Enantioselective synthesis of 4-substituted phenylalanines by cross- coupling reactions

Tetrahedron Letters

Volumn 40, Issue 2, 1999, Pages 213-216

  Firooznia, F ^a   Gude, C ^a   Chan, K ^a   Marcopulos, N ^a   Satoh, Y ^a  

^a NOVARTIS PHARMA AG   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

BORON DERIVATIVE; HALIDE; IODINE DERIVATIVE; N TERT BUTYLOXYCARBONYL(4 PINACOLYLBORONO)PHENYLALANINE METHYL ESTER; PALLADIUM; PHENYLALANINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CATALYST; ENANTIOMER; RACEMIC MIXTURE; SYNTHESIS;

EID: 0033534511     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(98)02272-2     Document Type: Article

References (10)

1. For a recent review, see: Miyaura N. Suzuki A. Chem. Rev. 95 1995 2457
2. Satoh Y. Gude C. Chan K. Firooznia F. Tetrahedron Lett. 38 1997 7645
3. Subsequent to our report (ref. 2), a recent publication described a synthesis of 4-aryl-phenylalanines by Stille cross-coupling reactions of N-Boc-4-trimethylstannylphenylalanine methyl ester : Morera E. Ortar G. Synlett 1997 1403
4. Firooznia F. Gude C. Chan K. Satoh Y. Tetrahedron Lett. 39 1998 3985
5. Fitzi R. Seebach D. Tetrahedron 44 1988 5277
6. Roberts D.C. Suda K. Samanen J. Kemp D.S. Tetrahedron Lett. 21 1980 3435 and references cited therein
7. For an alternative approach to the synthesis of 4-borono- L -phenylalanine see: Malan C. Morin C. Synlett 1996 167
8. Ishiyama T. Itoh Y. Kitano T. Miyaura N. Tetrahedron Lett. 38 1997 3447
9. Ishiyama T. Murata M. Miyaura N. J. Org. Chem. 60 1995 7508
10. Murata M. Watanabe S. Masuda Y. J. Org. Chem. 62 1997 6458