Expedient synthesis of α-substituted α,β-unsaturated γ-amino acids (dipeptide mimetics); Wittig reaction of α-amino aldehydes with α- substituted alkoxycarbonyl phosphoranes

Synthetic Communications

Volumn 29, Issue 7, 1999, Pages 1143-1155

  Scholz, Dieter ^a   Weber Roth, Sabine ^a   Macoratti, Elena ^a   Francotte, Eric ^b  

^a Novartis Pharma AG   (Austria)

^b NOVARTIS PHARMA AG   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACID; DIPEPTIDE; PHOSPHORANE DERIVATIVE;

ARTICLE; CHEMICAL REACTION; CHEMICAL STRUCTURE; CHIRALITY; ENANTIOMER; STEREOSPECIFICITY; SYNTHESIS;

EID: 0033029019     PISSN: 00397911     EISSN: None     Source Type: Journal    
DOI: 10.1080/00397919908086084     Document Type: Article

References (5)

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2. Scholz, D.; Billich, A.; Charpiot, B.; Ettmayer, P.; Lehr, P.; Rosenwirth, B.; Schreiner, E. and Gstach, H. J. Med. Chem. 1994, 37, 3079. and citations there in.
3. Britto, N.; Gore, V.G.; Mali, R.S. and Ranade, A.C. Synthetic Commmunications, 1989, 19, 1899.
4. Bestmann, H.J. and Schulz, H. Chem. Ber. 1962, 95, 2921.
5. Shue, Y-K.; Carrera Jr., G.M.; Tufano, M.D. and Nadzan, A.M. J. Med. Chem. 1991, 56, 2107.