Selective inactivation of protein tyrosine phosphatase PTP1B by sulfone analogue of naphthoquinone

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 2, 1999, Pages 185-186

  Seung Wook, Ham ^a   Park, Junguk ^a   Soo Jin, Lee ^a   Ji Sang, Yoo ^a  

^a Chung Ang University   (South Korea)

Author keywords

Antitumour compds; Enzyme inhibitors; Kinetics; Phosphorylaton

Indexed keywords

1,4 NAPHTHOQUINONE DERIVATIVE; MENADIONE (2 METHYL 1,4 NAPHTHOQUINONE); PROTEIN TYROSINE PHOSPHATASE; SULFONE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CATALYSIS; CONTROLLED STUDY; ENZYME ACTIVITY; ENZYME INACTIVATION; ENZYME INHIBITOR COMPLEX; PROTEIN PHOSPHORYLATION; SIGNAL TRANSDUCTION;

EID: 0033579861     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00725-2     Document Type: Article

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