Polyunsaturated fatty acid anilides as inhibitors of acyl- COA:Cholesterol acyltransferase (ACAT)

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 14, 1999, Pages 2039-2042

  Matsuyama, Naoto ^a   Kosaka, Tetsuya ^a   Fukuhara, Mina ^a   Soda, Yasuji ^a   Mizuno, Koji ^a  

^a Azwell Inc   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

2,2 DIMETHYL N (2,4,6 TRIMETHOXYPHENYL)DODECANAMIDE; ANILIDE; CHOLESTEROL ACYLTRANSFERASE; CHOLESTEROL ACYLTRANSFERASE INHIBITOR; HYPOCHOLESTEROLEMIC AGENT; N (2,6 DIISOPROPYLPHENYL) 4,7,10,13,16,19 DOCOSAHEXAENAMIDE; N (2,6 DIISOPROPYLPHENYL)TETRADECYLTHIOACETAMIDE; POLYUNSATURATED FATTY ACID; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTERIOSCLEROSIS; ARTICLE; CELL LINE; CONTROLLED STUDY; DOG; DRUG POTENCY; ENZYME INHIBITION; HUMAN; HUMAN CELL; MICROSOME; NONHUMAN; RABBIT;

ADRENAL GLANDS; ANILIDES; ANIMALS; ANTICHOLESTEREMIC AGENTS; CELL LINE; DOCOSAHEXAENOIC ACIDS; DOGS; DRUG EVALUATION, PRECLINICAL; EICOSAPENTAENOIC ACID; ENZYME INHIBITORS; FATTY ACIDS, UNSATURATED; HUMANS; INHIBITORY CONCENTRATION 50; INTESTINES; LIVER; MACROPHAGES; MICROSOMES; RABBITS; SPECIES SPECIFICITY; STEROL O-ACYLTRANSFERASE;

EID: 0033584147     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00330-3     Document Type: Article

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