메뉴 건너뛰기




Volumn 85, Issue 6, 1999, Pages 257-262

Rifampicin treatment greatly increases the apparent oral clearance of quinidine

Author keywords

[No Author keywords available]

Indexed keywords

QUINIDINE; QUINIDINE SULFATE; RIFAMPICIN; TOLBUTAMIDE;

EID: 0033452495     PISSN: 09019928     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1600-0773.1999.tb02019.x     Document Type: Article
Times cited : (25)

References (38)
  • 1
    • 0027523486 scopus 로고
    • Use of single sample clearance estimates of cytochrome P450 substrates to characterize human hepatic CYP status in vivo
    • Bachmann, K. A. & L. Jauregui: Use of single sample clearance estimates of cytochrome P450 substrates to characterize human hepatic CYP status in vivo. Xenobiotica 1993, 23, 307-315.
    • (1993) Xenobiotica , vol.23 , pp. 307-315
    • Bachmann, K.A.1    Jauregui, L.2
  • 2
    • 0031959294 scopus 로고    scopus 로고
    • The area under the plasma concentration-time curve for oral midazolam is 400-fold larger during treatment with itraconazole than with rifampicin
    • Backman, J. T., K. T. Kivistö, K. T. Olkkola & P. J. Neuvonen: The area under the plasma concentration-time curve for oral midazolam is 400-fold larger during treatment with itraconazole than with rifampicin. Eur. J. Clin. Pharmacol. 1998, 54, 53-58.
    • (1998) Eur. J. Clin. Pharmacol. , vol.54 , pp. 53-58
    • Backman, J.T.1    Kivistö, K.T.2    Olkkola, K.T.3    Neuvonen, P.J.4
  • 3
    • 0030068752 scopus 로고    scopus 로고
    • Rifampin drastically reduces plasma concentrations and effects of oral midazolam
    • Backman, J. T., K. T. Olkkola & P. J. Neuvonen: Rifampin drastically reduces plasma concentrations and effects of oral midazolam. Clin. Pharmacol. Therap. 1996, 59, 7-13.
    • (1996) Clin. Pharmacol. Therap. , vol.59 , pp. 7-13
    • Backman, J.T.1    Olkkola, K.T.2    Neuvonen, P.J.3
  • 5
    • 0031900997 scopus 로고    scopus 로고
    • Role of P-glycoprotein as a secretory mechanism in quinidine absorption from rat small intestine
    • Emi, Y., D. Tsunashima, K. Ogawara, K. Higaki, & T. Kimura: Role of P-glycoprotein as a secretory mechanism in quinidine absorption from rat small intestine. J. Pharm. Sci. 1998, 87, 295-299.
    • (1998) J. Pharm. Sci. , vol.87 , pp. 295-299
    • Emi, Y.1    Tsunashima, D.2    Ogawara, K.3    Higaki, K.4    Kimura, T.5
  • 6
    • 0031931510 scopus 로고    scopus 로고
    • The induction effect of rifampicin on activity of mephenytoin 4'-hydroxylase related to Ml mutation of CYP2C19 and gene dose
    • Feng, H. J., S. L. Huang, W Wang & H. H. Zhou: The induction effect of rifampicin on activity of mephenytoin 4'-hydroxylase related to Ml mutation of CYP2C19 and gene dose. Brit. J. Clin. Pharmacol. 1998, 45, 27-29.
    • (1998) Brit. J. Clin. Pharmacol. , vol.45 , pp. 27-29
    • Feng, H.J.1    Huang, S.L.2    Wang, W.3    Zhou, H.H.4
  • 7
    • 0030712276 scopus 로고    scopus 로고
    • Validation of the five-drug "Pittsburgh cocktail" approach for assessment of selective regulation of drug-metabolizing enzymes
    • Frye, R. F., G. R. Matzke, A. Adedoyin, J. A. Porter, & R. A. Branch: Validation of the five-drug "Pittsburgh cocktail" approach for assessment of selective regulation of drug-metabolizing enzymes. Clin. Pharmacol. Therap. 1997, 62, 365-376.
    • (1997) Clin. Pharmacol. Therap. , vol.62 , pp. 365-376
    • Frye, R.F.1    Matzke, G.R.2    Adedoyin, A.3    Porter, J.A.4    Branch, R.A.5
  • 11
    • 0022467917 scopus 로고
    • Oxidation of quinidine by human liver cytochrome P-450
    • Guengerich, F. P., D. Muller Enoch & I. A. Blair: Oxidation of quinidine by human liver cytochrome P-450. Mal. Pharmacol. 1986, 30, 287-295.
    • (1986) Mal. Pharmacol. , vol.30 , pp. 287-295
    • Guengerich, F.P.1    Muller Enoch, D.2    Blair, I.A.3
  • 12
    • 0032698375 scopus 로고    scopus 로고
    • Quantitative determination of tolbutamide and its metabolites in human plasma and urine by high-performance liquid chromatography and UV detection
    • in press
    • Hansen, L. L. & K. Brøsen: Quantitative determination of tolbutamide and its metabolites in human plasma and urine by high-performance liquid chromatography and UV detection. Ther. Drug Monit. 1999, in press.
    • (1999) Ther. Drug Monit.
    • Hansen, L.L.1    Brøsen, K.2
  • 13
    • 0026457407 scopus 로고
    • Bio-availability of cyclosporine with concomitant rifampin administration is markedly less than predicted by hepatic enzyme induction
    • Hebert, M.F., J. P. Roberts, T. Prueksaritanont & L. Z. Benet: Bio-availability of cyclosporine with concomitant rifampin administration is markedly less than predicted by hepatic enzyme induction. Clin. Pharmacol. Therap. 1992, 52, 453-457.
    • (1992) Clin. Pharmacol. Therap. , vol.52 , pp. 453-457
    • Hebert, M.F.1    Roberts, J.P.2    Prueksaritanont, T.3    Benet, L.Z.4
  • 14
    • 0029972195 scopus 로고    scopus 로고
    • The nifedipine-rifampin interaction. Evidence for induction of gut wall metabolism
    • Holtbecker, N., M. F. Fromm, H. K. Kroemer, E. E. Ohnhaus & H. Heidemann: The nifedipine-rifampin interaction. Evidence for induction of gut wall metabolism. Drug Metab. Disp. 1996, 24, 1121-1123.
    • (1996) Drug Metab. Disp. , vol.24 , pp. 1121-1123
    • Holtbecker, N.1    Fromm, M.F.2    Kroemer, H.K.3    Ohnhaus, E.E.4    Heidemann, H.5
  • 15
    • 0030897275 scopus 로고    scopus 로고
    • Use of probe drugs as predictors of drug metabolism in humans
    • Kivistö, K. T. & H. K. Kroemer: Use of probe drugs as predictors of drug metabolism in humans. J. Clin. Pharmacol. 1997, 37, 40-48.
    • (1997) J. Clin. Pharmacol. , vol.37 , pp. 40-48
    • Kivistö, K.T.1    Kroemer, H.K.2
  • 16
    • 0026464616 scopus 로고
    • Identification of rifampin-inducible P450IIIA4 (CYP3A4) in human small bowel enterocytes
    • Kolars, J. C., P. Schmiedlin Ren, J. D. Schuetz, C. Fang & P B. Watkins: Identification of rifampin-inducible P450IIIA4 (CYP3A4) in human small bowel enterocytes. J. Clin. Invest. 1992, 90, 1871-1878.
    • (1992) J. Clin. Invest. , vol.90 , pp. 1871-1878
    • Kolars, J.C.1    Schmiedlin Ren, P.2    Schuetz, J.D.3    Fang, C.4    Watkins, P.B.5
  • 18
    • 0028131815 scopus 로고
    • Simultaneous determination of urinary free cortisol and 6 beta- hydroxycortisol by high-performance liquid chromatography to measure human CYP3A activity
    • Lykkesfeldt, J., S. Loft & H. E. Poulsen: Simultaneous determination of urinary free cortisol and 6 beta- hydroxycortisol by high-performance liquid chromatography to measure human CYP3A activity. J. Chromatogr. B. Biomed. Appl. 1994, 660, 23-29.
    • (1994) J. Chromatogr. B. Biomed. Appl. , vol.660 , pp. 23-29
    • Lykkesfeldt, J.1    Loft, S.2    Poulsen, H.E.3
  • 19
    • 0030611023 scopus 로고    scopus 로고
    • The effect of single dose of rifampicin on the pharmacokinetics of oral nifedipine
    • Ndanusa, B. U., A. Mustapha & A. I. Abdu: The effect of single dose of rifampicin on the pharmacokinetics of oral nifedipine. J. Pharm. Biomed. Anal. 1997, 15, 1571-1575.
    • (1997) J. Pharm. Biomed. Anal. , vol.15 , pp. 1571-1575
    • Ndanusa, B.U.1    Mustapha, A.2    Abdu, A.I.3
  • 20
    • 0027941975 scopus 로고
    • Determination of quinidine, dihydroquinidine, (3S)-3- hydroxyquinidine and quinidine N-oxide in plasma and urine by high-performance liquid chromatography
    • Nielsen, F., K. K. Nielsen & K. Brosen: Determination of quinidine, dihydroquinidine, (3S)-3- hydroxyquinidine and quinidine N-oxide in plasma and urine by high-performance liquid chromatography. J. Chromatogr. B. Biomed. Appl. 1994, 660, 103-110.
    • (1994) J. Chromatogr. B. Biomed. Appl. , vol.660 , pp. 103-110
    • Nielsen, F.1    Nielsen, K.K.2    Brosen, K.3
  • 21
    • 0032947029 scopus 로고    scopus 로고
    • In vitro metabolism of quinidine: The (3S)-3-hydroxylation is a specific marker reaction for cytochrome P4503A4 activity in human liver microsomes
    • Nielsen, T. L., B. B. Rasmussen, J.-P. Flinois, P. Beaune & K. Brøsen: In vitro metabolism of quinidine: the (3S)-3-hydroxylation is a specific marker reaction for cytochrome P4503A4 activity in human liver microsomes. J. Pharmacol. Exp. Therap. 1999, 289, 31-37.
    • (1999) J. Pharmacol. Exp. Therap. , vol.289 , pp. 31-37
    • Nielsen, T.L.1    Rasmussen, B.B.2    Flinois, J.-P.3    Beaune, P.4    Brøsen, K.5
  • 22
    • 8044244218 scopus 로고    scopus 로고
    • Theophylline has no advantages over caffeine as a putative model drug for assessing CYPIA2 activity in humans
    • Rasmussen, B. B. & K. Brøsen: Theophylline has no advantages over caffeine as a putative model drug for assessing CYPIA2 activity in humans. Br. J. Clin. Pharmacol. 1997, 43, 253-258.
    • (1997) Br. J. Clin. Pharmacol. , vol.43 , pp. 253-258
    • Rasmussen, B.B.1    Brøsen, K.2
  • 23
    • 0021149092 scopus 로고
    • Theophylline-rifampicin interaction: Non-selective induction of theophylline metabolic pathways
    • Robson, R. A., J. O. Miners, L. H. Wing & D. J. Birkett: Theophylline-rifampicin interaction: Non-selective induction of theophylline metabolic pathways. Brit. J. Clin. Pharmacol. 1984, 18, 445-448.
    • (1984) Brit. J. Clin. Pharmacol. , vol.18 , pp. 445-448
    • Robson, R.A.1    Miners, J.O.2    Wing, L.H.3    Birkett, D.J.4
  • 24
    • 0024336503 scopus 로고
    • S-mephenytoin hydroxylation phenotypes in a Swedish population determined after coadministration with debrisoquin
    • Sanz, E. J., T. Villen, C. Alm & L. Bertilsson: S-mephenytoin hydroxylation phenotypes in a Swedish population determined after coadministration with debrisoquin. Clin. Pharmacol Therap. 1989, 45, 495-499.
    • (1989) Clin. Pharmacol Therap. , vol.45 , pp. 495-499
    • Sanz, E.J.1    Villen, T.2    Alm, C.3    Bertilsson, L.4
  • 25
    • 0030059953 scopus 로고    scopus 로고
    • Modulators and substrates of P-glycoprotein and cytochrome P4503A coordinately up-regulate these proteins in human colon carcinoma cells
    • Schuetz, E. G., W. T. Beck & J. D. Schuetz: Modulators and substrates of P-glycoprotein and cytochrome P4503A coordinately up-regulate these proteins in human colon carcinoma cells. Mol. Pharmacol. 1996, 49, 311-318.
    • (1996) Mol. Pharmacol. , vol.49 , pp. 311-318
    • Schuetz, E.G.1    Beck, W.T.2    Schuetz, J.D.3
  • 26
    • 0028237729 scopus 로고
    • Interindividual variations in human liver cytochrome P-450 enzymes involved in the oxidation of drugs, carcinogens and toxic chemicals: Studies with liver microsomes of 30 Japanese and 30 Caucasians
    • Shimada, H., T. Yamazaki, M. Mimura, Y. Inui & F. P. Guengerich: Interindividual variations in human liver cytochrome P-450 enzymes involved in the oxidation of drugs, carcinogens and toxic chemicals: studies with liver microsomes of 30 Japanese and 30 Caucasians. J. Pharm. Exp. Therap. 1994, 270, 414-423.
    • (1994) J. Pharm. Exp. Therap. , vol.270 , pp. 414-423
    • Shimada, H.1    Yamazaki, T.2    Mimura, M.3    Inui, Y.4    Guengerich, F.P.5
  • 27
    • 0030035251 scopus 로고    scopus 로고
    • Use of salivary caffeine tests to assess the inducer effect of a drug on hepatic metabolism
    • Soto, J., J. A. Sacristan & M. J. Alsar: Use of salivary caffeine tests to assess the inducer effect of a drug on hepatic metabolism. Ann. Pharmacother. 1996, 30, 736-739.
    • (1996) Ann. Pharmacother. , vol.30 , pp. 736-739
    • Soto, J.1    Sacristan, J.A.2    Alsar, M.J.3
  • 29
    • 0025264682 scopus 로고
    • Validation of the tolbutamide metabolic ratio for population screening with use of sulfaphenazole to produce model phenotypic poor metabolizers
    • Veronese, M. E., J. O. Miners, D. Randles, D. Gregov & D. J. Birkett: Validation of the tolbutamide metabolic ratio for population screening with use of sulfaphenazole to produce model phenotypic poor metabolizers. Clin. Pharmacol. Therap. 1990, 47, 403-411.
    • (1990) Clin. Pharmacol. Therap. , vol.47 , pp. 403-411
    • Veronese, M.E.1    Miners, J.O.2    Randles, D.3    Gregov, D.4    Birkett, D.J.5
  • 31
    • 0029028792 scopus 로고
    • Overlapping substrate specificities and tissue distribution of cytochrome P450 3A and P-glycoprotein: Implications for drug delivery and activity in cancer chemotherapy
    • Wacher, V. J., C. Y. Wu & L. Z. Benet: Overlapping substrate specificities and tissue distribution of cytochrome P450 3A and P-glycoprotein: implications for drug delivery and activity in cancer chemotherapy. Mol. Carcinogen. 1995, 13, 129-134.
    • (1995) Mol. Carcinogen. , vol.13 , pp. 129-134
    • Wacher, V.J.1    Wu, C.Y.2    Benet, L.Z.3
  • 32
    • 0028071759 scopus 로고
    • Noninvasive tests of CYP3A enzymes
    • Watkins, P. B.: Noninvasive tests of CYP3A enzymes. Pharmacogenetics 1994, 4, 171-184.
    • (1994) Pharmacogenetics , vol.4 , pp. 171-184
    • Watkins, P.B.1
  • 33
    • 0024556650 scopus 로고
    • Erythromycin breath test as an assay of glucocorticoid-inducible liver cytochromes P-450. Studies in rats and patients
    • Watkins, P. B., S. A. Murray, L. G. Winkelman, D. M. Heuman, S. A. Wrighton & P. S. Guzelian: Erythromycin breath test as an assay of glucocorticoid-inducible liver cytochromes P-450. Studies in rats and patients. J. Clin. Invest. 1989, 83, 688-697.
    • (1989) J. Clin. Invest. , vol.83 , pp. 688-697
    • Watkins, P.B.1    Murray, S.A.2    Winkelman, L.G.3    Heuman, D.M.4    Wrighton, S.A.5    Guzelian, P.S.6
  • 34
    • 0028890301 scopus 로고
    • The influence of rifampin treatment on caffeine clearance in healthy man
    • Wietholtz, H., T. Zysset, H. U. Marschall, K. Generet & S. Matern: The influence of rifampin treatment on caffeine clearance in healthy man. J. Hepatol. 1995, 22, 78-81.
    • (1995) J. Hepatol. , vol.22 , pp. 78-81
    • Wietholtz, H.1    Zysset, T.2    Marschall, H.U.3    Generet, K.4    Matern, S.5
  • 35
    • 0028820208 scopus 로고
    • Differentiation of absorption and first-pass gut and hepatic metabolism in humans: Studies with cyclosporine
    • Wu, C. Y., L. Z. Benet, M. F. Hebert, S. K. Gupta, M. Rowland, D. Y. Gomez & V. J. Wacher: Differentiation of absorption and first-pass gut and hepatic metabolism in humans: studies with cyclosporine. Clin. Pharmacol. Therap. 1995, 58, 492-497.
    • (1995) Clin. Pharmacol. Therap. , vol.58 , pp. 492-497
    • Wu, C.Y.1    Benet, L.Z.2    Hebert, M.F.3    Gupta, S.K.4    Rowland, M.5    Gomez, D.Y.6    Wacher, V.J.7
  • 36
  • 37
    • 0016758480 scopus 로고
    • Induction of drug metabolism in man after rifampicin treatment measured by increased hexobarbital and tolbutamide clearance
    • Zilly, W., D. D. Breimer & E. Richter: Induction of drug metabolism in man after rifampicin treatment measured by increased hexobarbital and tolbutamide clearance. Eur. J. Clin. Pharmacol. 1975, 9, 219-227.
    • (1975) Eur. J. Clin. Pharmacol. , vol.9 , pp. 219-227
    • Zilly, W.1    Breimer, D.D.2    Richter, E.3
  • 38
    • 0017596185 scopus 로고
    • Stimulation of drug metabolism by rifampicin in patients with cirrhosis or cholestasis measured by increased hexobarbital and tolbutamide clearance
    • Zilly, W, D. D. Breimer & E. Richter: Stimulation of drug metabolism by rifampicin in patients with cirrhosis or cholestasis measured by increased hexobarbital and tolbutamide clearance. Eur. J. Clin. Pharmacol. 1977, 11, 287-293.
    • (1977) Eur. J. Clin. Pharmacol. , vol.11 , pp. 287-293
    • Zilly, W.1    Breimer, D.D.2    Richter, E.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.