-
1
-
-
0031438735
-
Diastereoselective synthesis of the nonracemic methyl syn-(3-fluoroalkyl)isoserinates
-
Abouabdellah A, Bégué J-P, Bonnet-Delpon D, Nga TTT (1997) Diastereoselective synthesis of the nonracemic methyl syn-(3-fluoroalkyl)isoserinates. J Org Chem 62: 8826-8833
-
(1997)
J Org Chem
, vol.62
, pp. 8826-8833
-
-
Abouabdellah, A.1
Bégué, J.-P.2
Bonnet-Delpon, D.3
Nga, T.T.T.4
-
3
-
-
0027527844
-
Stereoselective synthesis of azetidin-2-ones precursors of biologically active syn-3-amino-2-hydroxybutanoic acids
-
Annunziata R, Benaglia M, Cinquini M, Cozzi F, Ponzini F (1993) Stereoselective synthesis of azetidin-2-ones precursors of biologically active syn-3-amino-2-hydroxybutanoic acids. J Org Chem 58: 4746-4748
-
(1993)
J Org Chem
, vol.58
, pp. 4746-4748
-
-
Annunziata, R.1
Benaglia, M.2
Cinquini, M.3
Cozzi, F.4
Ponzini, F.5
-
6
-
-
0028914757
-
Carbon based nucleophilic ring opening of activated monocyclic β-lactams; synthesis and stereochemical assignments of the ACE inhibitor WF-10129
-
Baldwin JE, Adlington RM, Russell AT, Smith ML (1995) Carbon based nucleophilic ring opening of activated monocyclic β-lactams; synthesis and stereochemical assignments of the ACE inhibitor WF-10129. Tetrahedron 51: 4733-4762
-
(1995)
Tetrahedron
, vol.51
, pp. 4733-4762
-
-
Baldwin, J.E.1
Adlington, R.M.2
Russell, A.T.3
Smith, M.L.4
-
8
-
-
14844312173
-
Asymmetric synthesis of β-amino acids and α-substituted β-amino acids
-
Cardillo G, Tomasini C (1996) Asymmetric synthesis of β-amino acids and α-substituted β-amino acids. Chem Soc Rev 25: 117-128
-
(1996)
Chem Soc Rev
, vol.25
, pp. 117-128
-
-
Cardillo, G.1
Tomasini, C.2
-
9
-
-
0028130028
-
Recent stereoselective synthetic approaches to β-amino acids
-
Cole DC (1994) Recent stereoselective synthetic approaches to β-amino acids. Tetrahedron 50: 9517-9582
-
(1994)
Tetrahedron
, vol.50
, pp. 9517-9582
-
-
Cole, D.C.1
-
10
-
-
0030577473
-
A new and quantitative synthesis of α-amino acid N-carboxy anhydrides (oxazolidine-2,5-diones)
-
Collet H, Bied C, Mion L, Taillades J, Commeyras A (1996) A new and quantitative synthesis of α-amino acid N-carboxy anhydrides (oxazolidine-2,5-diones). Tetrahedron Lett 37: 9043-9046
-
(1996)
Tetrahedron Lett
, vol.37
, pp. 9043-9046
-
-
Collet, H.1
Bied, C.2
Mion, L.3
Taillades, J.4
Commeyras, A.5
-
11
-
-
0023887955
-
Synthetic utility of azetidin-2,3-diones: A new approach to 3-hydroxyethyl-β-lactams and α-amino acid derivatives
-
Cossío FP, López C, Oiarbide M, Palomo C, Aparicio D, Rubiales G (1988) Synthetic utility of azetidin-2,3-diones: a new approach to 3-hydroxyethyl-β-lactams and α-amino acid derivatives. Tetrahedron Lett 29: 3133-3136
-
(1988)
Tetrahedron Lett
, vol.29
, pp. 3133-3136
-
-
Cossío, F.P.1
López, C.2
Oiarbide, M.3
Palomo, C.4
Aparicio, D.5
Rubiales, G.6
-
13
-
-
45549112115
-
The preparation of N-carboxy anhydrides of α-amino acids using bis(trichloromethyl)carbonate
-
Daly WH, Poche D (1988) The preparation of N-carboxy anhydrides of α-amino acids using bis(trichloromethyl)carbonate. Tetrahedron Lett 29: 5859-5862
-
(1988)
Tetrahedron Lett
, vol.29
, pp. 5859-5862
-
-
Daly, W.H.1
Poche, D.2
-
14
-
-
0024249184
-
Design of peptides and proteins
-
Degrado WF (1998) Design of peptides and proteins. Adv Protein Chem 39: 51-124
-
(1998)
Adv Protein Chem
, vol.39
, pp. 51-124
-
-
Degrado, W.F.1
-
15
-
-
0015827211
-
Synthesis of β-amino-acid peptides by aminolysis of substituted dihydro-1,3-oxazinones and amino-protected β-lactams
-
Drey CNC, Lawbridge J, Ridge RJ (1973) Synthesis of β-amino-acid peptides by aminolysis of substituted dihydro-1,3-oxazinones and amino-protected β-lactams. J Chem Soc Perkin Trans 1: 2001-2006
-
(1973)
J Chem Soc Perkin Trans
, vol.1
, pp. 2001-2006
-
-
Drey, C.N.C.1
Lawbridge, J.2
Ridge, R.J.3
-
16
-
-
0028355337
-
Recent developments in the stereoselective synthesis of α-amino acids
-
Duthaler RO (1994) Recent developments in the stereoselective synthesis of α-amino acids. Tetrahedron 50: 1539-1650
-
(1994)
Tetrahedron
, vol.50
, pp. 1539-1650
-
-
Duthaler, R.O.1
-
18
-
-
0001930562
-
-
Page MI (ed) Blackie, London
-
Frére JM, Nguyen-Disteche M, Coyette J, Joris B (1992) The chemistry of β-lactams. In: Page MI (ed) Blackie, London, pp 148-197
-
(1992)
The Chemistry of β-lactams
, pp. 148-197
-
-
Frére, J.M.1
Nguyen-Disteche, M.2
Coyette, J.3
Joris, B.4
-
19
-
-
0026642114
-
N-Methyl N-carboxyanhydride: An unexpected by-product when coupling Boc-N-methyl amino acids
-
Frerort E, Coste J, Poncot J, Jouin P (1992) N-Methyl N-carboxyanhydride: an unexpected by-product when coupling Boc-N-methyl amino acids. Tetrahedron Lett 33: 2815-2816
-
(1992)
Tetrahedron Lett
, vol.33
, pp. 2815-2816
-
-
Frerort, E.1
Coste, J.2
Poncot, J.3
Jouin, P.4
-
20
-
-
0025012066
-
Urethane-protected amino acid N-carboxy anhydrides and their use in peptide synthesis
-
Fuller WD, Cohen MP, Shakankareh M, Blair RK (1990) Urethane-protected amino acid N-carboxy anhydrides and their use in peptide synthesis. J Am Chem Soc 112: 7414-7416
-
(1990)
J Am Chem Soc
, vol.112
, pp. 7414-7416
-
-
Fuller, W.D.1
Cohen, M.P.2
Shakankareh, M.3
Blair, R.K.4
-
21
-
-
0028038601
-
Peptidomimetics. Tailored enzyme inhibitors
-
Gante J (1994) Peptidomimetics. Tailored enzyme inhibitors. Angew Chem Int Ed Engl 33: 1699-1720
-
(1994)
Angew Chem Int Ed Engl
, vol.33
, pp. 1699-1720
-
-
Gante, J.1
-
23
-
-
33745502124
-
Peptidomimetics for receptor ligands. Discovery, development, and medical perspectives
-
Giannis A, Kolter T (1993) Peptidomimetics for receptor ligands. Discovery, development, and medical perspectives. Angew Chem Int Ed Engl 32: 1244-1267
-
(1993)
Angew Chem Int Ed Engl
, vol.32
, pp. 1244-1267
-
-
Giannis, A.1
Kolter, T.2
-
24
-
-
0026506915
-
Synthesis of chiral zileuton, a potent and selective inhibitor of 5-lipoxygenase
-
Hsiao Ch-N, Kolasa T (1992) Synthesis of chiral zileuton, a potent and selective inhibitor of 5-lipoxygenase. Tetrahedron Lett 33: 2629-2632
-
(1992)
Tetrahedron Lett
, vol.33
, pp. 2629-2632
-
-
Hsiao, Ch.-N.1
Kolasa, T.2
-
25
-
-
0007193238
-
Chemical synthesis of natural product peptides: Coupling methods for the incorporation of noncoded amino acids into peptides
-
Humphrey JM, Chamberlin AR (1997) Chemical synthesis of natural product peptides: coupling methods for the incorporation of noncoded amino acids into peptides. Chem Rev 97: 2243-2266
-
(1997)
Chem Rev
, vol.97
, pp. 2243-2266
-
-
Humphrey, J.M.1
Chamberlin, A.R.2
-
26
-
-
0013593057
-
Friedel-Crafts α-aminoacylation of alkylbenzene with a chiral N-carboxy-α-amino acid anhydride without loss of chirality
-
Itoh O, Honnami T, Amiano A, Muruta K, Koichi Y, Sugita T (1992) Friedel-Crafts α-aminoacylation of alkylbenzene with a chiral N-carboxy-α-amino acid anhydride without loss of chirality. J Org Chem 57: 7334-7338
-
(1992)
J Org Chem
, vol.57
, pp. 7334-7338
-
-
Itoh, O.1
Honnami, T.2
Amiano, A.3
Muruta, K.4
Koichi, Y.5
Sugita, T.6
-
27
-
-
0028266056
-
Efficient asymmetric synthesis of cis-4-formyl β-lactams from L-(+)-tartaric acid
-
Jayaraman M, Deshmukh ARAS, Bhawal BM (1994) Efficient asymmetric synthesis of cis-4-formyl β-lactams from L-(+)-tartaric acid. J Org Chem 59: 932-934
-
(1994)
J Org Chem
, vol.59
, pp. 932-934
-
-
Jayaraman, M.1
Deshmukh, A.R.A.S.2
Bhawal, B.M.3
-
29
-
-
0030766109
-
β-Peptides: Novel secondary structures take shape
-
Koert U (1997) β-Peptides: novel secondary structures take shape. Angew Chem Int Ed Engl 36: 1836-1837
-
(1997)
Angew Chem Int Ed Engl
, vol.36
, pp. 1836-1837
-
-
Koert, U.1
-
30
-
-
0031468514
-
Antiparallel sheet formation in β-peptide foldamers: Effects of β-amino acid substitution on conformational preference
-
Krauthäuser S, Christianson LA, Powell DR, Gellman SH (1997) Antiparallel sheet formation in β-peptide foldamers: effects of β-amino acid substitution on conformational preference. J Am Chem Soc 119: 11719-11720
-
(1997)
J Am Chem Soc
, vol.119
, pp. 11719-11720
-
-
Krauthäuser, S.1
Christianson, L.A.2
Powell, D.R.3
Gellman, S.H.4
-
32
-
-
0013534646
-
Conformationally restricted amino acids and dipeptides, (non)peptidomimetics and secondary structure mimetics
-
Liskamp RMJ (1994) Conformationally restricted amino acids and dipeptides, (non)peptidomimetics and secondary structure mimetics. Recuell Trav Chim Pays Bas 113: 1-19
-
(1994)
Recuell Trav Chim Pays Bas
, vol.113
, pp. 1-19
-
-
Liskamp, R.M.J.1
-
33
-
-
0001197816
-
Conversion of β-lactams to versatile synthons via molecular rearrangement and lactam cleavage
-
Manhas MS, Wagle DR, Chang J, Bose AK (1988) Conversion of β-lactams to versatile synthons via molecular rearrangement and lactam cleavage. Heterocycles 27: 1755-1802
-
(1988)
Heterocycles
, vol.27
, pp. 1755-1802
-
-
Manhas, M.S.1
Wagle, D.R.2
Chang, J.3
Bose, A.K.4
-
34
-
-
0018189163
-
β-Lactams: Retrospect and prospect
-
Mukerjee AK, Singh AK (1978) β-Lactams: retrospect and prospect. Tetrahedron 34: 1731-1767
-
(1978)
Tetrahedron
, vol.34
, pp. 1731-1767
-
-
Mukerjee, A.K.1
Singh, A.K.2
-
35
-
-
0002738175
-
-
Page MT (ed) Blackie, London
-
Neu HC (1992) The chemistry of β-lactams In: Page MT (ed) Blackie, London, pp 101-128
-
(1992)
The Chemistry of β-lactams
, pp. 101-128
-
-
Neu, H.C.1
-
36
-
-
0001039009
-
α-Amino acid synthesis. Tetrahedron symposia
-
O'Donell (1988) α-Amino acid synthesis. Tetrahedron symposia. Tetrahedron 44: 5253-5614
-
(1988)
Tetrahedron
, vol.44
, pp. 5253-5614
-
-
O'Donell1
-
37
-
-
0000096261
-
Recent advances in the β-lactam synthon method
-
Ojima I (1995) Recent advances in the β-lactam synthon method. Acc Chem Res 28: 383-389
-
(1995)
Acc Chem Res
, vol.28
, pp. 383-389
-
-
Ojima, I.1
-
38
-
-
0000727123
-
Asymmetric synthesis of building-blocks for peptide and peptidomimetics by means of the β-lactam synthon method
-
Ojima I, Delaloge F (1997) Asymmetric synthesis of building-blocks for peptide and peptidomimetics by means of the β-lactam synthon method. Chem Soc Rev 26: 377-386
-
(1997)
Chem Soc Rev
, vol.26
, pp. 377-386
-
-
Ojima, I.1
Delaloge, F.2
-
39
-
-
0026686518
-
New and efficient approaches to the semisynthesis of taxol and its C-13 side chain analogs by means of β-lactam synthon method
-
Ojima I, Habus I, Zhao M, Zucco M, Park YH, Sun CM, Brigand T (1992) New and efficient approaches to the semisynthesis of taxol and its C-13 side chain analogs by means of β-lactam synthon method. Tetrahedron 48: 6985-7012
-
(1992)
Tetrahedron
, vol.48
, pp. 6985-7012
-
-
Ojima, I.1
Habus, I.2
Zhao, M.3
Zucco, M.4
Park, Y.H.5
Sun, C.M.6
Brigand, T.7
-
40
-
-
0029655687
-
Synthesis of new fluorine-containing taxoids by means of β-lactam synthon method
-
Ojima I, Kuduk SA, Slater JC, Gimi RH, Sun CM (1996) Synthesis of new fluorine-containing taxoids by means of β-lactam synthon method. Tetrahedron 52: 209-224
-
(1996)
Tetrahedron
, vol.52
, pp. 209-224
-
-
Ojima, I.1
Kuduk, S.A.2
Slater, J.C.3
Gimi, R.H.4
Sun, C.M.5
-
42
-
-
0002796008
-
-
Page MI (ed) Blackie, London
-
Page MI (1992) The chemistry of β-lactams. In: Page MI (ed) Blackie, London, pp 79-100, 129-147
-
(1992)
The Chemistry of β-lactams
, pp. 79-100
-
-
Page, M.I.1
-
43
-
-
0032555436
-
The mechanism of catalysis and the inhibition of β-lactamases
-
Page MI, Laws AP (1998) The mechanism of catalysis and the inhibition of β-lactamases. Chem Commun 1609-1617
-
(1998)
Chem Commun
, pp. 1609-1617
-
-
Page, M.I.1
Laws, A.P.2
-
44
-
-
0027076852
-
Contribution to the development of new substitution patterns of optically active β-lactams: Synthesis of homochiral 4-(1-aminoalkyl)azetidin-2-ones from N-(tert-butyloxycarbonyl) α-amino aldehyde-derived imines via asymmetric Staudinger reaction
-
Palomo C, Cossío FP, Cuevas C, Lecea B, Mielgo A, Román P, Luque A, Martínez-Ripoll M (1992) Contribution to the development of new substitution patterns of optically active β-lactams: synthesis of homochiral 4-(1-aminoalkyl)azetidin-2-ones from N-(tert-butyloxycarbonyl) α-amino aldehyde-derived imines via asymmetric Staudinger reaction. J Am Chem Soc 114: 9360-9369
-
(1992)
J Am Chem Soc
, vol.114
, pp. 9360-9369
-
-
Palomo, C.1
Cossío, F.P.2
Cuevas, C.3
Lecea, B.4
Mielgo, A.5
Román, P.6
Luque, A.7
Martínez-Ripoll, M.8
-
45
-
-
0028296561
-
From (S)-α-amino β-hydroxy acids to (R)-α,β-diamino-γ-hydroxy N-Carboxy anhydrides via β-lactams
-
Palomo C, Aizpurua JM, Cabré F, Cuevas C, Munt S, Odriozola JM (1994a) From (S)-α-amino β-hydroxy acids to (R)-α,β-diamino-γ-hydroxy N-Carboxy anhydrides via β-lactams. Tetrahedron Lett 35: 2725-2728
-
(1994)
Tetrahedron Lett
, vol.35
, pp. 2725-2728
-
-
Palomo, C.1
Aizpurua, J.M.2
Cabré, F.3
Cuevas, C.4
Munt, S.5
Odriozola, J.M.6
-
46
-
-
0028348213
-
Synthesis of β-alkylserine-N-carboxy anhydrides through β-lactams via cycloaddition reaction of alkoxyketenes to chiral α-alkoxy aldehyde-derived imines
-
Palomo C, Aizpurua JM, Cabré F, García JM, Odriozola JM (1994b) Synthesis of β-alkylserine-N-carboxy anhydrides through β-lactams via cycloaddition reaction of alkoxyketenes to chiral α-alkoxy aldehyde-derived imines. Tetrahedron Lett 35: 2721-2724
-
(1994)
Tetrahedron Lett
, vol.35
, pp. 2721-2724
-
-
Palomo, C.1
Aizpurua, J.M.2
Cabré, F.3
García, J.M.4
Odriozola, J.M.5
-
47
-
-
37049070296
-
A β-lactam framework as a β-alanyl dication equivalent: New synthesis of α-amino acid N-carboxy anhydrides (NCAs) derived from β-substituled alanines
-
Palomo C, Aizpurua JM, Ganboa I, Maneiro E, Odriozola B (1994c) A β-lactam framework as a β-alanyl dication equivalent: new synthesis of α-amino acid N-carboxy anhydrides (NCAs) derived from β-substituled alanines. J Chem Soc Chem Commun: 1505-1507
-
(1994)
J Chem Soc Chem Commun
, pp. 1505-1507
-
-
Palomo, C.1
Aizpurua, J.M.2
Ganboa, I.3
Maneiro, E.4
Odriozola, B.5
-
48
-
-
0028076811
-
A route to dipeptides containing β-amino-α-hydroxy acid fragments by coupling of N-Boc-β-lactams with α-amino esters. Application to the synthesis of (-)-bestatin
-
Palomo C, Aizpurua JM, Cuevas C (1994d) A route to dipeptides containing β-amino-α-hydroxy acid fragments by coupling of N-Boc-β-lactams with α-amino esters. Application to the synthesis of (-)-bestatin. J Chem Soc Chem Commun: 1957-1958
-
(1994)
J Chem Soc Chem Commun
, pp. 1957-1958
-
-
Palomo, C.1
Aizpurua, J.M.2
Cuevas, C.3
-
49
-
-
0000411026
-
Concise general synthesis of α,γ-disubstituted β-amino ketones from β-lactams
-
Palomo C, Aizpurua JM, Garcia JM, Iturburu M, Odriozola JM (1994e) Concise general synthesis of α,γ-disubstituted β-amino ketones from β-lactams. J Org Chem 59: 5184-5188
-
(1994)
J Org Chem
, vol.59
, pp. 5184-5188
-
-
Palomo, C.1
Aizpurua, J.M.2
Garcia, J.M.3
Iturburu, M.4
Odriozola, J.M.5
-
50
-
-
0028791544
-
A facile access to peptides containing D-α-methyl β-alkylserines by coupling of α-branched Leuchs anhydrides with α-amino esters
-
Palomo C, Aizpurua JM, Urchegui R, García JM (1995a) A facile access to peptides containing D-α-methyl β-alkylserines by coupling of α-branched Leuchs anhydrides with α-amino esters. J Chem Soc Chem Commun: 2327-2328
-
(1995)
J Chem Soc Chem Commun
, pp. 2327-2328
-
-
Palomo, C.1
Aizpurua, J.M.2
Urchegui, R.3
García, J.M.4
-
51
-
-
0028877350
-
A mild method for the alcoholysis of β-lactams
-
Palomo C, Aizpurua JM, Cuevas C, Mielgo A, Galarza R (1995b) A mild method for the alcoholysis of β-lactams. Tetrahedron Lett 36: 9027-9030
-
(1995)
Tetrahedron Lett
, vol.36
, pp. 9027-9030
-
-
Palomo, C.1
Aizpurua, J.M.2
Cuevas, C.3
Mielgo, A.4
Galarza, R.5
-
52
-
-
0030018754
-
Generation of threonine and azathreonine N-carboxy anhydrides from α-hydroxy β-lactams promoted by 2,2,6,6-tetramethylpiperidinyl-l-oxyl (TEMPO) in combination with sodium hypochlorite
-
Palomo C, Aizpurua JM, Cuevas C, Urchegui R, Linden A (1996a) Generation of threonine and azathreonine N-carboxy anhydrides from α-hydroxy β-lactams promoted by 2,2,6,6-tetramethylpiperidinyl-l-oxyl (TEMPO) in combination with sodium hypochlorite. J Org Chem 61: 4400-4404
-
(1996)
J Org Chem
, vol.61
, pp. 4400-4404
-
-
Palomo, C.1
Aizpurua, J.M.2
Cuevas, C.3
Urchegui, R.4
Linden, A.5
-
53
-
-
0030039884
-
Simple access to the nonproteinogenic peptide fragments of lysobactin from azetidin-2-one frameworks
-
Palomo C, Aizpurua JM, Ganboa I, Odriozola B, Maneiro M, Miranda JI, Urchegui R (1996b) Simple access to the nonproteinogenic peptide fragments of lysobactin from azetidin-2-one frameworks. Chem Commun: 161-162
-
(1996)
Chem Commun
, pp. 161-162
-
-
Palomo, C.1
Aizpurua, J.M.2
Ganboa, I.3
Odriozola, B.4
Maneiro, M.5
Miranda, J.I.6
Urchegui, R.7
-
54
-
-
0029903149
-
Concise synthesis of α-alkyl α-amino acids and their incorporation into peptides via β-lactam-derived α-amino acid N-carboxy anhydrides
-
Palomo C, Aizpurua JM, Ganboa I, Odriozola B, Urchegui R, Gorls H (1996c) Concise synthesis of α-alkyl α-amino acids and their incorporation into peptides via β-lactam-derived α-amino acid N-carboxy anhydrides. Chem Commun: 1269-1270
-
(1996)
Chem Commun
, pp. 1269-1270
-
-
Palomo, C.1
Aizpurua, J.M.2
Ganboa, I.3
Odriozola, B.4
Urchegui, R.5
Gorls, H.6
-
55
-
-
0029790915
-
Imine substituent effects on [2 + 2]cycloadditions with ketenes
-
Palomo C, Aizpurua JM, Legido M, Galarza R, Deyá P, Dunogues J, Picard JP, Ricci A, Seconi G (1996d) Imine substituent effects on [2 + 2]cycloadditions with ketenes. Angew Chem Int Ed Engl 35: 1239-1241
-
(1996)
Angew Chem Int Ed Engl
, vol.35
, pp. 1239-1241
-
-
Palomo, C.1
Aizpurua, J.M.2
Legido, M.3
Galarza, R.4
Deyá, P.5
Dunogues, J.6
Picard, J.P.7
Ricci, A.8
Seconi, G.9
-
56
-
-
0029877120
-
A new and versatile procedure for the incorporation of α,β-diamino acids into peptides
-
Palomo C, Aizpurua JM, Galarza R, Mielgo A (1996e) A new and versatile procedure for the incorporation of α,β-diamino acids into peptides. Chem Commun: 633-634
-
(1996)
Chem Commun
, pp. 633-634
-
-
Palomo, C.1
Aizpurua, J.M.2
Galarza, R.3
Mielgo, A.4
-
58
-
-
0030989647
-
A concise synthesis of piperazine-2-carboxylic acids via β-lactam-derived α-amino acid N-carboxy anhydrides
-
Palomo C, Ganboa I, Cuevas C, Boschetti C, Linden A (1997b) A concise synthesis of piperazine-2-carboxylic acids via β-lactam-derived α-amino acid N-carboxy anhydrides. Tetrahedron Lett 38: 4643-4646
-
(1997)
Tetrahedron Lett
, vol.38
, pp. 4643-4646
-
-
Palomo, C.1
Ganboa, I.2
Cuevas, C.3
Boschetti, C.4
Linden, A.5
-
59
-
-
8244235132
-
Construction of quaternary stereogenic centers via [2 + 2] cycloaddition reactions. Synthesis of homochiral 4,4-disubstituted 2-azetidinones and imine substituent effects on β-lactam formation
-
Palomo C, Aizpurua JM, García JM, Galarza R, Legido M, Urchegui R, Román P, Luque A, Server-Carro J, Linden A (1997c) Construction of quaternary stereogenic centers via [2 + 2] cycloaddition reactions. Synthesis of homochiral 4,4-disubstituted 2-azetidinones and imine substituent effects on β-lactam formation. J Org Chem 62: 2070-2079
-
(1997)
J Org Chem
, vol.62
, pp. 2070-2079
-
-
Palomo, C.1
Aizpurua, J.M.2
García, J.M.3
Galarza, R.4
Legido, M.5
Urchegui, R.6
Román, P.7
Luque, A.8
Server-Carro, J.9
Linden, A.10
-
60
-
-
0030947166
-
Synthetic studies towards peptidyl nucleoside antibiotics: First synthesis of a polyoxamic derivative enabling direct coupling with α-amino acid esters
-
Palomo C, Oiarbide M, Esnal A (1997d) Synthetic studies towards peptidyl nucleoside antibiotics: first synthesis of a polyoxamic derivative enabling direct coupling with α-amino acid esters. J Chem Soc Chem Commun: 691-692
-
(1997)
J Chem Soc Chem Commun
, pp. 691-692
-
-
Palomo, C.1
Oiarbide, M.2
Esnal, A.3
-
61
-
-
0030890690
-
Synthesis of (S)- and (R)-tertleucine enabling direct coupling with α-amino acid esters via β-lactam-derived α-amino acid N-carboxy anhydrides
-
Palomo C, Ganboa I, Odriozola B, Linden A (1997e) Synthesis of (S)- and (R)-tertleucine enabling direct coupling with α-amino acid esters via β-lactam-derived α-amino acid N-carboxy anhydrides. Tetrahedron Lett 38: 3093-3097
-
(1997)
Tetrahedron Lett
, vol.38
, pp. 3093-3097
-
-
Palomo, C.1
Ganboa, I.2
Odriozola, B.3
Linden, A.4
-
62
-
-
0030870477
-
A contribution to the asymmetric synthesis of 3-amino β-lactams: The diastereoselective [2 + 2] cycloaddition reaction of chiral aminoketene equivalents with enolizable aldehyde-derived imines
-
Palomo C, Aizpurua JM, Legido M, Mielgo A, Galarza R (1997f) A contribution to the asymmetric synthesis of 3-amino β-lactams: the diastereoselective [2 + 2] cycloaddition reaction of chiral aminoketene equivalents with enolizable aldehyde-derived imines. Chem Eur J 3: 1432-1441
-
(1997)
Chem Eur J
, vol.3
, pp. 1432-1441
-
-
Palomo, C.1
Aizpurua, J.M.2
Legido, M.3
Mielgo, A.4
Galarza, R.5
-
63
-
-
0032555405
-
Practical synthesis of α-amino acid N-carboxy anhydrides of polyhydroxylated α-amino acids from β-lactam frameworks. Model studies towards the synthesis of directly linked peptidyl nucleoside antibiotics
-
Palomo C, Oiarbide M, Esnal A, Landa A, Miranda JI, Linden A (1998a) Practical synthesis of α-amino acid N-carboxy anhydrides of polyhydroxylated α-amino acids from β-lactam frameworks. Model studies towards the synthesis of directly linked peptidyl nucleoside antibiotics. J Org Chem 63: 5838-5846
-
(1998)
J Org Chem
, vol.63
, pp. 5838-5846
-
-
Palomo, C.1
Oiarbide, M.2
Esnal, A.3
Landa, A.4
Miranda, J.I.5
Linden, A.6
-
64
-
-
0001448817
-
A concise β-lactam route to short peptide segments containing β,β-disubstituted β-amino acids
-
Palomo C, Oiarbide M, Bindi S (1998b) A concise β-lactam route to short peptide segments containing β,β-disubstituted β-amino acids. J Org Chem 63: 2469-2474
-
(1998)
J Org Chem
, vol.63
, pp. 2469-2474
-
-
Palomo, C.1
Oiarbide, M.2
Bindi, S.3
-
65
-
-
0032573890
-
Total synthesis of the novel immunosupressive agent (-)-panteamine A from mycale sp. Employing a β-lactam-based macrocyclization
-
Rzasa RM, Shea HA, Romo D (1998) Total synthesis of the novel immunosupressive agent (-)-panteamine A from mycale sp. employing a β-lactam-based macrocyclization. J Am Chem Soc 120: 591-592
-
(1998)
J Am Chem Soc
, vol.120
, pp. 591-592
-
-
Rzasa, R.M.1
Shea, H.A.2
Romo, D.3
-
67
-
-
37049075008
-
N-Alkoxycarbonyl amino acid N-carboxy anhydrides and N,N-dialkoxycarbonyl amino acid fluorides from N,N-diprotected amino acids
-
Savrda J, Wakselman MJ (1992) N-Alkoxycarbonyl amino acid N-carboxy anhydrides and N,N-dialkoxycarbonyl amino acid fluorides from N,N-diprotected amino acids. J Chem Soc Chem Commun: 812-813
-
(1992)
J Chem Soc Chem Commun
, pp. 812-813
-
-
Savrda, J.1
Wakselman, M.J.2
-
68
-
-
0026599529
-
Peptide modification by introduction of α-trifluoromethyl α-amino acids via 4-trifluoromethyl-1,3-oxazolidin-2,5-diones
-
Schierlinger C, Burger K (1992) Peptide modification by introduction of α-trifluoromethyl α-amino acids via 4-trifluoromethyl-1,3-oxazolidin-2,5-diones. Tetrahedron Lett 33: 193-194
-
(1992)
Tetrahedron Lett
, vol.33
, pp. 193-194
-
-
Schierlinger, C.1
Burger, K.2
-
69
-
-
0030785114
-
β-Peptides: A surprise at every turn
-
Seebach D, Matthews JL (1997) β-Peptides: a surprise at every turn. Chem Commun: 2015-2022
-
(1997)
Chem Commun
, pp. 2015-2022
-
-
Seebach, D.1
Matthews, J.L.2
-
70
-
-
84987279356
-
III-catalyzed acetalizations of aldehydes with urethane-protected serine and threonine esters and with dipeptides containing serine or threonine residues at the N-terminus
-
III-catalyzed acetalizations of aldehydes with urethane-protected serine and threonine esters and with dipeptides containing serine or threonine residues at the N-terminus. Helv Chim Acta 77: 1313-1330
-
(1994)
Helv Chim Acta
, vol.77
, pp. 1313-1330
-
-
Seebach, D.1
Sommerfeld, T.L.2
Jiang, Q.3
Venanci, L.M.4
-
72
-
-
0029022534
-
Enantioselective synthesis of the (syn,anti)-1-amino-2,3-diol subunit of renin inhibitors by reaction of β-lactams with a Grignard reagent
-
Spero DM, Kapadia S, Farina V (1995) Enantioselective synthesis of the (syn,anti)-1-amino-2,3-diol subunit of renin inhibitors by reaction of β-lactams with a Grignard reagent. Tetrahedron Lett 36: 4543-4546
-
(1995)
Tetrahedron Lett
, vol.36
, pp. 4543-4546
-
-
Spero, D.M.1
Kapadia, S.2
Farina, V.3
-
73
-
-
0025370346
-
Conformationally restricted peptides through short-range cyclizations
-
Toniolo C (1990) Conformationally restricted peptides through short-range cyclizations. Int Peptide Protein Res 35: 287-300
-
(1990)
Int Peptide Protein Res
, vol.35
, pp. 287-300
-
-
Toniolo, C.1
-
74
-
-
0001318920
-
Studies on lactams: Enantispecific synthesis and absolute configuration of substituted β-lactams from D-gliceraldehyde acetonide
-
Wagle DR, Garai G, Chiang J, Monteleone MG, Kurys BE, Strohmeyer TW, Hedge VR, Manhas MS, Bose AK (1988) Studies on lactams: enantispecific synthesis and absolute configuration of substituted β-lactams from D-gliceraldehyde acetonide. J Org Chem 53: 4227-4236
-
(1988)
J Org Chem
, vol.53
, pp. 4227-4236
-
-
Wagle, D.R.1
Garai, G.2
Chiang, J.3
Monteleone, M.G.4
Kurys, B.E.5
Strohmeyer, T.W.6
Hedge, V.R.7
Manhas, M.S.8
Bose, A.K.9
-
76
-
-
0001468317
-
The use of triphosgene in prepration of N-carboxy-α-amino acid anhydrides
-
Wilder R, Mobashery S (1992) The use of triphosgene in prepration of N-carboxy-α-amino acid anhydrides. J Org Chem 57: 2755-2756
-
(1992)
J Org Chem
, vol.57
, pp. 2755-2756
-
-
Wilder, R.1
Mobashery, S.2
-
78
-
-
0029073801
-
Pseudo-prolines in peptide synthesis: Direct insertion of serine and threonine derived oxazolidines in dipeptides
-
Wohr T, Mutter M (1995) Pseudo-prolines in peptide synthesis: direct insertion of serine and threonine derived oxazolidines in dipeptides. Tetrahedron Lett 36: 3847-3848
-
(1995)
Tetrahedron Lett
, vol.36
, pp. 3847-3848
-
-
Wohr, T.1
Mutter, M.2
-
79
-
-
0000836324
-
Application of N-(tert-butyloxycarbonyl)amino acid N-carboxyanhydrides in solid-phase peptide synthesis
-
Xue Ch-B, Naider F (1993) Application of N-(tert-butyloxycarbonyl)amino acid N-carboxyanhydrides in solid-phase peptide synthesis. J Org Chem 58: 350-355
-
(1993)
J Org Chem
, vol.58
, pp. 350-355
-
-
Xue, Ch.-B.1
Naider, F.2
|