Synthesis of an imidazo[1,2-e]purine-acridine heterodimer for targeting abasic sites in DNA

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 2, 1999, Pages 233-236

  Belmont, Philippe ^a   Alarcon, Karine ^a   Demeunynck, Martine ^a   Lhomme, Jean ^a  

^a CNRS   (France)

Author keywords

[No Author keywords available]

Indexed keywords

ANTINEOPLASTIC AGENT; IMIDAZO[1,2 E]PURINE ACRIDINE; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CONFORMATIONAL TRANSITION; CYCLIZATION; DRUG DESIGN; DRUG DNA BINDING; DRUG SYNTHESIS; GENE TARGETING; STRUCTURE ACTIVITY RELATION;

DNA; IMIDAZOLES; PURINES; TEMPERATURE;

EID: 0033579976     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00703-3     Document Type: Article

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10. ++1].
11. 79Br].
12. 35Cl 532.2340; Found 532.2341; UV/Vis (EtOH) λmax (1g ε) 221 (4.65), 269 (4.75), 342 (3.47), 359 (3.54), 418 (3.87).
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