Synthesis of novel peptidomimetics, cyclic hexamers of unnatural amino acids, 2,5-disubstituted 3-aminobenzoic acids

Heterocycles

Volumn 51, Issue 2, 1999, Pages 337-344

  Endo, Katsuya ^a   Takahashi, Hiroyasu ^a  

^a TOHOKU PHARMACEUTICAL UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

3 AMINOBENZOIC ACID; CYCLOPEPTIDE; HEXAPEPTIDE; MESYLIC ACID DERIVATIVE;

ARTICLE; CYCLIZATION; DRUG CONFORMATION; DRUG DESIGN; DRUG SYNTHESIS; MOLECULAR DYNAMICS; NUCLEAR OVERHAUSER EFFECT; TRANS ISOMER;

EID: 0033080397     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/COM-98-8445     Document Type: Article

References (11)

1. Unnatural Benzoic Amino Acids and their Derivatives. Part IV. Part III, ref. 4.
2. G. E. Schults and R. H. Schirmer, Principles of Protein Structure, Springer-Verlag, New York, 1979; C. Chothia, Ann. Rev. Biochem., 1984, 53, 537.
3. G. E. Schults and R. H. Schirmer, Principles of Protein Structure, Springer-Verlag, New York, 1979; C. Chothia, Ann. Rev. Biochem., 1984, 53, 537.
4. K. Endo, K. Kano, and H. Takahashi, Annual Report of Tohoku College of Pharmacy, 1995, 42, 77; H. Takahashi, Y. Matsuda, K. Kaji, and K. Endo, ibid., 1997, 44, 79.
5. K. Endo, K. Kano, and H. Takahashi, Annual Report of Tohoku College of Pharmacy, 1995, 42, 77; H. Takahashi, Y. Matsuda, K. Kaji, and K. Endo, ibid., 1997, 44, 79.
6. H. Takahashi, K. Wada, and K. Endo, Synthesis of Natural Amino Acid Analogues, Annual Report of Tohoku College of Pharmacy, 1998, 45, accepted for publication.
7. J. C. Sheehan and D. H. Yang, J. Am. Chem. Soc., 1958, 80, 1154.
8. CDI; 1,1-carbonyldiimidazole; R. Paul and G. W. Anderson, J. Org. Chem., 1962, 27, 2094.
9. K. Endo, H. Takahashi, and T. Kurusu, The 25th European Peptide Symposium, Budapest, Hungary, September 1988, Abstracts p.40; idem, Methanesulfonyl Chloride, a Facile and Powerful Coupling Reagent for Peptide Synthesis, to be published.
10. K. Endo, H. Takahashi, and T. Kurusu, The 25th European Peptide Symposium, Budapest, Hungary, September 1988, Abstracts p.40; idem, Methanesulfonyl Chloride, a Facile and Powerful Coupling Reagent for Peptide Synthesis, to be published.
11. K. Endo, H. Takahashi, T. Kurusu, K. Kaji, and A. Sida, The First International Peptide Symposium, Kyoto, Japan, December 1997, Abstracts p. 95.