One pot synthesis of (±)/(S)-atenolol and (±)/(S)-propranolol by employing polymer supported reagent

Synthetic Communications

Volumn 29, Issue 10, 1999, Pages 1639-1644

  Damle, Subhash V ^a   Patil, Prashant N ^a   Salunkhe, Manikrao M ^a  

^a INSTITUTE OF SCIENCE   (India)

Author keywords

[No Author keywords available]

Indexed keywords

ANION; ATENOLOL; EPICHLOROHYDRIN; ISOPROPYLAMINE; POLYMER; PROPRANOLOL; PROPYLAMINE; REAGENT; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS; REACTION ANALYSIS;

EID: 0033009451     PISSN: 00397911     EISSN: None     Source Type: Journal    
DOI: 10.1080/00397919908086148     Document Type: Article

References (16)

1. Schmalk ,S.J. and Zimmer, H. Synthesis 1984 ,29.
2. Deegan, A. ; Hull, R. ; Warren, P. and Smith L.H., U. S. Pat., 1,391 444, 1975; C.A.: 83: 9783v.
3. Capler, V. Anal. Profiles Drugs Subt. 1984, 13, 1.
4. Smith ,L. H. Brit., 1,079,534, 1967; C.A.: 67: 99907u.
5. a) Nelson, W. L. and Burke T. R. J. Org. Chem. 1978, 43, 3641.
6. b) Howe, R. and Rao, B. S. J. Med. Chem. 1968, 11, 1118.
7. a) Noritada, M. and Nobuo, O. Tetrahedron Lett. 1985, 26 (45), 5533.
8. b) Bevinakatti H. S. and Banerji A. A. J. Org. Chem. 1991, 56 (18), 5372.
9. Takahashi H. ; Sakuraba S. ; Takeda H. And Achiwa K. J. Am. Chem. Soc 1990, 112(15), 5876.
10. Klunder J. M. ; Ko S. Y. and Sharpless K. B. J. Org. Chem. 1986, 51, 3710.
11. Veloo R. A. and Koomen G. J. Tetrahedron Asymmetry 1993, 4 (12), 2401.
12. Kitaori K. ; Takehira Y. ; Furukawa Y. ; Yoshimoto H. and Otera J. Chem. Pharm. Bull. 1997, 45 (2), 412.
13. Phillips G. T. ; Bertola M. A. ; Friedrich M. A. and Simon K. H. Eur. Pat. Appl. 256, 586 ; 24 Feb 1988. C. A.: 110: 78
14. Bevinakatti H. S. and Banerji A. A. J. Org. Chem. 1992, 57 (22), 6003.
15. Ford, W. T. "Polymeric Reagents and Catalysis", American Chemical Society", Washington, D.C.,1986, pp. 12.
16. Lednicer, D and Mitscher, L. A. "The Organic Chemistry of Drug Synthesis, John Wiley and Sons; New york, 1980, 2, pp. 109.