Effect of a dynorphin a analog, E2078, on phospholipid membrane properties

Biological and Pharmaceutical Bulletin

Volumn 22, Issue 5, 1999, Pages 543-545

  Asai, Yasuyuki ^a   Watanabe, Sumio ^a  

^a EISAI CO LTD   (Japan)

Author keywords

Binding isotherm; Dynorphin A; Lipid charge; Membrane permeability

Indexed keywords

CALCEIN; DIPALMITOYLPHOSPHATIDYLGLYCEROL; DYNORPHIN A DERIVATIVE; DYNORPHIN A [1-8][1 (N METHYLTYROSINE) 7 (N METHYLARGININE) 8 DEXTRO LEUCINE N ETHYLAMIDE]; PEPTIDE; PHOSPHOLIPID;

ARTICLE; BINDING AFFINITY; BINDING SITE; CELL MEMBRANE FLUIDITY; CELL MEMBRANE PERMEABILITY; DRUG EFFECT; ELECTRICITY; LIPID COMPOSITION; MEMBRANE BINDING; MOLECULAR INTERACTION; PHOSPHOLIPID MEMBRANE; PHYSICAL CHEMISTRY;

EID: 0032976352     PISSN: 09186158     EISSN: None     Source Type: Journal    
DOI: 10.1248/bpb.22.543     Document Type: Article

References (15)

1. Goldstein A., Tachibana S., Lowney L. I., Hood M., Proc. Natl. Acad. Sci. U.S.A., 76, 6666-6670 (1979).
2. Goldstein A., Fishli W., Lowney L. I., Hankapillier M., Hood L., Proc. Natl. Acad. Sci. U.S.A., 78, 7219-7223 (1981).
3. Yoshino H., Nakazawa T., Arakawa Y., Kaneko T., Tsuchiya Y., Matsunaga M., Araki S., Ikeda M., Yamatsu K., Tachibana S., J. Med. Chem., 33, 206-212 (1990).
4. Tachibana S., Yoshino H., Arakawa Y., Nakazawa T., Araki S., Kanako T., Yamatsu K., Abstract of Papers, International Narcotics Research Conference, Adelaide, South Australia, August 1987, p. 18.
5. Matsuzaki K., Harada M., Handa T., Funakoshi S., Fujii N., Yajima H., Miyajima K., Biochim Biophys. Acta, 981, 130-134 (1989).
6. Katsu T., Kuroko M., Morikawa T., Sanchika K., Yamanaka H., Shinoda S., Fujita Y., Biochim. Biophys. Acta, 1027, 185-190 (1990).
7. Alford D. R., Rengopalakrishna V., Düzgünes N., Int. J. Pept. Protein Res., 47, 84-90 (1996).
8. Matsuzaki K., Nakai S., Handa T., Takaishi Y., Fujita T., Miyajima K., Biochemistry, 28, 9392-9398 (1989).
9. Epand R. M., Epand R. F., Orlowski R. C., Schlueter R. J., Boni L. T., Hui S. W., Biochemistry. 22, 5074-5084 (1983).
10. Bartlett G. R., J. Biol. Chem., 234, 466-468 (1959).
11. Yianni Y. P., Fitton J. E., Morgan C. G., Biochim. Biophys. Acta, 856, 91-100 (1986).
12. Iwamoto K., Sunamoto J., Inoue K., Endo T., Nojima S., Biochim. Biophys. Acta. 691, 44-51 (1982).
13. Thron C. D., J. Pharmacol. Exp. Ther., 145, 194-201 (1964).
14. Matsuzaki K., Handa T., Miyajima K., Mikura Y., Shimizu H., Toguchi H., Chem. Pharm. Bull, 36, 4253-4260 (1988).
15. Adamson A. W., "Physical Chemistry of Surfaces," 2nd ed., Interscience Publishers, New York, 1967, Chapter 8.