A new efficient synthesis of efaroxan

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 20, 1999, Pages 3021-3022

  Mayer, P ^a   Brunel, P ^a   Imbert, T ^a  

^a INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

[No Author keywords available]

Indexed keywords

EFAROXAN; METHANOL;

ARTICLE; CHEMICAL MODIFICATION; CHEMICAL REACTION; CYCLIZATION; DRUG SYNTHESIS; REACTION ANALYSIS;

ADRENERGIC ALPHA-ANTAGONISTS; BENZOFURANS; IMIDAZOLES;

EID: 0033581559     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00531-4     Document Type: Article

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4. Palucki, M.; Wolfe, J.P.; Buchwald, S.L. J. Amer. Chem. Soc. 1996, 118, 10333-10334.
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7. Imbert, T.; Mayer, P. Patent WO 96/35682.
8. Chapleo, C.B.; Doxey, J.C.; Stillings, M.R. Patent WO 92/05171.
9. Couture, K.; Gouverneur, V.; Mioskowski, C. Bioorg. Med. Chem. Lett. 1999, 9, 3023-3026.