Fentanyl analogues with a modified propanamido group as potential affinity labels: Synthesis and in vivo activity

Pharmazie

Volumn 54, Issue 4, 1999, Pages 307-308

  Essawi, M Y H ^a  

^a CAIRO UNIVERSITY   (Egypt)

Author keywords

[No Author keywords available]

Indexed keywords

FENTANYL; FENTANYL DERIVATIVE; MORPHINE SULFATE; NALOXONE;

ANALGESIA; ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ARTICLE; BINDING AFFINITY; DOSE RESPONSE; DRUG EFFECT; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; INTRAPERITONEAL DRUG ADMINISTRATION; MOUSE; NONHUMAN; REACTION TIME; STRUCTURE ACTIVITY RELATION;

AFFINITY LABELS; ANALGESICS, OPIOID; ANIMALS; FENTANYL; INJECTIONS, INTRAPERITONEAL; MAGNETIC RESONANCE SPECTROSCOPY; MICE; NALOXONE; NARCOTIC ANTAGONISTS; PAIN MEASUREMENT; SPECTROPHOTOMETRY, INFRARED;

EID: 0033027631     PISSN: 00317144     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (10)

1. Takemori, A. E.; Portoghese, P. S.: Annu. Rev. Pharmacol. Toxicol. 25, 193 (1985)
2. Korlipara, V. L.; Takemori, A. E.; Portoghese, P. S.: J. Med. Chem. 38, 1337 (1995)
3. Zhu, J.; Yin, J.; Law, P.-Y.; Claude, P. A.; Rice, K. C.; Evans, C. J.; Chen. C.; Yu, L.; Liu-Chen, L.-Y.: J. Biol. Chem. 271, 1430 (1996)
4. Janssen, P. A. J.: Br. J. Anaesth. 34, 260 (1962)
5. Acheson, R. M.; Feinberg, R. S.; Hands, A. R.: J. Chem. Soc. 526 (1964)
6. Eddy, N. B.; Leimbach, D.: J. Pharmacol. Exp. Ther. 107, 385 (1953)
7. Cowi, A. L.; Kosterlitz, H. W.; Watt, A. J.; Nature (London) 220, 1040 (1968)
8. Sayer, L. M.; Larson, D. L.; Takemori, A. E.; Portoghese, P. S.: J. Med. Chem. 27, 1325 (1984)
9. Caruso, T. P.; Takemori, A. E.; Larson, D. L., Portoghese, P. S.; Science 204, 316 (1979)
10. Portoghese, P. S.: J. Med. Chem. 8, 609 (1965)