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Volumn 126, Issue 6, 1999, Pages 1496-1503

Analysis of the behaviour of selected CCK(B)/gastrin receptor antagonists in radioligand binding assays performed in mouse and rat cerebral cortex

Author keywords

CCK(B) gastrin receptor; Guinea pig pancreas; JB93182; Mouse cortex; Rat cortex

Indexed keywords

1 [2,3 DIHYDRO 1 (2' METHYLPHENACYL) 2 OXO 5 PHENYL 1H 1,4 BENZODIAZEPIN 3 YL] 3 (3 METHYLPHENYL)UREA; 4 [[2 [2 [[(2 ADAMANTYLOXY)CARBONYL]AMINO] 3 (1H INDOL 3 YL) 2 METHYLPROPIONAMIDO] 1 PHENYLETHYL]AMINO] 4 OXOBUTYRIC ACID MEGLUMINE; 5 [[[[(3,5 DICARBOXYPHENYL)AMINO]CARBONYL] 2 PHENYLETHYLAMINO] CARBONYL] 6 [[(1 ADAMANTYLMETHYL) AMINO]CARBONYL]INDOLE; CHOLECYSTOKININ B RECEPTOR; CHOLECYSTOKININ B RECEPTOR ANTAGONIST; GASTRIN ANTAGONIST; GASTRIN RECEPTOR; PD 140376; UNCLASSIFIED DRUG;

EID: 0033042405     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0702448     Document Type: Article
Times cited : (17)

References (35)
  • 1
    • 0027460624 scopus 로고
    • A single amino acid of the cholecystokinin-B/gastrin receptor determines specificity for non-peptide antagonists
    • BEINBORN, M., LEE, Y.-M., MCBRIDE, E.W., QUINN, S.M. & KOPIN, A.S. (1993). A single amino acid of the cholecystokinin-B/gastrin receptor determines specificity for non-peptide antagonists. Nature, 362, 348-350.
    • (1993) Nature , vol.362 , pp. 348-350
    • Beinborn, M.1    Lee, Y.-M.2    McBride, E.W.3    Quinn, S.M.4    Kopin, A.S.5
  • 4
    • 4243388802 scopus 로고
    • β/gastrin receptor mRNA in colonic cell lines, human colonic carcinomas and hepatic metastasis: Study of co-expression with gastrin, somatostatin, cholecystokinin (CCK) and TGF α mRNA
    • β/gastrin receptor mRNA in colonic cell lines, human colonic carcinomas and hepatic metastasis: study of co-expression with gastrin, somatostatin, cholecystokinin (CCK) and TGF α mRNA. Gastroenterol., 108, A952.
    • (1995) Gastroenterol. , vol.108
    • Biagini, P.H.1    Cantaloube, J.F.2    Chicheportiche, C.3    Parriaux, D.4    Giovannini, M.5    Monges, G.6
  • 7
    • 0022516131 scopus 로고
    • A study of the cerebral cortex cholecystokinin receptor using two radiolabelled probes: Evidence for a common CCK8 and CCK4 cholecystokinin receptor binding site
    • CLARKE. C.R., DAUM, P. & HUGHES, J. (1986). A study of the cerebral cortex cholecystokinin receptor using two radiolabelled probes: evidence for a common CCK8 and CCK4 cholecystokinin receptor binding site. J. Neurochem., 46, 1094-1101.
    • (1986) J. Neurochem. , vol.46 , pp. 1094-1101
    • Clarke, C.R.1    Daum, P.2    Hughes, J.3
  • 9
    • 0019137579 scopus 로고
    • A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled β-adrenergic receptor
    • DE LEAN, A., STADEL, J.M. & LEFOKOWITZ, R. (1980). A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled β-adrenergic receptor. J. Biol. Chem., 255, 7108-7117.
    • (1980) J. Biol. Chem. , vol.255 , pp. 7108-7117
    • De Lean, A.1    Stadel, J.M.2    Lefokowitz, R.3
  • 14
    • 0029899545 scopus 로고    scopus 로고
    • Analysis of variation in L-365,260 competition curves in radioligand binding assays
    • HARPER, E.A., ROBERTS. S.P., SHANKLEY, N.P. & BLACK, J.W. (1996a). Analysis of variation in L-365,260 competition curves in radioligand binding assays. Br. J. Pharmacol., 118, 1717-1726.
    • (1996) Br. J. Pharmacol. , vol.118 , pp. 1717-1726
    • Harper, E.A.1    Roberts, S.P.2    Shankley, N.P.3    Black, J.W.4
  • 16
    • 0026092714 scopus 로고
    • Rationally designed 'dipeptoid' analogues of CCK. α-methyltryptophan derivatives as highly selective and orally active gastrin and CCK-β antagonists with potent anxiolytic properties
    • HORWELL, D.C., HUGHES, J., HUNTER, J.C., PRITCHARD, M.C., RICHARDSON, R., ROBERTS, E. & WOODRUFF, G.N. (1991). Rationally designed 'dipeptoid' analogues of CCK. α-methyltryptophan derivatives as highly selective and orally active gastrin and CCK-β antagonists with potent anxiolytic properties. J. Med. Chem., 34, 404-414.
    • (1991) J. Med. Chem. , vol.34 , pp. 404-414
    • Horwell, D.C.1    Hughes, J.2    Hunter, J.C.3    Pritchard, M.C.4    Richardson, R.5    Roberts, E.6    Woodruff, G.N.7
  • 17
    • 0027158477 scopus 로고
    • Diphenylpyrazolidinone and benzodiazepine cholecystokinin antagonists: A case of convergent evolution in medical chemistry
    • HOWBERT, J.J., LOBB, K.L., BRITTON. T.C., MASON, N.R. & BRUNS, R.F. (1993). Diphenylpyrazolidinone and benzodiazepine cholecystokinin antagonists: a case of convergent evolution in medical chemistry. Bioorgan. Med. Chem. Lett., 3, 875-880.
    • (1993) Bioorgan. Med. Chem. Lett. , vol.3 , pp. 875-880
    • Howbert, J.J.1    Lobb, K.L.2    Britton, T.C.3    Mason, N.R.4    Bruns, R.F.5
  • 20
    • 0028096885 scopus 로고
    • Functional characterisation of two cholecystokinin-β/gastrin receptor isoforms: A preferential splice donor site in the human receptor gene
    • ITO, M., IWATA, N., TANIGUCHI, T., MURAYAMA, T., CHICARA, K. & MATSUI, T. (1994). Functional characterisation of two cholecystokinin-β/gastrin receptor isoforms: A preferential splice donor site in the human receptor gene. Cell Growth Differentiation, 5, 1127- 1135.
    • (1994) Cell Growth Differentiation , vol.5 , pp. 1127-1135
    • Ito, M.1    Iwata, N.2    Taniguchi, T.3    Murayama, T.4    Chicara, K.5    Matsui, T.6
  • 23
    • 0025774950 scopus 로고
    • Novel and potent gastrin and brain cholecystokinin antagonists from streptomyces olivaceus. Taxonomy, fermentation, isolation, chemical conversions, and physico-chemical and biochemical properties
    • LAM, Y.K.T., BOGEN, D., CHANG, R.S., FAUST, K.A., HENSENS, O.D., ZINK, D.L., SCHWARTZ, C.D., ZITANG, L., GARRITY, G.M., GAGLIARDI, M.M., CURRIE, S.A. & WOODRUFF, H.B. (1990). Novel and potent gastrin and brain cholecystokinin antagonists from streptomyces olivaceus. Taxonomy, fermentation, isolation, chemical conversions, and physico-chemical and biochemical properties. J. Antibiotics, 44, 613-625.
    • (1990) J. Antibiotics , vol.44 , pp. 613-625
    • Lam, Y.K.T.1    Bogen, D.2    Chang, R.S.3    Faust, K.A.4    Hensens, O.D.5    Zink, D.L.6    Schwartz, C.D.7    Zitang, L.8    Garrity, G.M.9    Gagliardi, M.M.10    Currie, S.A.11    Woodruff, H.B.12
  • 24
    • 0024520619 scopus 로고
    • A new potent and selective non-peptide gastrin antagonist and brain cholecystokinin receptor (CCK-β) ligand: L-365,260
    • LOTTI, V.L. & CHANG, R.S.L. (1989). A new potent and selective non-peptide gastrin antagonist and brain cholecystokinin receptor (CCK-β) ligand: L-365,260. Eur. J. Pharmacol., 162, 273-280.
    • (1989) Eur. J. Pharmacol. , vol.162 , pp. 273-280
    • Lotti, V.L.1    Chang, R.S.L.2
  • 26
    • 0028290641 scopus 로고
    • Pharmacological profile of (R)-1-[2,3-dihydro-1-(2′-methyl-phenacyl)-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-y1]-3-(3-methylphenyl)urea (YM022), a new potent and selective gastrin/cholecystokinin- β receptor antagonist, in Vitro and in Vivo
    • NISHIDA, A., MIYATA, K., TSUTSUMI, R., YUKI, H., AKUZAWA, S., KOBAYASHI, A., KAMATO, T., ITO, H., YAMANO, M., KATUYAMA, Y., SATOH, M.. OHTA, M. & HONDA, K. (1994). Pharmacological profile of (R)-1-[2,3-dihydro-1-(2′-methyl-phenacyl)-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-y1]-3-(3-methylphenyl)urea (YM022), a new potent and selective gastrin/cholecystokinin- β receptor antagonist, in Vitro and in Vivo. J. Pharmacol. Exp. Ther., 269, 725-731.
    • (1994) J. Pharmacol. Exp. Ther. , vol.269 , pp. 725-731
    • Nishida, A.1    Miyata, K.2    Tsutsumi, R.3    Yuki, H.4    Akuzawa, S.5    Kobayashi, A.6    Kamato, T.7    Ito, H.8    Yamano, M.9    Katuyama, Y.10    Satoh, M.11    Ohta, M.12    Honda, K.13
  • 29
    • 0027052598 scopus 로고
    • Molecular cloning of the human brain and gastric cholecystokinin receptor: Structure, functional expression and chromosomal localisation
    • PISEGNA, J.R., DE WEERTH, A., HUPPI, K. & WANK, S.A. (1992). Molecular cloning of the human brain and gastric cholecystokinin receptor: Structure, functional expression and chromosomal localisation. Biochem. Biophys. Res. Common., 189, 295-303.
    • (1992) Biochem. Biophys. Res. Common. , vol.189 , pp. 295-303
    • Pisegna, J.R.1    Weerth, D.E.2    Huppi, A.3    Wank, K.S.A.4
  • 30
    • 0027450750 scopus 로고
    • Receptor antagonists for gastrointestinal peptides
    • PRESTI, M.E. & GARDNER, J.D. (1993). Receptor antagonists for gastrointestinal peptides. Am. J. Physiol., 264, G399-G406.
    • (1993) Am. J. Physiol. , vol.264
    • Presti, M.E.1    Gardner, J.D.2
  • 33
    • 0002502080 scopus 로고    scopus 로고
    • Analysis of the complex pharmacology expressed by the CCK-β/gastrin ligand PD134,308 on gastric assays
    • SHANKLEY, N.P., ROBERTS, S.P., WATT, G.F., KOTECHA, A., HULL, R. & BLACK, J.W. (1997). Analysis of the complex pharmacology expressed by the CCK-β/gastrin ligand PD134,308 on gastric assays. ASPET Pharmacol., 39, P65.
    • (1997) ASPET Pharmacol. , vol.39 , pp. 65
    • Shankley, N.P.1    Roberts, S.P.2    Watt, G.F.3    Kotecha, A.4    Hull, R.5    Black, J.W.6
  • 34
    • 0027379255 scopus 로고
    • The human gastrin/cholecystokinin type β receptor gene: Alternative splice donor site in exon 4 generate two variant mRNAs
    • SONG, I., BROWN, D.R., WILTSHIRE, R.N., GANTZ, I., TRENT, J.M. & YAMADA, T. (1993). The human gastrin/cholecystokinin type β receptor gene: Alternative splice donor site in exon 4 generate two variant mRNAs. Proc. Natl. Acad. Sci. U.S.A., 90, 9085-9089.
    • (1993) Proc. Natl. Acad. Sci. U.S.A. , vol.90 , pp. 9085-9089
    • Song, I.1    Brown, D.R.2    Wiltshire, R.N.3    Gantz, I.4    Trent, J.M.5    Yamada, T.6
  • 35
    • 0000274943 scopus 로고
    • Functional significance of potential splice variants of the human cholecystokinin (CCK) β receptor
    • WANK, S.A., PISEGNA, J.R. & POIROT, S.S. (1994). Functional significance of potential splice variants of the human cholecystokinin (CCK) β receptor. Gastroenterology, 106, A850.
    • (1994) Gastroenterology , vol.106
    • Wank, S.A.1    Pisegna, J.R.2    Poirot, S.S.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.