Site-selective trifluoroacetylation of dimethylamino-substituted pyridines and its use as a building block for trifluoromethyl-containing heterocycles

Chemical and Pharmaceutical Bulletin

Volumn 47, Issue 5, 1999, Pages 718-719

  Kawase, Masami ^a   Koyanagi, Jyunichi ^a   Saito, Setsuo ^a  

^a JOSAI UNIVERSITY   (Japan)

Author keywords

Dimethylaminopyridine; Pyrazolo 4,3 c pyridine; Trifluoroacetylation; Trifluoromethyl

Indexed keywords

3 TRIFLUOROMETHYLPYRAZOLO[4,3 C]PYRIDINE DERIVATIVE; PYRIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ACETYLATION; ARTICLE; NUCLEAR OVERHAUSER EFFECT; REACTION ANALYSIS; STRUCTURE ANALYSIS; SYNTHESIS;

EID: 0032991018     PISSN: 00092363     EISSN: None     Source Type: Journal    
DOI: 10.1248/cpb.47.718     Document Type: Article

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