Solid phase synthesis of β-lactams via the Staudinger reaction

Tetrahedron Letters

Volumn 40, Issue 7, 1999, Pages 1249-1252

  Singh, Rajinder ^a   Nuss, John M ^a  

^a NOVARTIS PHARMA AG   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

BETA LACTAM ANTIBIOTIC;

ARTICLE; CHEMICAL ANALYSIS; CHEMICAL REACTION; CHEMICAL STRUCTURE; DRUG SYNTHESIS;

EID: 0033547938     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(98)02672-0     Document Type: Article

References (12)

1. (a) Gallop, M. A.; Barrett, R. W.; Dower, W. J.; Fodor, S. P. A.; Gordon, E. M. J. Med. Chem. 1994, 37, 1233-1251.
2. (b) Gallop, M. A.; Barrett, R. W.; Dower, W. J.; Fodor, S. P. A.; Gordon, E. M. J. Med.Chem. 1994, 37, 1385-1401.
3. (c) Desai, M. C; Zuckermann, R. N.; Moos, W. H. Drug Development Research. 1994, 174-188.
4. Drug Discovery & Development; Williams, M.; Malick, J. B. Eds.; Humana Press: New York, 1987.
5. Terrett, N. K.; Gardner, M.; Gordon, D. W.; Kobylecki, R. J.; Steele, J. Tetrahedron. 1995, 51, 8135-8173.
6. For recent reviews see. (a) The Chemistry of β-Lactams; Page, M. I. Ed.; Cambridge University Press, 1992.
7. (b) The Organic Chemistry of β-Lactams; Georg, G. I. Ed.; VCH Publishers, 1993.
8. Look, G. C.; Murphy, M. M.; Campbell, D. A.; Gallop, M. A. Tetrahedron Lett. 1995, 36, 2937-2940.
9. Bose, A. K.; Lal, B.; Manhas, M. S. Tetrahedron Lett. 1974, 2633.
10. (a) Schkeryantz, J. M.; Danishefsky, S. J. J. Am. Chem. Soc. 1995, 117, 4722-4723.
11. (b) Plattner, J. J.; Gless, R. D.; Rapoport, H. J. Am. Chem. Soc. 1972, 94, 8613-8615.
12. +, 100%).