메뉴 건너뛰기




Volumn 5, Issue 2, 1999, Pages 95-101

Structural modification from agonists to antagonists in the synthesis of new 5-hydroxytryptamine (5-HT3) receptor antagonists and preliminary in-vitro pharmacological evaluation on guinea-pig ileum

Author keywords

[No Author keywords available]

Indexed keywords

ACETONE; ONDANSETRON; PIPERAZINE; SEROTONIN 3 ANTAGONIST;

EID: 0033033238     PISSN: 14608081     EISSN: None     Source Type: Journal    
DOI: 10.1211/146080899128734523     Document Type: Article
Times cited : (3)

References (14)
  • 1
    • 0025917723 scopus 로고
    • 3 receptor antagonists. An overview of their present status and future potential in cancer therapy-induced emesis
    • 3 receptor antagonists. An overview of their present status and future potential in cancer therapy-induced emesis. Drugs 42: 551-558
    • (1991) Drugs , vol.42 , pp. 551-558
    • Aapro, M.S.1
  • 3
    • 0023767669 scopus 로고
    • Pharmacological properties of GR 63032F, a novel antagonist at 5-HT3 receptors
    • Butler, A., Hill, J. M., Ireland, S. J., Jordan, C. C., Tyers, M. B. (1988) Pharmacological properties of GR 63032F, a novel antagonist at 5-HT3 receptors. Br. J. Pharmacol. 94: 387-412
    • (1988) Br. J. Pharmacol. , vol.94 , pp. 387-412
    • Butler, A.1    Hill, J.M.2    Ireland, S.J.3    Jordan, C.C.4    Tyers, M.B.5
  • 6
    • 13344280365 scopus 로고    scopus 로고
    • Classification and nomenclature of 5-HT receptors: A comment on current issues
    • Hoyer, D., Martin, G. R. (1996) Classification and nomenclature of 5-HT receptors: a comment on current issues. Behav. Brain Res. 73: 263-268
    • (1996) Behav. Brain Res. , vol.73 , pp. 263-268
    • Hoyer, D.1    Martin, G.R.2
  • 8
    • 0027526944 scopus 로고
    • Structural modification patterns from agonists to antagonists and their application to drug design
    • Jucker, E. (ed.), Verlag, Basel, Switzerland
    • Ohtaka, H., Fujita, T. (1994) Structural modification patterns from agonists to antagonists and their application to drug design. In: Jucker, E. (ed.) Progress in Drug Research. Vol. 41, Verlag, Basel, Switzerland, pp 313-357
    • (1994) Progress in Drug Research , vol.41 , pp. 313-357
    • Ohtaka, H.1    Fujita, T.2
  • 10
    • 0021812342 scopus 로고
    • Identification of serotonin M-receptor subtypes and their specific blockade by a new class of drugs
    • Richardson, B. P., Engel, G., Donatsch, P., Stadler, P. A. (1985) Identification of serotonin M-receptor subtypes and their specific blockade by a new class of drugs. Nature 316: 126-131
    • (1985) Nature , vol.316 , pp. 126-131
    • Richardson, B.P.1    Engel, G.2    Donatsch, P.3    Stadler, P.A.4
  • 11
    • 0024587689 scopus 로고
    • 3 receptor antagonism by BRL 43694 (granisetron)
    • 3 receptor antagonism by BRL 43694 (granisetron). Eur. J. Pharmacol. 159: 113-124
    • (1989) Eur. J. Pharmacol. , vol.159 , pp. 113-124
    • Sanger, G.J.1    Nelson, G.R.2
  • 12
    • 0009766924 scopus 로고
    • The reaction between indole and acetic anhydride
    • Saxton, J. E. (1952) The reaction between indole and acetic anhydride. J. Chem. Soc. 3592-3594
    • (1952) J. Chem. Soc. , pp. 3592-3594
    • Saxton, J.E.1
  • 13
    • 0010359019 scopus 로고
    • 3-Acylindole mannich bases and their transformation products
    • Szmuszkovicz, J. (1960) 3-Acylindole mannich bases and their transformation products. J. Am. Chem. Soc. 82: 1180-1186
    • (1960) J. Am. Chem. Soc. , vol.82 , pp. 1180-1186
    • Szmuszkovicz, J.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.