메뉴 건너뛰기




Volumn 16, Issue 3-4, 1999, Pages 425-440

Synthesis and anti-phlogistic potency of some new nonproteinogenic amino acid conjugates of 'Diclofenac'

Author keywords

Amino acids; Anti phlogistics; Cyclo oxygenase inhibitors; Diclofenac; Non proteinogenic amino acids; Ulcerogenic gastritis; Voltaren . Thionation

Indexed keywords

AMINO ACID; BETA ALANINE; DICLOFENAC; DICLOFENAC DERIVATIVE; LEUCINE; NONSTEROID ANTIINFLAMMATORY AGENT; PHENYLALANINE; SARCOSINE; THIOAMIDE;

EID: 0033045488     PISSN: 09394451     EISSN: None     Source Type: Journal    
DOI: 10.1007/BF01388181     Document Type: Article
Times cited : (14)

References (32)
  • 1
    • 0029877868 scopus 로고    scopus 로고
    • Synthesis and anti-schistosomal activity of a new 2-nicotinoyl dipeptide analogue of praziquantel
    • Abo-Ghalia MH, Soliman AM (1996) Synthesis and anti-schistosomal activity of a new 2-nicotinoyl dipeptide analogue of praziquantel. Arzneimittelforschung/Drug Res 46/I 2: 207-209
    • (1996) Arzneimittelforschung/Drug Res , vol.46 , Issue.1-2 , pp. 207-209
    • Abo-Ghalia, M.H.1    Soliman, A.M.2
  • 2
    • 4243341530 scopus 로고    scopus 로고
    • "Studies on praziquantel". Synthesis and anti-schistosomal activity of some new analogues
    • in press
    • Abo-Ghalia MH, Soliman AM (1997) "Studies on praziquantel". Synthesis and anti-schistosomal activity of some new analogues. Egypt J Pharm Sci (in press)
    • (1997) Egypt J Pharm Sci
    • Abo-Ghalia, M.H.1    Soliman, A.M.2
  • 3
    • 0013593066 scopus 로고
    • Synthesis of some N-nicotinoyl amino acid derivatives with high anti-tubercular activity
    • Abo-Ghalia MH, Salem EMS, Shoeb S, Zedan M (1979) Synthesis of some N-nicotinoyl amino acid derivatives with high anti-tubercular activity. Polish J Chem 53: 2239-2250
    • (1979) Polish J Chem , vol.53 , pp. 2239-2250
    • Abo-Ghalia, M.H.1    Salem, E.M.S.2    Shoeb, S.3    Zedan, M.4
  • 4
    • 0022401034 scopus 로고
    • Specificity of uridine diphosphate-N-acetylmuramyl-L-alanyl-D-glutamate meso 2,6-diaminopimelate synthetase from Escherichia coli
    • Abo-Ghalia MH, Michaud C, Blanot D, Van Heijenoort J (1985) Specificity of uridine diphosphate-N-acetylmuramyl-L-alanyl-D-glutamate meso 2,6-diaminopimelate synthetase from Escherichia coli. Eur J Biochem 153: 81-87
    • (1985) Eur J Biochem , vol.153 , pp. 81-87
    • Abo-Ghalia, M.H.1    Michaud, C.2    Blanot, D.3    Van Heijenoort, J.4
  • 5
    • 0000540830 scopus 로고
    • Studies on amino acids and peptides IV. 1,2,4-Triazines from thioacylated amino acid esters
    • Andersen TP, Ghattas AB, Lawesson S-O (1983) Studies on amino acids and peptides IV. 1,2,4-Triazines from thioacylated amino acid esters. Tetrahydron 39/20: 3419-3427
    • (1983) Tetrahydron , vol.39 , Issue.20 , pp. 3419-3427
    • Andersen, T.P.1    Ghattas, A.B.2    Lawesson, S.-O.3
  • 7
    • 73049147644 scopus 로고    scopus 로고
    • Pharmacology of anti-tussive, 1-phcnethyl(2-propynyl)-4-propionoxy-piperidine acid fumarate
    • Charlier R, Prost M, Binon F, Deitor G (1961) Pharmacology of anti-tussive, 1-phcnethyl(2-propynyl)-4-propionoxy-piperidine acid fumarate. Arch Intern Pharmacodynamic 134: 306 & Chem Abst 56: 12251i
    • (1961) Arch Intern Pharmacodynamic , vol.134 , pp. 306
    • Charlier, R.1    Prost, M.2    Binon, F.3    Deitor, G.4
  • 8
    • 73049147644 scopus 로고    scopus 로고
    • Charlier R, Prost M, Binon F, Deitor G (1961) Pharmacology of anti-tussive, 1-phcnethyl(2-propynyl)-4-propionoxy-piperidine acid fumarate. Arch Intern Pharmacodynamic 134: 306 & Chem Abst 56: 12251i
    • Chem Abst , vol.56
  • 10
    • 0000986474 scopus 로고
    • Studies on amino acids and peptides-I. Synthesis of N-benzyloxycarbonyl endothiodipeptide esters
    • Clausen K, Thorsen M, Lawesson S-O (1981) Studies on amino acids and peptides-I. Synthesis of N-benzyloxycarbonyl endothiodipeptide esters. Tetrahydron 37/21; 3635
    • (1981) Tetrahydron , vol.37 , Issue.21 , pp. 3635
    • Clausen, K.1    Thorsen, M.2    Lawesson, S.-O.3
  • 11
    • 0020618647 scopus 로고
    • Pharmacodynamic and toxicology of Fenjhmizol, a new nonsterioidal anti-inflammatory drug. Imidazol derivative
    • Corell T, Hasselmann G (1983) Pharmacodynamic and toxicology of Fenjhmizol, a new nonsterioidal anti-inflammatory drug. Imidazol derivative. Acta Pharmacol Toxicol 53: 288
    • (1983) Acta Pharmacol Toxicol , vol.53 , pp. 288
    • Corell, T.1    Hasselmann, G.2
  • 12
    • 0018649742 scopus 로고
    • Interaction of salicylates and other non steroidal anti-inflammatory agents in rats as shown by gastro ulcerogenic and anti-inflammatory activities and plasma concentration
    • Corell T, Jensen KM, Splawinski J (1979) Interaction of salicylates and other non steroidal anti-inflammatory agents in rats as shown by gastro ulcerogenic and anti-inflammatory activities and plasma concentration. Acta Pharmacol Toxicol 45: 232-239
    • (1979) Acta Pharmacol Toxicol , vol.45 , pp. 232-239
    • Corell, T.1    Jensen, K.M.2    Splawinski, J.3
  • 13
    • 0018426518 scopus 로고
    • Drug therapy reviews. Anti-rheumatic agents
    • Evens RP (1979) Drug therapy reviews. Anti-rheumatic agents. Am J Hosp Pharm 36: 622
    • (1979) Am J Hosp Pharm , vol.36 , pp. 622
    • Evens, R.P.1
  • 14
    • 0018710274 scopus 로고
    • "Voltarol" Diclofenac sodium
    • Fowler PD (1979) "Voltarol" Diclofenac sodium. Clin Rheum Dis G B 5/2: 427-464
    • (1979) Clin Rheum Dis G B , vol.5 , Issue.2 , pp. 427-464
    • Fowler, P.D.1
  • 16
    • 0013616039 scopus 로고
    • JP 57081409 A2 820521 Showa. Chem Abst 97 8: 61070x
    • Kogyo TY (1982) "Poultices", JP 57081409 A2 820521 Showa. Chem Abst 97 8: 61070x
    • (1982) Poultices
    • Kogyo, T.Y.1
  • 17
    • 1542422767 scopus 로고
    • Zur frage des mechanismus der hemmung des bindegewebewachstums durch colisone
    • Meier R, Schuler W, Degulles P (1950) Zur Frage des Mechanismus der Hemmung des Bindegewebewachstums durch Colisone. Experientia (Basel) 6: 469-471
    • (1950) Experientia (Basel) , vol.6 , pp. 469-471
    • Meier, R.1    Schuler, W.2    Degulles, P.3
  • 23
    • 0030901759 scopus 로고    scopus 로고
    • Studies on o-[2,6-dichlorophenyl-1-amino]phenyl acetic acid I. Synthesis, anti-inflammatory, analgesic and ulcrogenic activities of some new amino acid conjugates
    • Shalaby AM, El-Eraky (1997) Studies on o-[2,6-dichlorophenyl-1-amino]phenyl acetic acid I. Synthesis, anti-inflammatory, analgesic and ulcrogenic activities of some new amino acid conjugates. El-Farmaco 5 22: 83-87
    • (1997) El-farmaco , vol.5 , Issue.22 , pp. 83-87
    • Shalaby, A.M.1
  • 24
    • 12444283342 scopus 로고
    • A new method of forming peptide bonds
    • Sheehan JC, Hess GP (1955) A new method of forming peptide bonds. J Am Chem Soc 77: 1067-1068
    • (1955) J Am Chem Soc , vol.77 , pp. 1067-1068
    • Sheehan, J.C.1    Hess, G.P.2
  • 25
    • 0015045998 scopus 로고
    • Zur behandlung säureempfindlicher aminosäure und peptidderivate
    • Spangenberg R, Thamm P, Wunsh E (1971) Zur Behandlung säureempfindlicher Aminosäure und Peptidderivate. Hoppe-Seyler's Z Physiol Chem 352: 655-656
    • (1971) Hoppe-seyler's Z Physiol Chem , vol.352 , pp. 655-656
    • Spangenberg, R.1    Thamm, P.2    Wunsh, E.3
  • 26
    • 0021056762 scopus 로고
    • Studies on amino acids and peptides, V. Synthesis of endothionated Melanostatin analogs
    • Thorsen M, Yde B, Pedersen U, Clausen K, Lawesson S-O (1983) Studies on amino acids and peptides, V. Synthesis of endothionated Melanostatin analogs. Tetrahydron 39/20: 3429-3435
    • (1983) Tetrahydron , vol.39 , Issue.20 , pp. 3429-3435
    • Thorsen, M.1    Yde, B.2    Pedersen, U.3    Clausen, K.4    Lawesson, S.-O.5
  • 28
    • 67249094291 scopus 로고
    • Carrageenan-induced oedema in hind paw of the rat as an assay for anti-inflammatory drugs
    • Winter CA, Rishey EA, Nuss GW (1962) Carrageenan-induced oedema in hind paw of the rat as an assay for anti-inflammatory drugs. Proc Soc Exp Biol Med 111: 544-547
    • (1962) Proc Soc Exp Biol Med , vol.111 , pp. 544-547
    • Winter, C.A.1    Rishey, E.A.2    Nuss, G.W.3
  • 29
    • 0019799424 scopus 로고
    • Rectal delivery of anti-inflammatory drugs, II. The influence of basic amino acid salts on retal absorption of Diclofenac
    • Yaginuma H, Isoda Y, Wada Y, Itoh S, Yamazaki M, Kamada A, Shimazu H, Makita I (1981) Rectal delivery of anti-inflammatory drugs, II. The influence of basic amino acid salts on retal absorption of Diclofenac. Chem Pharm Bull 29 11: 3326-3333
    • (1981) Chem Pharm Bull , vol.29 , Issue.11 , pp. 3326-3333
    • Yaginuma, H.1    Isoda, Y.2    Wada, Y.3    Itoh, S.4    Yamazaki, M.5    Kamada, A.6    Shimazu, H.7    Makita, I.8
  • 30
    • 0020395349 scopus 로고
    • Rectal delivery of anti-inflammatory drugs IV. Effect of amino acids on the change in the rectal mucosa induced by Diclofenac sodium
    • Yaginuma H, Isoda Y, Wada Y, Itoh S, Yamazaki M, Kamada A, Shimazu H, Makita I (1982a) Rectal delivery of anti-inflammatory drugs IV. Effect of amino acids on the change in the rectal mucosa induced by Diclofenac sodium. Chem Pharm Bull 30/9: 3302-3309
    • (1982) Chem Pharm Bull , vol.30 , Issue.9 , pp. 3302-3309
    • Yaginuma, H.1    Isoda, Y.2    Wada, Y.3    Itoh, S.4    Yamazaki, M.5    Kamada, A.6    Shimazu, H.7    Makita, I.8
  • 31
    • 0019988156 scopus 로고
    • Rectal delivery of anti-inflammatory drugs, III, effect of basic amino acid salts of Diclofenac on the retal absorption of Ampicilline sodium
    • Yaginuma H, Isoda Y, Wada Y, Itoh S, Yamazaki M, Kamada A, Shimazu H, Makita I (1982b) Rectal delivery of anti-inflammatory drugs, III, effect of basic amino acid salts of Diclofenac on the retal absorption of Ampicilline sodium. Chem Pharm Bull 30/3: 1073-1076
    • (1982) Chem Pharm Bull , vol.30 , Issue.3 , pp. 1073-1076
    • Yaginuma, H.1    Isoda, Y.2    Wada, Y.3    Itoh, S.4    Yamazaki, M.5    Kamada, A.6    Shimazu, H.7    Makita, I.8
  • 32
    • 0002860425 scopus 로고
    • Studies on amino acids and peptides, VII. Synthesis of aspartam and thioaspartam
    • Yde B, Thomsen I, Thorsen M, Clausen K, Lawesson S-O (1983) Studies on amino acids and peptides, VII. Synthesis of aspartam and thioaspartam. Tetrahydron 30/24: 4121-4126
    • (1983) Tetrahydron , vol.30 , Issue.24 , pp. 4121-4126
    • Yde, B.1    Thomsen, I.2    Thorsen, M.3    Clausen, K.4    Lawesson, S.-O.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.