New opioid affinity labels containing maleoyl moiety

Life Sciences

Volumn 65, Issue 17, 1999, Pages 1795-1805

  Szatmári, Ildikó ^a   Orosz, György ^b   Rónai, András Z ^c   Makó, Éva ^c   Medzihradszky, Kálmán ^b   Borsodi, Anna ^a  

^a INSTITUTE OF EXPERIMENTAL MEDICINE   (Hungary)

^b EÖTVÖS LORÁND UNIVERSITY   (Hungary)

^c NONE

Author keywords

Affinity labels; Ligand binding; Maleoyl peptides; Opioid receptor

Indexed keywords

DEXTRO ALANINE; ENKEPHALIN; GLYCINE; MALEOYL PEPTIDE; OPIATE RECEPTOR; PEPTIDE DERIVATIVE; UNCLASSIFIED DRUG;

AFFINITY LABELING; AMINO ACID SUBSTITUTION; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; LIGAND BINDING; MALE; MOUSE; NONHUMAN; RAT; RECEPTOR AFFINITY;

AFFINITY LABELS; AMINO ACID SUBSTITUTION; ANIMALS; BRAIN; ENKEPHALINS; GUINEA PIGS; LIGANDS; MALE; MALEATES; MEMBRANES; MICE; MUSCLE CONTRACTION; MUSCLE, SMOOTH; OPIOID PEPTIDES; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, OPIOID;

ANIMALIA; CAVIA PORCELLUS; SUS SCROFA;

EID: 0033578967     PISSN: 00243205     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0024-3205(99)00432-4     Document Type: Article

References (44)

1. J. Hughes, T.W. Smith, H.W. Kosterlitz, L.A. Fothergill, B.A. Morgan, H.R. Morris, Nature 258 577-579 (1975).
2. H. Akil, S.J. Watson, E. Young, M.E. Lewis, H. Khachaturian, J.M. Walker, Annu Rev Neurosci 7 223-255 (1984).
3. A.Z. Rónai, J. Hepp, A. Magyar, A. Borsodi, K. Medzihradszky, Pharmacology 49 121-131 (1994).
4. C.A. Gehrig, O. Prakash, G. Tóth, V.J. Hruby, NIDA Res. Monogr. 105 378-379 (1991).
5. G.W. Pasternak, The Opiate Receptors, 23-71, The Humana Press, New-Jersey (1988).
6. S. Benyhe, J. Hepp, J. Simon, A. Borsodi, K. Medzihradszky, M. Wollemann, Neuropeptides 9 225-235 (1987).
7. H.A. Ôktem, É. Varga, J. Hepp, K. Medzihradszky, A. Lajtha, A. Borsodi, Life Sci. 48 1757-1762 (1991).
8. P.S. Portoghese, J Med Chem 35 1927-1937 (1992).
9. P.S. Portoghese, D.L. Larson, J.B. Jiang, T.P. Caruso, A.E. Takemori, J. Med. Chem. 22 168-173 (1979).
10. P.S. Portoghese, D.L. Larson, L.M. Sayre, D.S. Fries, A.E. Takemori, J. Med. Chem. 23 233-234 (1980).
11. S. Benyhe, A. Ketevan, J. Simon, J. Hepp, K. Medzihradszky, A. Borsodi, Neuropeptides 31 52-59 (1997).
12. R. Venn, E.A. Barnard, J. Biol. Chem. 256 1529-1532 (1981).
13. M. Szucs, K. Di Gleria, K. Medzihradszky, FEBS 179 87-90 (1985).
14. M. Szucs, K. Di Gleria, K. Medzihradszky, Life Sci. 33 435-438 (1983).
15. F. Pasquini, C. Jomary, C. Garbay-Jaureguiberry, B.P. Roques, A. Beaudet, Eur. J. Pharmacol. 243 39-45 (1993).
16. P. Bochet, C. Icard-Liepkalns, F. Pasquini, C. Garbay-Jaureguiberry, A. Beaudet, B.P. Roques, J. Rossier, Mol. Pharmacol. 34 436-443 (1988).
17. G.W. Pasternak, H.A. Wilson, S.H. Snyder, Molecular Pharmacology 11 340-351 (1975).
18. J.R. Smith and E.J. Simon, Proc.Natl.Acad.Sci. USA 77 281-284 (1980).
19. J. Zawilska, A. Lajtha, A. Borsodi, J. Neurochem. 51 736-741 (1988).
20. G. Tóth, M. Krámer, F. Sirokmán, A. Borsodi, J. Label. Comp. RadioPharm 19 1021-1030 (1982).
21. S.T. Nevin, L. Kabasakal, F. Ötvös, G. Tóth, A. Borsodi, Neuropeptides 26 261-265 (1994).
22. D.H. Rich, P.D. Gesellchen, A. Tong, A. Cheung, C.K. Buckner, J. Med. Chem. 18 1004-1010 (1975).
23. th European Peptide Symposium, Edinburgh, 1996.
24. J. Simon, S. Benyhe, K. Abutidze, A. Borsodi, M. Szûcs, M. Wollemann, J. Neurochem. 46 695-701 (1986).
25. M.M. Bradford, Anal. Biochem. 72 248-254 (1986).
26. P.J. Munson, D. Rodbard, Anal. Biochem. 107 220-227 (1980).
27. G. Orosz, A.Z. Rónai, S. Bajusz, K. Medzihradszky, Biophys. Biochem. Res. Comm. 202 1285-1290 (1994).
28. A.Z. Rónai, A. Magyar, G. Orosz, A. Borsodi, S. Benyhe, G. Tóth, É. Makó, E. Kátay, E. Babka, K. Medzihradszky, Arch. Int Pharmacodyn. 330 361-369 (1995).
29. N. Appelmans, J.A. Carroll, M.J. Rance, E.J. Simon, J.A. Traynor, Neuropeptides 7 139-143 (1986).
30. A.Z. Rónai, J. Botyánszki, J. Hepp, K. Medzihradszky, Life Sci. 50 1371-1378 (1992).
31. S. Benyhe, J. Farkas, G. Tóth, M. Wollemann, J. Neurosci. Res. 48 249-258 (1997).
32. W.B. Bowen, S.B. Hellewell, M. Kelemen, R. Huey, D. Stewart, J. Biol. Chem. 262 13434-13439 (1987).
33. S. Benyhe, J. Hepp, M. Szucs, J. Simon, A. Borsodi, K. Medzihradszky, M. Wollemann, Neuropeptides 8 173-184 (1986).
34. M. Szûcs, S. Benyhe, A. Borsodi, M. Wollemann, G. Jancsó, J. Szécsi, K. Medzihradszky, Life Sci. 32 2777-2784 (1983).
35. S.J. Ward, D.S. Fries, D.L. Larson, P.S. Portoghese, A.E. Takemori, Eur. J. Pharmacol. 107 323-330 (1985).
36. D. Krizsán, É. Varga, S. Hosztafi, S. Benyhe, M. Szûcs, A. Borsodi, Life Sci. 48 439-451 (1991).
37. S. Fürst, A. Borsodi, T. Friedmann, S. Hosztafi, Pharmacol. Res. 25 31-32 (1992).
38. E. Hazum, K.J. Chang, P. Cuatrecasas, G.W. Pasternak, Life Sci. 28 2973-2979 (1981).
39. E.F. Hahn, M. Carroll-Buatti, G.W. Pasternak, J. Neurosci, 2 572-576 (1982).
40. A.Z. Rónai, J. Hepp, A. Magyar, A. Borsodi, K. Medzihradszky, Pharmacology 49 121-131 (1994).
41. L.M. Sayre, A.E. Takemori, P.S. Portoghese, J.Med.Chem. 24 503-506 (1983).
42. H.W. Kosterlitz, S.J. Paterson, Proc. R. Soc. London, Ser.B. 210 113-122 (1980).
43. J. Zawilska, A. Lajtha, A. Borsodi, J. Neurochem. 51 736-739 (1988).
44. C. Chen, J. Yin, J.K. Deriel, R.L. Desjarlais, L.F. Raveglia, J. Zhu, L.Y. Liu-Chen, J.Biol.Chem. 271 21422-21429 (1996).