Synthesis, binding affinity and selectivity of new β1- and β2- adrenoceptor blockers

Farmaco

Volumn 54, Issue 11-12, 1999, Pages 713-720

  Brizzi, Vittorio ^a   Francioli, Marco ^a   Brufani, Mario ^b   Filocamo, Luigi ^b   Bruni, Giancarlo ^a   Massarelli, Paola ^a  

^a UNIVERSITY OF SIENA   (Italy)

^b SAPIENZA UNIVERSITY OF ROME   (Italy)

Author keywords

Adrenoceptor blockers; Antihypertensive; Cardiovascular diseases; Sesamol

Indexed keywords

3 ISOPROPYLAMINO 1 (7 METHYL 4 INDANYLOXY) 2 BUTANOL; BETA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; BETA 2 ADRENERGIC RECEPTOR BLOCKING AGENT; PROPRANOLOL; SESAMOL DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BETA ADRENERGIC RECEPTOR BLOCKING; BINDING AFFINITY; DRUG PURIFICATION; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; RAT;

ADRENERGIC BETA-ANTAGONISTS; ANIMALS; LUNG; MAGNETIC RESONANCE SPECTROSCOPY; MALE; PROPANOLAMINES; PROTEIN BINDING; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, ADRENERGIC, BETA-1; RECEPTORS, ADRENERGIC, BETA-2; SPECTROPHOTOMETRY, INFRARED;

EID: 0033436358     PISSN: 0014827X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-827X(99)00077-4     Document Type: Article

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