Thermal ring contraction of 3H-1,4-benzo- diazepines into quinazolines

Heterocycles

Volumn 51, Issue 10, 1999, Pages 2407-2413

  Kaname, Mamoru ^a   Tsuchiya, Takashi ^a   Sashida, Haruki ^a  

^a HOKURIKU UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

BENZODIAZEPINE DERIVATIVE; QUINAZOLINE DERIVATIVE;

ARTICLE; DRUG STRUCTURE; DRUG TRANSFORMATION;

EID: 0033214276     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/com-99-8639     Document Type: Article

References (17)

1. M. B. Stringer, V. Candeloro, J. H. Bowie, R. H. Prager, L. M. Engelhardt, and A. H. White, J. Chem. Soc., Perkin Trans. 1, 1984, 2529; M. Flammang, C. R. Seances Acad. Sci., Ser C, 1980, 290, 349 (Chem. Abstr., 1980, 93, 167330q); M. Flammang and C. G. Wermuth, C. R. Seances Acad. Sci., Ser C, 1980, 290, 361 (Chem. Abstr., 1980, 93, 203556d); Ch. K. Reddy, P. S. N. Reddy, and C. V. Ratnam, Indian J. Chem., Sect. B, 1985, 24B, 695 (Chem. Abstr., 1986, 105, 172419w).
2. M. B. Stringer, V. Candeloro, J. H. Bowie, R. H. Prager, L. M. Engelhardt, and A. H. White, J. Chem. Soc., Perkin Trans. 1, 1984, 2529; M. Flammang, C. R. Seances Acad. Sci., Ser C, 1980, 290, 349 (Chem. Abstr., 1980, 93, 167330q); M. Flammang and C. G. Wermuth, C. R. Seances Acad. Sci., Ser C, 1980, 290, 361 (Chem. Abstr., 1980, 93, 203556d); Ch. K. Reddy, P. S. N. Reddy, and C. V. Ratnam, Indian J. Chem., Sect. B, 1985, 24B, 695 (Chem. Abstr., 1986, 105, 172419w).
3. M. B. Stringer, V. Candeloro, J. H. Bowie, R. H. Prager, L. M. Engelhardt, and A. H. White, J. Chem. Soc., Perkin Trans. 1, 1984, 2529; M. Flammang, C. R. Seances Acad. Sci., Ser C, 1980, 290, 349 (Chem. Abstr., 1980, 93, 167330q); M. Flammang and C. G. Wermuth, C. R. Seances Acad. Sci., Ser C, 1980, 290, 361 (Chem. Abstr., 1980, 93, 203556d); Ch. K. Reddy, P. S. N. Reddy, and C. V. Ratnam, Indian J. Chem., Sect. B, 1985, 24B, 695 (Chem. Abstr., 1986, 105, 172419w).
4. M. B. Stringer, V. Candeloro, J. H. Bowie, R. H. Prager, L. M. Engelhardt, and A. H. White, J. Chem. Soc., Perkin Trans. 1, 1984, 2529; M. Flammang, C. R. Seances Acad. Sci., Ser C, 1980, 290, 349 (Chem. Abstr., 1980, 93, 167330q); M. Flammang and C. G. Wermuth, C. R. Seances Acad. Sci., Ser C, 1980, 290, 361 (Chem. Abstr., 1980, 93, 203556d); Ch. K. Reddy, P. S. N. Reddy, and C. V. Ratnam, Indian J. Chem., Sect. B, 1985, 24B, 695 (Chem. Abstr., 1986, 105, 172419w).
5. M. B. Stringer, V. Candeloro, J. H. Bowie, R. H. Prager, L. M. Engelhardt, and A. H. White, J. Chem. Soc., Perkin Trans. 1, 1984, 2529; M. Flammang, C. R. Seances Acad. Sci., Ser C, 1980, 290, 349 (Chem. Abstr., 1980, 93, 167330q); M. Flammang and C. G. Wermuth, C. R. Seances Acad. Sci., Ser C, 1980, 290, 361 (Chem. Abstr., 1980, 93, 203556d); Ch. K. Reddy, P. S. N. Reddy, and C. V. Ratnam, Indian J. Chem., Sect. B, 1985, 24B, 695 (Chem. Abstr., 1986, 105, 172419w).
6. M. B. Stringer, V. Candeloro, J. H. Bowie, R. H. Prager, L. M. Engelhardt, and A. H. White, J. Chem. Soc., Perkin Trans. 1, 1984, 2529; M. Flammang, C. R. Seances Acad. Sci., Ser C, 1980, 290, 349 (Chem. Abstr., 1980, 93, 167330q); M. Flammang and C. G. Wermuth, C. R. Seances Acad. Sci., Ser C, 1980, 290, 361 (Chem. Abstr., 1980, 93, 203556d); Ch. K. Reddy, P. S. N. Reddy, and C. V. Ratnam, Indian J. Chem., Sect. B, 1985, 24B, 695 (Chem. Abstr., 1986, 105, 172419w).
7. M. B. Stringer, V. Candeloro, J. H. Bowie, R. H. Prager, L. M. Engelhardt, and A. H. White, J. Chem. Soc., Perkin Trans. 1, 1984, 2529; M. Flammang, C. R. Seances Acad. Sci., Ser C, 1980, 290, 349 (Chem. Abstr., 1980, 93, 167330q); M. Flammang and C. G. Wermuth, C. R. Seances Acad. Sci., Ser C, 1980, 290, 361 (Chem. Abstr., 1980, 93, 203556d); Ch. K. Reddy, P. S. N. Reddy, and C. V. Ratnam, Indian J. Chem., Sect. B, 1985, 24B, 695 (Chem. Abstr., 1986, 105, 172419w).
8. L. H. Sternbach, Angew. Chem., Int. Ed. Engl., 1971, 10, 34; G. Mohiuddin, P. S. Reddy, K. Ahmed, and C. V. Ratnam, Heterocycles, 1986, 24, 3489.
9. L. H. Sternbach, Angew. Chem., Int. Ed. Engl., 1971, 10, 34; G. Mohiuddin, P. S. Reddy, K. Ahmed, and C. V. Ratnam, Heterocycles, 1986, 24, 3489.
10. S. C. Bell and S. J. Childress, J. Org. Chem., 1962, 27, 1691.
11. L. H. Sternbach, E. Reeder, A. Stempel, and A. L. Rachlin, J. Org. Chem., 1964, 29, 332.
12. D. W. Combs, J. B. Press, D. Mulvey, Y.G-Nunez, and S. C. Bell, J. Heterocycl. Chem., 1986, 23, 1263.
13. H. Sashida, A. Fujii, H. Sawanishi, and T. Tsuchiya, Heterocycles, 1986, 24, 2147; H. Sashida, A. Fujii, and T. Tsuchiya, Chem. Pharm. Bull., 1987, 35, 3182.
14. H. Sashida, A. Fujii, H. Sawanishi, and T. Tsuchiya, Heterocycles, 1986, 24, 2147; H. Sashida, A. Fujii, and T. Tsuchiya, Chem. Pharm. Bull., 1987, 35, 3182.
15. K. W. Breukink, L. H. Krol, P. E. Verkade, and B. M. Wepster, Rec. Trav. Chim., 1957, 76, 401 (Chem. Abstr., 1957, 51, 15527d).
16. K. W. Breukink, L. H. Krol, P. E. Verkade, and B. M. Wepster, Rec. Trav. Chim., 1957, 76, 401 (Chem. Abstr., 1957, 51, 15527d).
17. S. Kwee and H. Lund, Acta. Chem. Scand., 1971, 25, 1813.