Synthesis and spectral properties of 5-methylthio-4H-1-(p-substituted- phenyl)-3a-(p-substituted-phenyl)-9-([(m-; and p-substituted)-phenoxyl-3a,4- dihydro[1,2,4]oxadiazolo[4,5-a][1,5]benzodiazepines

Journal of Heterocyclic Chemistry

Volumn 36, Issue 2, 1999, Pages 477-480

  Cortés, Eduardo Cortés ^a   Mellado, Olivia García ^b   Cruz, Elide Hernández ^a  

^a UNIVERSIDAD NACIONAL AUTÓNOMA DE MÉXICO   (Mexico)

^b UNIVERSIDAD NACIONAL AUTÓNOMA DE MÉXICO   (Mexico)

Author keywords

[No Author keywords available]

Indexed keywords

5 METHYLTHIO 4H 1 (4 CHLOROPHENYL) 3A (4 METHOXYPHENYL) 9 (3 METHOXYPHENOXY) 3A,4 DIHYDRO[1,2,4]OXADIAZOLO[4,5 A][1,5]BENZODIAZEPINE; BENZODIAZEPINE DERIVATIVE; UNCLASSIFIED DRUG;

CARBON NUCLEAR MAGNETIC RESONANCE; CHEMICAL REACTION; DRUG ACTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; INFRARED RADIATION; MASS SPECTROMETRY; PROTON NUCLEAR MAGNETIC RESONANCE; REVIEW;

EID: 0032898521     PISSN: 0022152X     EISSN: None     Source Type: Journal    
DOI: 10.1002/jhet.5570360224     Document Type: Review

References (23)

1. Author to whom correspondece should be addressed.
2. Contribution No. 1678 from Instituto de Química, UNAM.
3. J. B. Hester, A. D. Rudzik, and B. V. Kamdar, J. Med. Chem., 14, 1078 (1971); K. Meguro, H. Tawada, H. Miyano, Y. Sato and Y. Kuwada, Chem. Pharm. Bull., 21, 2382 (1973); A. Walser and G. Zenchoff, J. Med. Chem., 20, 1694 (1977).
4. J. B. Hester, A. D. Rudzik, and B. V. Kamdar, J. Med. Chem., 14, 1078 (1971); K. Meguro, H. Tawada, H. Miyano, Y. Sato and Y. Kuwada, Chem. Pharm. Bull., 21, 2382 (1973); A. Walser and G. Zenchoff, J. Med. Chem., 20, 1694 (1977).
5. J. B. Hester, A. D. Rudzik, and B. V. Kamdar, J. Med. Chem., 14, 1078 (1971); K. Meguro, H. Tawada, H. Miyano, Y. Sato and Y. Kuwada, Chem. Pharm. Bull., 21, 2382 (1973); A. Walser and G. Zenchoff, J. Med. Chem., 20, 1694 (1977).
6. A. Gagneux, R. Heckendorn, and R. Meier, German Offen., 2,304,307 (1973); Chem. Abstr., 79 126535c (1973).
7. A. Gagneux, R. Heckendorn, and R. Meier, German Offen., 2,304,307 (1973); Chem. Abstr., 79 126535c (1973).
8. D. L. Coffen, R. I. Fryer, D. A. Katonak and F. Wong, J. Org. Chem., 40, 894 (1975).
9. N. W. Gillman and R. I. Fryer, J. Heterocyclic Chem., 14, 1171 (1977); R. B. Moffett, G. N. Evenson, and P. F. Von Voigtander, J. Heterocyclic Chem., 14, 1231 (1977), I. R. Ager, G. W. Danswan, D. R. Harrison, D. P. Kay, P. D. Kennewell, and J. B. Taylor, J. Med. Chem., 20, 1035 (1977); T. Hara, Y. Kayama, T. Mori, K. Itoh, H. Fujimori, T. Sunami, Y. Hashimoto, and S. Ishimoti, J. Heterocyclic Chem., 21, 263 (1978); G. W. H. Cheseman and S. G. Greenberg, J. Heterocyclic Chem., 16, 241 (1979).
10. N. W. Gillman and R. I. Fryer, J. Heterocyclic Chem., 14, 1171 (1977); R. B. Moffett, G. N. Evenson, and P. F. Von Voigtander, J. Heterocyclic Chem., 14, 1231 (1977), I. R. Ager, G. W. Danswan, D. R. Harrison, D. P. Kay, P. D. Kennewell, and J. B. Taylor, J. Med. Chem., 20, 1035 (1977); T. Hara, Y. Kayama, T. Mori, K. Itoh, H. Fujimori, T. Sunami, Y. Hashimoto, and S. Ishimoti, J. Heterocyclic Chem., 21, 263 (1978); G. W. H. Cheseman and S. G. Greenberg, J. Heterocyclic Chem., 16, 241 (1979).
11. N. W. Gillman and R. I. Fryer, J. Heterocyclic Chem., 14, 1171 (1977); R. B. Moffett, G. N. Evenson, and P. F. Von Voigtander, J. Heterocyclic Chem., 14, 1231 (1977), I. R. Ager, G. W. Danswan, D. R. Harrison, D. P. Kay, P. D. Kennewell, and J. B. Taylor, J. Med. Chem., 20, 1035 (1977); T. Hara, Y. Kayama, T. Mori, K. Itoh, H. Fujimori, T. Sunami, Y. Hashimoto, and S. Ishimoti, J. Heterocyclic Chem., 21, 263 (1978); G. W. H. Cheseman and S. G. Greenberg, J. Heterocyclic Chem., 16, 241 (1979).
12. N. W. Gillman and R. I. Fryer, J. Heterocyclic Chem., 14, 1171 (1977); R. B. Moffett, G. N. Evenson, and P. F. Von Voigtander, J. Heterocyclic Chem., 14, 1231 (1977), I. R. Ager, G. W. Danswan, D. R. Harrison, D. P. Kay, P. D. Kennewell, and J. B. Taylor, J. Med. Chem., 20, 1035 (1977); T. Hara, Y. Kayama, T. Mori, K. Itoh, H. Fujimori, T. Sunami, Y. Hashimoto, and S. Ishimoti, J. Heterocyclic Chem., 21, 263 (1978); G. W. H. Cheseman and S. G. Greenberg, J. Heterocyclic Chem., 16, 241 (1979).
13. N. W. Gillman and R. I. Fryer, J. Heterocyclic Chem., 14, 1171 (1977); R. B. Moffett, G. N. Evenson, and P. F. Von Voigtander, J. Heterocyclic Chem., 14, 1231 (1977), I. R. Ager, G. W. Danswan, D. R. Harrison, D. P. Kay, P. D. Kennewell, and J. B. Taylor, J. Med. Chem., 20, 1035 (1977); T. Hara, Y. Kayama, T. Mori, K. Itoh, H. Fujimori, T. Sunami, Y. Hashimoto, and S. Ishimoti, J. Heterocyclic Chem., 21, 263 (1978); G. W. H. Cheseman and S. G. Greenberg, J. Heterocyclic Chem., 16, 241 (1979).
14. J. B. Hester, D. J. Duchamp, and C. G. Chidester, Tetrahedron Letters, 1609 (1971).
15. R. Madronero and S. Vega, J. Heterocyclic Chem., 15, 1127 (1978);
16. P. C. Wade, B. R. Vogt, B. Toeplitz, M. S. Puar, and J. Z. Gougoutas, J. Org. Chem., 44, 88 (1979);
17. E. Aiello, G. Dattolo, G. Cirrincione, S. Plecia, and G. Daidone, J. Heterocyclic Chem., 16, 209 (1979).
18. A. Chimirri, S. Grasso, R. Ottana, G. Romero and M. Zappala, J. Heterocyclic Chem., 27, 371 (1990).
19. E. Cortés and A. M. Mendoza, J. Heterocyclic Chem., 33, 1159 (1996).
20. C. B. de Sarro, M. Zappala, S. Grasso, A. Chimirri, C. Spagnolo, and A. de Sarro, Mol. Neuropharmacol., 1, 195 (1992).
21. E. Cortés, R. Martínez, M. Ugalde and N. Maldonado, J. Heterocyclic Chem., 28, 365 (1991).
22. K.-C. Liu, B. R. Shelton and R. K. Howe, J. Org. Chem., 45, 3916 (1980).
23. E. Cortés and L. A. Araluce, J. Heterocyclic Chem., 34, 745 (1997)