Synthesis of 1,2-benzisothiazole derivatives and investigation of their putative histaminergic activity

Farmaco

Volumn 54, Issue 11-12, 1999, Pages 740-746

  Morini, Giovanni ^a   Pozzoli, Cristina ^a   Adami, Maristella ^a   Poli, Enzo ^a   Coruzzi, Gabriella ^a  

^a UNIVERSITY OF PARMA   (Italy)

Author keywords

1,2 Benzisothiazole derivatives; Duodenum; Gangliomimetic effect; Gastric mucosa; Histamine receptors; Papillary muscle

Indexed keywords

1 (1,2 BENZISOTHIAZOL 3 YL)ETHYLAMINE; 1,2 BENZISOTHIAZOLE DERIVATIVE; ATROPINE; FAMOTIDINE; HEXAMETHONIUM; HISTAMINE RECEPTOR; HISTAMINERGIC RECEPTOR AFFECTING AGENT; MEPYRAMINE; N,N,N TRIMETHYL 2 (1,2 BENZISOTHIAZOL 3 YL)ETHYLAMMONIUM IODIDE; NICOTINIC RECEPTOR; ONDANSETRON; SEROTONIN 3 RECEPTOR; TETRODOTOXIN; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG EFFECT; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; DUODENUM; GUINEA PIG; HEART PAPILLARY MUSCLE; INOTROPISM; INTESTINE CONTRACTION; MALE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; STOMACH MUCOSA;

ANIMALS; DUODENUM; GASTRIC MUCOSA; GUINEA PIGS; HISTAMINE H1 ANTAGONISTS; MUSCLE CONTRACTION; THIAZOLES;

EID: 0033430301     PISSN: 0014827X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-827X(99)00093-2     Document Type: Article

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