAENOIC ACID; 7 [3 (4 ACETYL 3 HYDROXY 2 PROPYLPHENOXY) 2 HYDROXYPROPOXY] 4 OXO 8 PROPYL 4H 1 BENZOPYRAN 2 CARBOXYLIC ACID; GLUTATHIONE TRANSFERASE; LEUKOTRIENE C4; LEUKOTRIENE RECEPTOR BLOCKING AGENT; MICROSOME ENZYME; PIRIPROST; POBILUKAST; PRANLUKAST; UNCLASSIFIED DRUG; VERLUKAST; ZD 230487; ZILEUTON; ARACHIDONIC ACID; ENZYME INHIBITOR;

ANIMAL TISSUE; ARTICLE; ASTHMA; ENZYME ACTIVATION; ENZYME INHIBITION; ENZYME SUBSTRATE; LIVER MICROSOME; NONHUMAN; PRIORITY JOURNAL; RAT; STOICHIOMETRY; ANIMAL; DRUG ANTAGONISM; ENZYMOLOGY; MALE; METABOLISM; PROTEIN BINDING; SPRAGUE DAWLEY RAT;

ANIMALIA;

ANIMALS; ARACHIDONIC ACID; ENZYME INHIBITORS; GLUTATHIONE TRANSFERASE; LEUKOTRIENE C4; MALE; MICROSOMES, LIVER; PROTEIN BINDING; RATS; RATS, SPRAGUE-DAWLEY;

EID: 0033593117     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.274.4.1994     Document Type: Article

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