메뉴 건너뛰기




Volumn 7, Issue 4, 1999, Pages 325-330

Investigation of the mechanism of flux across human skin in vitro by quantitative structure-permeability relationships

Author keywords

Human skin; Polydimethylsiloxane; Quantitative structure activity relationships; Quantitative structure permeability relationships; Transdermal drug delivery

Indexed keywords

ORGANIC COMPOUND;

EID: 0033038344     PISSN: 09280987     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0928-0987(98)00041-4     Document Type: Article
Times cited : (136)

References (30)
  • 2
    • 0028898732 scopus 로고
    • Quantitative structure-activity relationships for permeability
    • Barratt M.D. Quantitative structure-activity relationships for permeability. Toxicol. In Vitro. 9:1995;27-37.
    • (1995) Toxicol. in Vitro , vol.9 , pp. 27-37
    • Barratt, M.D.1
  • 3
    • 0020371598 scopus 로고
    • The structural dependence of amino acid hydrophobicity parameters
    • Charton M., Charton B.I. The structural dependence of amino acid hydrophobicity parameters. J. Theoret. Biol. 99:1982;619-624.
    • (1982) J. Theoret. Biol. , vol.99 , pp. 619-624
    • Charton, M.1    Charton, B.I.2
  • 5
    • 0031889726 scopus 로고    scopus 로고
    • An investigation of the mechanism of flux across polydimethylsiloxane membranes by quantitative structure-permeability relationships
    • Cronin M.T.D., Dearden J.C., Gupta R., Moss G.P. An investigation of the mechanism of flux across polydimethylsiloxane membranes by quantitative structure-permeability relationships. J. Pharm. Pharmacol. 50:1998;143-152.
    • (1998) J. Pharm. Pharmacol. , vol.50 , pp. 143-152
    • Cronin, M.T.D.1    Dearden, J.C.2    Gupta, R.3    Moss, G.P.4
  • 6
    • 0022272070 scopus 로고
    • Partitioning and lipophilicity in quantitative structure-activity relationships
    • Dearden J.C. Partitioning and lipophilicity in quantitative structure-activity relationships. Environ. Health Persp. 61:1985;203-228.
    • (1985) Environ. Health Persp. , vol.61 , pp. 203-228
    • Dearden, J.C.1
  • 8
    • 0842341771 scopus 로고
    • The development and use of quantum-mechanical models. 76. AM1 - A new general-purpose quantum-mechanical molecular model
    • Dewar M.J.S., Zoebisch E.G., Healy E.F., Stewart J.J.P. The development and use of quantum-mechanical models. 76. AM1 - A new general-purpose quantum-mechanical molecular model. J. Am. Chem. Soc. 107:1985;3902-3909.
    • (1985) J. Am. Chem. Soc. , vol.107 , pp. 3902-3909
    • Dewar, M.J.S.1    Zoebisch, E.G.2    Healy, E.F.3    Stewart, J.J.P.4
  • 9
    • 0002584744 scopus 로고
    • Physicochemical determinants of skin absorption
    • In: Gerrity, T.R., Henry, C.J. (Eds.), Elsevier, New York
    • Flynn, G.L., 1990. Physicochemical determinants of skin absorption. In: Gerrity, T.R., Henry, C.J. (Eds.), Principle of Route-to-Route Extrapolation for Risk Assessment. Elsevier, New York, pp. 93-127.
    • (1990) Principle of Route-to-Route Extrapolation for Risk Assessment , pp. 93-127
    • Flynn, G.L.1
  • 10
    • 0026504445 scopus 로고
    • In vitro skin permeation techniques
    • Friend D.R. In vitro skin permeation techniques. J. Cont. Rel. 18:1992;235-248.
    • (1992) J. Cont. Rel. , vol.18 , pp. 235-248
    • Friend, D.R.1
  • 11
    • 0017645935 scopus 로고
    • Hydrogen-bonding parameter and its significance in quantitative structure-activity studies
    • Fujita T., Nishioka T., Nakajima M. Hydrogen-bonding parameter and its significance in quantitative structure-activity studies. J. Med. Chem. 20:1977;1071-1081.
    • (1977) J. Med. Chem. , vol.20 , pp. 1071-1081
    • Fujita, T.1    Nishioka, T.2    Nakajima, M.3
  • 12
    • 0014298182 scopus 로고
    • Evaluation, control and prediction of drug diffusion through polymeric membranes II
    • Garrett E.R., Chemburkar P.B. Evaluation, control and prediction of drug diffusion through polymeric membranes II. J. Pharm. Sci. 57:1968;949-959.
    • (1968) J. Pharm. Sci. , vol.57 , pp. 949-959
    • Garrett, E.R.1    Chemburkar, P.B.2
  • 14
    • 0001970191 scopus 로고
    • Drug structure vs. penetration
    • In: Kydonieus, A.F., Berner, B. (Eds.), CRC Press, Boca Raton, FL
    • Idson, B., Charanjit, R.B., 1987. Drug structure vs. penetration. In: Kydonieus, A.F., Berner, B. (Eds.), Transdermal Delivery of Drugs, Vol. III. CRC Press, Boca Raton, FL, pp. 85-151.
    • (1987) Transdermal Delivery of Drugs , vol.3 , pp. 85-151
    • Idson, B.1    Charanjit, R.B.2
  • 17
    • 2542594118 scopus 로고    scopus 로고
    • The prediction of skin permeability by using physicochemical data
    • Kirchner L.A., Moody R.P., Doyle E., Bose B., Jeffry J., Chu I. The prediction of skin permeability by using physicochemical data. ATLA. 25:1997;359-370.
    • (1997) ATLA , vol.25 , pp. 359-370
    • Kirchner, L.A.1    Moody, R.P.2    Doyle, E.3    Bose, B.4    Jeffry, J.5    Chu, I.6
  • 18
    • 0031024171 scopus 로고    scopus 로고
    • Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
    • Lipinski C.A., Lombardo F., Dominy B.W., Feeney P.J. Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings. Adv. Drug Deliv. Rev. 23:1997;3-25.
    • (1997) Adv. Drug Deliv. Rev. , vol.23 , pp. 3-25
    • Lipinski, C.A.1    Lombardo, F.2    Dominy, B.W.3    Feeney, P.J.4
  • 19
    • 0023857071 scopus 로고
    • Comparative in vivo and in vitro assessment of percutaneous absorption of local anaesthetics
    • McCafferty D.F., Woolfson A.D., McClelland K.H., Boston V. Comparative in vivo and in vitro assessment of percutaneous absorption of local anaesthetics. Br. J. Anaesth. 60:1988;64-69.
    • (1988) Br. J. Anaesth. , vol.60 , pp. 64-69
    • McCafferty, D.F.1    Woolfson, A.D.2    McClelland, K.H.3    Boston, V.4
  • 20
    • 0028884828 scopus 로고
    • Estradiol permeation through human skin and silastic membrane - effects of propylene glycol and supersaturation
    • Magrab N.A., Williams A.C., Barry B.W. Estradiol permeation through human skin and silastic membrane - effects of propylene glycol and supersaturation. J. Control. Release. 36:1995;277-294.
    • (1995) J. Control. Release , vol.36 , pp. 277-294
    • Magrab, N.A.1    Williams, A.C.2    Barry, B.W.3
  • 21
    • 0026606514 scopus 로고
    • Predicting skin permeability
    • Potts R.O., Guy R.H. Predicting skin permeability. Pharm. Res. 9:1992;663-669.
    • (1992) Pharm. Res. , vol.9 , pp. 663-669
    • Potts, R.O.1    Guy, R.H.2
  • 22
    • 0029618807 scopus 로고
    • A predictive algorithm for skin permeability: The effects of molecular size and hydrogen bond activity
    • Potts R.O., Guy R.H. A predictive algorithm for skin permeability: the effects of molecular size and hydrogen bond activity. Pharm. Res. 12:1995;1628-1633.
    • (1995) Pharm. Res. , vol.12 , pp. 1628-1633
    • Potts, R.O.1    Guy, R.H.2
  • 23
    • 0028013532 scopus 로고
    • Ab initio prediction of human skin permeability coefficients
    • Pugh W.J., Hadgraft J. Ab initio prediction of human skin permeability coefficients. Int. J. Pharm. 103:1994;163-178.
    • (1994) Int. J. Pharm. , vol.103 , pp. 163-178
    • Pugh, W.J.1    Hadgraft, J.2
  • 24
    • 0029768028 scopus 로고    scopus 로고
    • Epidermal permeability - penetrant structure relationships: 3. The effect of hydrogen bonding interactions and molecular size on diffusion across the stratum corneum
    • Pugh W.J., Roberts M.S., Hadgraft J. Epidermal permeability - penetrant structure relationships: 3. The effect of hydrogen bonding interactions and molecular size on diffusion across the stratum corneum. Int. J. Pharm. 138:1996;149-165.
    • (1996) Int. J. Pharm. , vol.138 , pp. 149-165
    • Pugh, W.J.1    Roberts, M.S.2    Hadgraft, J.3
  • 28
    • 0344485409 scopus 로고
    • OSHA chemical referred to the ISCA Interagency Testing Committee for percutaneous absorption testing and prioritization and analysis of OSHA skin notation criteria
    • Wittiker C., Walker J.D., Gay D.A., Neal M.W. OSHA chemical referred to the ISCA Interagency Testing Committee for percutaneous absorption testing and prioritization and analysis of OSHA skin notation criteria. Toxicologist. 13:1993;101.
    • (1993) Toxicologist , vol.13 , pp. 101
    • Wittiker, C.1    Walker, J.D.2    Gay, D.A.3    Neal, M.W.4
  • 29
    • 0027301194 scopus 로고
    • Percutaneous local anaesthesia: Drug release characteristics of the amethocaine phase-change system
    • Woolfson A.D., McCafferty D.F. Percutaneous local anaesthesia: drug release characteristics of the amethocaine phase-change system. Int. J. Pharm. 94:1993;75-80.
    • (1993) Int. J. Pharm. , vol.94 , pp. 75-80
    • Woolfson, A.D.1    McCafferty, D.F.2
  • 30
    • 0022650034 scopus 로고
    • Physical factors contributing to hydrophobic constant π
    • Yang G., Lien E.J., Gao Z. Physical factors contributing to hydrophobic constant π Quant. Struct.-Act. Relat. 5:1986;12-18.
    • (1986) Quant. Struct.-Act. Relat. , vol.5 , pp. 12-18
    • Yang, G.1    Lien, E.J.2    Gao, Z.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.