Synthesis of boron-containing cholesterol derivatives for incorporation into unilamellar liposomes and evaluation as potential agents for BNCT

Tetrahedron

Volumn 55, Issue 37, 1999, Pages 11177-11186

  Feakes, Debra A ^a   Spinler, Jennifer K ^a   Harris, Fred R ^a  

^a Texas State University   (United States)

Author keywords

Boron and Compounds; Carborane; Esters; Ethers

Indexed keywords

1 (6 (1,2 DICARBADODECABORAN 1 YL)HEXOXYCHOLESTEROL; BORON; CARBORANE DERIVATIVE; CHOLESTEROL DERIVATIVE; CHOLESTERYL 6 (1,2 DICARBADODECABORAN 1 YL)HEXANOATE; ESTER; ETHER DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CANCER; DRUG DELIVERY SYSTEM; DRUG SPECIFICITY; DRUG STABILITY; DRUG SYNTHESIS; NEUTRON CAPTURE THERAPY; PRIORITY JOURNAL; TUMOR CELL DESTRUCTION;

EID: 0033543490     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4020(99)00640-7     Document Type: Article

References (21)

1. Fairchild, R. G.; Bond, V. P. J. Radiat. Oncol. Biol. Phys. 1985, 11, 831-840.
2. Shelly, K.; Feakes, D. A.; Hawthorne, M. F.; Schmidt, P. G.; Krisch, T. A.; Bauer, W. F. Proc. Natl. Acad. Sci. USA 1992, 89, 9039-9043.
3. Feakes, D. A.; Shelly, K.; Knobler, C. B.; Hawthorne, M. F. Proc. Natl. Acad. Sci. USA 1994, 91, 3029-3033.
4. Straubinger, R. M.; Papahadjopoulos, D.; Hong, K. Biochemistry 1990, 29, 4929-4939.
5. Wallingford, R. H.; Williams, L. E. J. Nucl. Med. 1985, 26, 1180-1185.
6. Proffitt, R. T.; Williams, L. E.; Presant, C.; Tin, G. W.; Uliana, J. A.; Gamble, R. C.; Baldeschwieler, J. D. J. Nucl. Med. 1983, 24, 45-55.
7. Coderre, J. A.; Kalef-Ezra, J. A.; Fairchild, R. G.; Micca, P. L.; Reinstein, L. E.; Glass, J. D. Cancer Res. 1988, 48, 6313-6316.
8. Clendonen, N. R.; Barth, R. F.; Gordon, W. A.; Goodman, J. H.; Alam, F.; Staubus, A. E.; Boesel, C. P.; Yates, A. J.; Moeschberger, M. L.; Fairchild, R. G.; Kalef-Ezra, J. A. Neurosurgery 1990, 26, 47-55.
9. Gabel, D.; Holstein, H.; Larsson, B.; Gille, L.; Ericson, G.; Sacker, D.; Som, P.; Fairchild, R. G. Cancer Res. 1987, 47, 5451-5454.
10. Slatkin, D.; Micca, P.; Forman, A.; Gabel, D.; Wielopolski, L.; Fairchild, R. G. Biochem. Pharmacol. 1986, 35, 1771-1776.
11. Soloway, A. H.; Hatanaka, H.; Davis, M. A. J. Medicinal Chem. 1967, 10, 714-717.
12. Sweet, W. H.; Soloway, A. H.; Wright, R. L. J. Pharmacol. Exp. Ther. 1962, 137, 263-266.
13. Deamer, D. W.; Uster, P. S. In Lipsomes;Ostro, M. J., Ed.; Dekker: New York, 1983, pp. 31-35.
14. Feakes, D. A.; Shelly, K.; Hawthorne, M. F. Proc. Natl. Acad. Sci. USA 1995, 92, 1367-1370.
15. Straubinger, R. M.; Hong, K.; Friend, D. S.; Paphadjopoulos, D. Cell 1983, 32, 1069-1079.
16. Fraley, R.; Straubinger, R.; Rule, G.; Springer, L.; Papahadjopoulos, D. Biochemistry 1981, 20, 6978-6987.
17. Macaulay, S. R. J. Org. Chem. 1980, 45, 734-735.
18. Srivastava, R. R.; Kabalka, G. W. J. Org. Chem. 1997, 62, 8730-8734.
19. Hawthorne, M. F.; Andrews, T. D.; Garrett, P. M.; Olsen, F. P.; Reintjes, M.; Tebbe, F. N.; Warren, L. F. Wegner, P. A.; Young, D. C. Inorg. Synth. 1967, 10, 91-118.
20. Tomita, H.; Luu, H.; Onak, T. Inorg. Chem. 1991, 30, 812-815.
21. Hawthorne, M. F.; Pilling, R. L. Inorg. Synth. 1967, 9, 16-19.