High-throughput nuclear magnetic resonance-based screening

Journal of Medicinal Chemistry

Volumn 42, Issue 13, 1999, Pages 2315-2317

  Hajduk, Philip J ^a   Gerfin, Tobias ^b   Boehlen, Jean Marc ^b   Häberli, Markus ^b   Marek, Daniel ^b   Fesik, Stephen W ^a  

^a ABBOTT LABORATORIES   (United States)

^b Bruker AG   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

3 [4 (4 CYANOPHENYL)PHENOXY]PROPANOHYDROXAMIC ACID; LIGAND; PROTEIN; STROMELYSIN; STROMELYSIN INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CRYOPRESERVATION; DISSOCIATION CONSTANT; DRUG SCREENING; DRUG SOLUBILITY; LIGAND BINDING; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PROTON NUCLEAR MAGNETIC RESONANCE; SIGNAL NOISE RATIO; STRUCTURE ACTIVITY RELATION;

COLD; DRUG DESIGN; LIGANDS; MAGNETIC RESONANCE SPECTROSCOPY; MATRIX METALLOPROTEINASE 3; PROTEIN BINDING; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0033168872     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm9901475     Document Type: Article

References (14)

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