메뉴 건너뛰기




Volumn 368, Issue 2-3, 1999, Pages 161-172

Changes of benzodiazepine receptors during chronic benzodiazepine administration in humans

Author keywords

Benzodiazepine; Down regulation; GABA(A) benzodiazepine receptor; Human; SPECT (single photon emission computed tomography)

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR; ALPRAZOLAM; BENZODIAZEPINE RECEPTOR; BENZODIAZEPINE RECEPTOR STIMULATING AGENT;

EID: 0033012659     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(99)00013-8     Document Type: Article
Times cited : (46)

References (57)
  • 5
    • 0025890255 scopus 로고
    • The Hopkins Verbal Learning Test: Development of a new memory test with six equivalent forms
    • Brandt J. The Hopkins Verbal Learning Test: development of a new memory test with six equivalent forms. Clin. Neuropsychol. 5:1991;125-142.
    • (1991) Clin. Neuropsychol. , vol.5 , pp. 125-142
    • Brandt, J.1
  • 7
    • 0343591959 scopus 로고
    • 3H]flunitrazepam binding after chronic low dose diazepam treatment in rats
    • 3H ]flunitrazepam binding after chronic low dose diazepam treatment in rats Proc. Br. J. Pharmacol. 105:1992;172P.
    • (1992) Proc. Br. J. Pharmacol. , vol.105
    • Brett, R.R.1    Pratt, J.A.2
  • 9
    • 0027416840 scopus 로고
    • Chronic benzodiazepine administration: XII. Anticonvulsant cross-tolerance but distinct neurochemical effects of alprazolam and lorazepam
    • Byrnes J.J., Miller L.G., Greenblatt D.J., Shader R.I. Chronic benzodiazepine administration: XII. Anticonvulsant cross-tolerance but distinct neurochemical effects of alprazolam and lorazepam. Psychopharmacology. 111:1993;91-95.
    • (1993) Psychopharmacology , vol.111 , pp. 91-95
    • Byrnes, J.J.1    Miller, L.G.2    Greenblatt, D.J.3    Shader, R.I.4
  • 11
    • 0022636251 scopus 로고
    • Pharmacokinetics and clinical effects of alprazolam following single and multiple oral doses in patients with panic disorder
    • Ciraulo C., Barnhill J.G., Boxenbaum H.G., Greenblatt D.J., Smith R.B. Pharmacokinetics and clinical effects of alprazolam following single and multiple oral doses in patients with panic disorder. J. Clin. Pharmacol. 26:1986;292-298.
    • (1986) J. Clin. Pharmacol. , vol.26 , pp. 292-298
    • Ciraulo, C.1    Barnhill, J.G.2    Boxenbaum, H.G.3    Greenblatt, D.J.4    Smith, R.B.5
  • 13
    • 84944656328 scopus 로고
    • Comparison of alprazolam, imipramine and placebo in the treatment of depression
    • Feighner J.P., Aden G.C., Fabre L.F., Rickels K., Smith W.T. Comparison of alprazolam, imipramine and placebo in the treatment of depression. JAMA. 249:1983;3057-3064.
    • (1983) JAMA , vol.249 , pp. 3057-3064
    • Feighner, J.P.1    Aden, G.C.2    Fabre, L.F.3    Rickels, K.4    Smith, W.T.5
  • 14
    • 0022570677 scopus 로고
    • The pharmacokinetics of diazepam and desmethyldiazepam in rat brain and plasma
    • Friedman H., Abernethy D.R., Greenblatt D.J., Shader R.I. The pharmacokinetics of diazepam and desmethyldiazepam in rat brain and plasma. Psychopharmacology. 88:1986;267-270.
    • (1986) Psychopharmacology , vol.88 , pp. 267-270
    • Friedman, H.1    Abernethy, D.R.2    Greenblatt, D.J.3    Shader, R.I.4
  • 15
    • 0025881775 scopus 로고
    • Comparative pharmacokinetics of alprazolam and lorazepam in humans and in African Green Monkeys
    • Friedman H., Redmond D. Jr., Greenblatt D.J. Comparative pharmacokinetics of alprazolam and lorazepam in humans and in African Green Monkeys. Psychopharmacology. 104:1991;103-105.
    • (1991) Psychopharmacology , vol.104 , pp. 103-105
    • Friedman, H.1    Redmond D., Jr.2    Greenblatt, D.J.3
  • 17
    • 0021240080 scopus 로고
    • Chronic benzodiazepine treatment decreases postsynaptic GABA sensitivity
    • Gallager D.W., Lakoski J.M., Gonsalves S.F., Rauch S.L. Chronic benzodiazepine treatment decreases postsynaptic GABA sensitivity. Nature. 308:1984;74-77.
    • (1984) Nature , vol.308 , pp. 74-77
    • Gallager, D.W.1    Lakoski, J.M.2    Gonsalves, S.F.3    Rauch, S.L.4
  • 19
    • 0028289554 scopus 로고
    • Evaluation of ultrafiltration for the free fraction determination of single photon emission computed tomography (SPECT) tracers: Β-CIT, IBF, and iomazenil
    • Gandelman M.S., Baldwin R.M., Zoghbi S.S., Zea-Ponce Y., Innis R.B. Evaluation of ultrafiltration for the free fraction determination of single photon emission computed tomography (SPECT) tracers: β-CIT, IBF, and iomazenil. J. Pharm. Sci. 83:1994;1014-1019.
    • (1994) J. Pharm. Sci. , vol.83 , pp. 1014-1019
    • Gandelman, M.S.1    Baldwin, R.M.2    Zoghbi, S.S.3    Zea-Ponce, Y.4    Innis, R.B.5
  • 20
    • 0022474635 scopus 로고
    • Long-term administration of benzodiazepines: Pharmacokinetic versus pharmacodynamic tolerance
    • Greenblatt D.J., Shader R.I. Long-term administration of benzodiazepines: pharmacokinetic versus pharmacodynamic tolerance. Psychopharmacol. Bull. 22:1986;416-423.
    • (1986) Psychopharmacol. Bull. , vol.22 , pp. 416-423
    • Greenblatt, D.J.1    Shader, R.I.2
  • 21
    • 0027215914 scopus 로고
    • Clinical pharmacokinetics of alprazolam, therapeutic implications
    • Greenblatt D.J., Wright C.E. Clinical pharmacokinetics of alprazolam, therapeutic implications. Clin. Pharmacokinet. 24:1993;453-471.
    • (1993) Clin. Pharmacokinet. , vol.24 , pp. 453-471
    • Greenblatt, D.J.1    Wright, C.E.2
  • 24
    • 0029895184 scopus 로고    scopus 로고
    • The behavioural and neuronal effects of the chronic administration of benzodiazepine anxiolytic and hypnotic drugs
    • Hutchinson M.A., Smith P.F., Darlington C.L. The behavioural and neuronal effects of the chronic administration of benzodiazepine anxiolytic and hypnotic drugs. Prog. Neurobiol. 49:1996;73-97.
    • (1996) Prog. Neurobiol. , vol.49 , pp. 73-97
    • Hutchinson, M.A.1    Smith, P.F.2    Darlington, C.L.3
  • 27
    • 0025922261 scopus 로고
    • A receptor subunit mRNA concentrations following chronic lorazepam administration
    • A receptor subunit mRNA concentrations following chronic lorazepam administration. Br. J. Pharmacol. 103:1991;1285-1287.
    • (1991) Br. J. Pharmacol. , vol.103 , pp. 1285-1287
    • Kang, I.1    Miller, L.G.2
  • 29
    • 0017181881 scopus 로고
    • Pharmacokinetics and plasma binding of diazepam in man, dog, rabbit, guinea pig and rat
    • Klotz U., Antonin K.H., Bieck T. Pharmacokinetics and plasma binding of diazepam in man, dog, rabbit, guinea pig and rat. J. Pharmacol. Exp. Ther. 199:1976;67-73.
    • (1976) J. Pharmacol. Exp. Ther. , vol.199 , pp. 67-73
    • Klotz, U.1    Antonin, K.H.2    Bieck, T.3
  • 31
    • 0030299874 scopus 로고    scopus 로고
    • A receptor subunit mRNA expression during tolerance to diazepam-induced cognition dysfunction
    • A receptor subunit mRNA expression during tolerance to diazepam-induced cognition dysfunction. Neuropharmacology. 35:1996;1465-1473.
    • (1996) Neuropharmacology , vol.35 , pp. 1465-1473
    • Longone, P.1    Impagnatiello, F.2    Guidotti, A.3    Costa, E.4
  • 33
    • 0022568707 scopus 로고
    • Chronic use of benzodiazepines and psychomotor and cognitive test performance
    • Lucki I., Rickels K., Geller A.M. Chronic use of benzodiazepines and psychomotor and cognitive test performance. Psychopharmacolgy. 88:1986;426-433.
    • (1986) Psychopharmacolgy , vol.88 , pp. 426-433
    • Lucki, I.1    Rickels, K.2    Geller, A.M.3
  • 34
    • 0021706289 scopus 로고
    • Quantification of alprazolam in serum or plasma by liquid chromatography
    • McCormick S.R., Nielsen J., Jatlow P. Quantification of alprazolam in serum or plasma by liquid chromatography. Clin. Chem. 30:1984;1662-1665.
    • (1984) Clin. Chem. , vol.30 , pp. 1662-1665
    • McCormick, S.R.1    Nielsen, J.2    Jatlow, P.3
  • 35
    • 0021691143 scopus 로고
    • Chronic administration of diazepam to rats causes changes in EEG patterns and in coupling between GABA receptors and benzodiazepine binding sites in vitro
    • Mele L., Sagratella S., Massotti M. Chronic administration of diazepam to rats causes changes in EEG patterns and in coupling between GABA receptors and benzodiazepine binding sites in vitro. Brain Res. 323:1984;93-102.
    • (1984) Brain Res. , vol.323 , pp. 93-102
    • Mele, L.1    Sagratella, S.2    Massotti, M.3
  • 36
    • 0030036620 scopus 로고    scopus 로고
    • Long-term use of benzodiazepines: Tolerance, dependence and clinical problems in anxiety and mood disorders
    • Michelini S., Cassano G.B., Frare F., Perugi G. Long-term use of benzodiazepines: tolerance, dependence and clinical problems in anxiety and mood disorders. Pharmacopsychiatry. 29:1996;127-134.
    • (1996) Pharmacopsychiatry , vol.29 , pp. 127-134
    • Michelini, S.1    Cassano, G.B.2    Frare, F.3    Perugi, G.4
  • 37
    • 0023280697 scopus 로고
    • Benzodiazepine receptor binding of triazolobenzodiazepines in vivo: Increased receptor number with low-dose alprazolam
    • Miller L.G., Greenblatt D.J., Barnhill J.G., Deutsch S.I., Shader R.I., Paul S.M. Benzodiazepine receptor binding of triazolobenzodiazepines in vivo: increased receptor number with low-dose alprazolam. J. Neurochem. 49:1987;1595-1601.
    • (1987) J. Neurochem. , vol.49 , pp. 1595-1601
    • Miller, L.G.1    Greenblatt, D.J.2    Barnhill, J.G.3    Deutsch, S.I.4    Shader, R.I.5    Paul, S.M.6
  • 39
    • 0023762604 scopus 로고
    • Chronic benzodiazepine administration: I. Tolerance is associated with benzodiazepine receptor downregulation and decreased gamma-aminobutyric acid receptor function
    • Miller L.G., Greenblatt D.J., Barnhill J.G., Shader R.I. Chronic benzodiazepine administration: I. Tolerance is associated with benzodiazepine receptor downregulation and decreased gamma-aminobutyric acid receptor function. J. Pharmacol. Exp. Ther. 246:1988;170-176.
    • (1988) J. Pharmacol. Exp. Ther. , vol.246 , pp. 170-176
    • Miller, L.G.1    Greenblatt, D.J.2    Barnhill, J.G.3    Shader, R.I.4
  • 41
    • 0024438915 scopus 로고
    • Chronic benzodiazepine administration: IV. Rapid development of tolerance and receptor down regulation associated with alprazolam administration
    • Miller L.G., Woolverton S., Greenblatt D.J., Lopez F., Roy B., Shader R.I. Chronic benzodiazepine administration: IV. Rapid development of tolerance and receptor down regulation associated with alprazolam administration. Biochem. Pharmacol. 38:1989;3773-3777.
    • (1989) Biochem. Pharmacol. , vol.38 , pp. 3773-3777
    • Miller, L.G.1    Woolverton, S.2    Greenblatt, D.J.3    Lopez, F.4    Roy, B.5    Shader, R.I.6
  • 43
    • 0028283102 scopus 로고
    • Comparison of anticonvulsant tolerance, crosstolerance, and benzodiazepine receptor binding following chronic treatment with diazepam or midazolam
    • Ramsey-Williams V.A., Wu Y., Rosenberg H.C. Comparison of anticonvulsant tolerance, crosstolerance, and benzodiazepine receptor binding following chronic treatment with diazepam or midazolam. Pharmacol. Biochem. Behav. 48:1994;765-772.
    • (1994) Pharmacol. Biochem. Behav. , vol.48 , pp. 765-772
    • Ramsey-Williams, V.A.1    Wu, Y.2    Rosenberg, H.C.3
  • 44
    • 0025904589 scopus 로고
    • Binding of benzodiazepines and some major metabolites at their sites in normal human frontal cortex in vitro
    • Richelson E., Nelson A., Neeper R. Binding of benzodiazepines and some major metabolites at their sites in normal human frontal cortex in vitro. J. Pharmacol. Exp. Ther. 256:1991;897-901.
    • (1991) J. Pharmacol. Exp. Ther. , vol.256 , pp. 897-901
    • Richelson, E.1    Nelson, A.2    Neeper, R.3
  • 45
    • 0019448956 scopus 로고
    • Tolerance during chronic benzodiazepine treatment associated with decreased receptor binding
    • Rosenberg H.C., Chiu T.H. Tolerance during chronic benzodiazepine treatment associated with decreased receptor binding. Eur. J. Pharmacol. 70:1981;453-460.
    • (1981) Eur. J. Pharmacol. , vol.70 , pp. 453-460
    • Rosenberg, H.C.1    Chiu, T.H.2
  • 47
    • 0027213217 scopus 로고
    • Use of benzodiazepines in anxiety disorders
    • Shader R.I., Greenblatt D.J. Use of benzodiazepines in anxiety disorders. New Engl. J. Med. 13:1993;1398-1405.
    • (1993) New Engl. J. Med. , vol.13 , pp. 1398-1405
    • Shader, R.I.1    Greenblatt, D.J.2
  • 48
    • 21844502513 scopus 로고
    • The behavioural effects of long-term use of benzodiazepine sedative and hypnotic drugs: What can be learned from animal studies?
    • Smith P.F., Darlington C.L. The behavioural effects of long-term use of benzodiazepine sedative and hypnotic drugs: what can be learned from animal studies? New Zealand J. Psychol. 23:1994;48-63.
    • (1994) New Zealand J. Psychol. , vol.23 , pp. 48-63
    • Smith, P.F.1    Darlington, C.L.2
  • 50
    • 0003261386 scopus 로고
    • Co-planar stereotaxic atlas of the human brain
    • New York, NY
    • Talairach, J., Tournoux, P., 1988. Co-planar stereotaxic atlas of the human brain. Thieme, New York, NY.
    • (1988) Thieme
    • Talairach, J.1    Tournoux, P.2
  • 51
    • 0024349677 scopus 로고
    • Regional GABA/benzodiazepine receptor/chloride channel coupling after acute and chronic benzodiazepine treatment
    • Tietz E.I., Chiu T.H., Rosenberg H.C. Regional GABA/benzodiazepine receptor/chloride channel coupling after acute and chronic benzodiazepine treatment. Eur. J. Pharmacol. 167:1989;57-65.
    • (1989) Eur. J. Pharmacol. , vol.167 , pp. 57-65
    • Tietz, E.I.1    Chiu, T.H.2    Rosenberg, H.C.3
  • 54
    • 7144239118 scopus 로고
    • Benzodiazepines
    • In: Last, C.G., Hersen, M. (Eds.) Pergamon, New York, NY
    • Woods, S.W., Charney, D.S., 1988. Benzodiazepines. In: Last, C.G., Hersen, M. (Eds.), Handbook of Anxiety Disorders. Pergamon, New York, NY.
    • (1988) Handbook of Anxiety Disorders
    • Woods, S.W.1    Charney, D.S.2
  • 55
    • 0344374013 scopus 로고
    • Sterility tests (71)
    • USP XXIII United States Pharmacopeial Convention, Rockville, MD
    • USP XXIII, 1995. Sterility tests (71). In: The United States Pharmacopeia, 23rd Revision, United States Pharmacopeial Convention, Rockville, MD, pp. 1686-1690.
    • (1995) In: The United States Pharmacopeia, 23rd Revision , pp. 1686-1690


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.