An analysis of solute structure-human epidermal transport relationships in epidermal iontophoresis using the ionic mobility: Pore model

Journal of Controlled Release

Volumn 58, Issue 3, 1999, Pages 323-333

  Lai, Pamela M ^a   Roberts, Michael S ^a  

^a UNIVERSITY OF QUEENSLAND   (Australia)

Author keywords

Free volume; Hydration; Ionic mobility; Iontophoresis; Pore model

Indexed keywords

CALCIUM ION; CATION; CHLORIDE; DICLOFENAC; FLUOROURACIL; GLUCOSE; HYDROCORTISONE; INDOMETACIN; INSULIN DERIVATIVE; LIDOCAINE; LITHIUM ION; MAGNESIUM ION; NAPROXEN; PEPTIDE; PHENAZONE; PHENETHYLAMINE; PHENOL; POTASSIUM ION; PROGESTERONE; PROPRANOLOL; SALICYLIC ACID; SPIPERONE; SUCROSE;

ARTICLE; CONDUCTANCE; IONTOPHORESIS; MODEL; PRIORITY JOURNAL; SKIN PERMEABILITY; THEORY;

EPIDERMIS; HUMANS; IONTOPHORESIS; MEMBRANES, ARTIFICIAL; MODELS, BIOLOGICAL;

EID: 0033003071     PISSN: 01683659     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0168-3659(98)00172-2     Document Type: Article

References (28)

1. M.S. Roberts, J. Singh, N. Yoshida, K.I. Currie, Iontophoretic transport of selected solutes through human epidermis, in: R.C. Scott, J. Hadgraft, R. Guy (Eds.), Prediction of Percutaneous Absorption, IBC, London, 1990, pp 231-241.
2. Phipps J.B., Gyory J.R. Transdermal ion migration. Adv. Drug Deliv. Rev. 9:1992;137-176.
3. Yoshida N.H., Roberts M.S. Solute molecular size and transdermal iontophoresis across excised human skin. J. Control. Release. 25:1993;177-195.
4. Yoshida N.H., Roberts M.S. Role of conductivity in iontophoresis. 2. Anodal iontophoretic transport of phenylethylamine and sodium across excised human skin. J. Pharm. Sci. 83:1994;344-350.
5. Yoshida N.H., Roberts M.S. Prediction of cathodal iontophoretic transport of various anions across excised skin from different vehicles using conductivity measurements. J. Pharm. Pharmacol. 47:1995;883-890.
6. Dinh S., Luo C.W., Berner B. Upper and lower limits of human skin electrical resistance in iontophoresis. Am. Inst. Chem. Eng. J. 39:1993;2011-2018.
7. Hirvonen J., Guy R.H. Iontophoretic delivery across the skin: electroosmosis and its modulation by drug substances. Pharm. Res. 14:1997;1258-1263.
8. Burnette R.R., Ongpipattanakul B. Characterisation of permselective properties of excised human skin through iontophoresis. J. Pharm. Sci. 76:1987;765-773.
9. Phipps J.B., Padmanabham R.V., Lattin G.A. Iontophoretic delivery of model inorganic and drug ions. J. Pharm. Sci. 78:1989;365-369.
10. Pikal M.J. The role of electroosmotic flow in transdermal iontophoresis. Adv. Drug Deliv. Rev. 9:1992;201-237.
11. Roberts M.S., Lai P.M., Anissimov Y.G. Epidermal iontophoresis. I. Development of the ionic mobility-pore model. Pharm. Res. 15:1998;1569-1578.
12. Lai P.M., Roberts M.S. Epidermal iontophoresis. II. Application of the ionic mobility-pore model to the transport of local anesthetics. Pharm. Res. 15:1998;1579-1588.
13. Yoshida N.H., Roberts M.S. Structure-transport relations in transdermal iontophoresis. Adv. Drug Deliv. Rev. 9:1992;239-264.
14. Munch W.D., Zestar L.P., Anderson J.L. Rejection of polyelectrolytes from microporous membranes. J. Membr. Sci. 5:1979;77-102.
15. Deen W.M., Smith F.G. Hindered diffusion of synthetic polyelectrolytes in charged microporous membranes. J. Membr. Sci. 12:1982;217-237.
16. B.H. Sage, R.A. Hoke, A.C. McFarland, K. Kowalczyk, The importance of skin pH in the iontophoresis of peptides, in: K.R. Brain, J. Hadgraft, V.J. James, K.A. Walters (Eds), Prediction of Percutaneous Penetration, vol. 3B, 1993.
17. T. Hanai, Maku to ion, 1978, ch. 1, pp. 1-37.
18. Yalkowsky S.H., Zografi G. Calculation of partial molal volume in micellar systems. J. Pharm. Sci. 61:1972;793-795.
19. Pau P.C.F., Berg J.O., McMillan W.G. Application of Stokes' law to ions in aqueous solution. J. Phys. Chem. 94:1990;2671-2679.
20. Purves R.D. Accuracy of numerical inversion of Laplace transforms for pharmacokinetic parameter estimation. J. Pharm. Sci. 84:1995;71-74.
21. Davidson M.G., Deen W.M. Hydrodynamic theory for the hindered transport of flexible macromolecules in porous membranes. J. Membr. Sci. 35:1988;167-192.
22. Ruddy S.B., Hadzija B.A. Iontophoretic permeability of polyethylene glycols through hairless rat skin: application of hydrodynamic theory for hindered transport through liquid-filled pores. Drug Des. Discovery. 8:1992;207-224.
23. Banga A.K., Chien Y.W. Iontophoretic delivery of drugs: fundamentals, developments and biomedical applications. J. Control. Release. 7:1988;1-24.
24. Snyder E.E., Buoscio B.W., Falke J.J. Calcium(II) site specificity: effect of size and charge on metal ion binding to an EF-hand-like site. Biochemistry. 29:1990;3937-3943.
25. Bellantone N.H., Rim S., Francoeur M.L., Rasadi B. Enhanced percutaneous absorption via iontophoresis. I. Evaluation of an in vitro system and transport of model compounds. Int. J. Pharmacol. 30:1986;63-72.
26. Del Terzo S., Behl C.R., Nash R.A. Iontophoretic transport of a homologous series of ionised and nonionised model compounds: influence of hydrophobicity and mechanistic interpretation. Pharm. Res. 6:1989;85-90.
27. Burnette R.R., Marrero D. Comparison between the iontophoretic and passive transport of thyrotropin releasing hormone across excised nude mouse skin. J. Pharm. Sci. 75:1986;738-743.
28. Mukerjee P. On ion-solvent interactions. Part I. Partial molal volumes of ions in aqueous solution. J. Phys. Chem. 65:1961;740-744.