A new synthetic route to 10β-alkyldeoxoartemisinins

Tetrahedron Letters

Volumn 40, Issue 49, 1999, Pages 8543-8545

  Ma, Jingyuan ^a   Katz, Esther ^b   Ziffer, Herman ^a  

^a NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

^b ISRAEL INSTITUTE FOR BIOLOGICAL RESEARCH   (Israel)

Author keywords

Artemisinin; Lactol acetate; Titanium tetrachloride; Trimethyloxy group

Indexed keywords

ARTEMISININ; ARTEMISININ DERIVATIVE; FUNCTIONAL GROUP; TITANIUM DERIVATIVE;

ARTICLE; DERIVATIZATION; DRUG SYNTHESIS; REDUCTION;

EID: 0033520961     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(99)01824-9     Document Type: Article

References (11)

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10. 3 solution, dried and evaporated. The residue was purified by chromatography on silica gel to give 150 mg white solid in 76% yield.
11. 1H NMR spectra, mass spectra and microanalysis or high solution mass spectra.