New synthesis of 5-cyano-1,2,4-thiadiazoles

Heterocycles

Volumn 51, Issue 4, 1999, Pages 811-819

  Iwakawa, Tsuneo ^a   Murabayashi, Akira ^a  

^a SHIONOGI AND CO LTD   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

5 CYANO 1,2,4 THIADIAZOLE DERIVATIVE; DICHLOROMETHANE; PIPERIDINE; THIADIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; REACTION ANALYSIS; SYNTHESIS;

EID: 0033117356     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/COM-98-8459     Document Type: Article

References (16)

1. (a) R. Appel, H. Janssen, M. Siray, and F. Knoch, Chem. Ber., 1985, 118, 1632.
2. (b) J. J. Folmer and S. M. Weinreb, Tetrahedron Lett., 1993, 34, 2737.
3. (c) A. M. Cuadro and J. Alvarez-Builla, Tetrahedron, 1994, 50, 10037.
4. C. W. Rees, J. Heterocycl. Chem., 1992, 29, 639.
5. (a) J. E. Moore, U.S. Patent, 1977, 4059590 [Chem. Abstr., 1978, 88, 50874a].
6. (b) R. Mayer, E. Foerster, and B. Matauschek, Ger. (East) DD, 1984, 212387 [Chem. Abstr., 1985, 102, 113064s].
7. (c) G. Cottenceau, T. Besson, V. Gautier, C. W. Rees, and A.-M. Pons, Bio. Med. Chem. Lett., 1996, 6, 529.
8. (d) V. Thiéry, C. W. Rees, T. Besson, G. Cottenceau, and A.-M. Pons, Eur. J. Med. Chem.,1998, 33, 149.
9. (a) K. C. Oh, H. Lee, and K. Kim, Tetrahedron Lett, 1992, 33, 4963.
10. (b) H. Lee and K. Kim, J. Org. Chem., 1993, 58, 7001.
11. (c) H. Lee, K. Kim, D. Whang, and K. Kim, J. Org. Chem., 1994, 59, 6179.
12. (d) H.-S. Lee and K. Kim, Tetrahedron Lett, 1996, 37, 869.
13. N. Vivona, G. Cusmano, and G. Macaluso, J. Chem. Soc., Perkin Trans. 1, 1977, 1616.
14. (a) J. Goerdeler, H. Groschopp, and U. Sommerlad, Chem. Ber., 1957, 90, 182.
15. (b) J. Goerdeler and K.-H. Heller, Chem. Ber., 1964, 97, 225.
16. H.W. Roesky, K. Keller, and J.W. Bats, Angew. Chem., Int. Ed. Engl., 1983, 22, 881.