Synthesis and 11C-radiolabelling of a tropane derivative lacking the 2β ester group: A potential pet-tracer for the dopamine transporter

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 42, Issue 5, 1999, Pages 447-456

  Schönbächler, Roland ^a   Ametamey, Simon M ^a   Schubiger, Pius A ^a  

^a PAUL SCHERRER INSTITUTE   (Switzerland)

Author keywords

Dopamine transporter; PET; CPPIT

Indexed keywords

ALKYLATION; NEUROPHYSIOLOGY; PHASE INTERFACES;

DOPAMINE TRANSPORTERS; ESTER GROUPS; GAS-PHASE REACTIONS; METHYL IODIDE; N-METHYLATION; PET TRACER; RADIOCHEMICAL YIELD; RADIOLABELLING; REACTION SEQUENCES; Β-CPPIT;

AMINES;

CARBON 11; COCAINE; DOPAMINE TRANSPORTER; ESTER; IODINE; METHANE; METHYL IODIDE; TROPANE DERIVATIVE;

ARTICLE; BLOOD BRAIN BARRIER; CHEMICAL REACTION; DIFFUSION; DRUG ACTIVITY; DRUG SYNTHESIS; HUMAN; ISOTOPE LABELING; METHYLATION; POSITRON EMISSION TOMOGRAPHY; TIME;

EID: 0032897811     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199905)42:5<447::AID-JLCR204>3.0.CO;2-9     Document Type: Article

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